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1-(4-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}piperidin-1-yl)ethan-1-one
N-(1-benzylpyrrolidin-3-yl)-1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-(propan-2-yl)-1H-pyrazole-4-carboxamide
5-{[2-(2,1,3-benzoxadiazol-4-yl)-1H-imidazol-1-yl]methyl}thiophene-2-carboxylic acid
4-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-2-phenylmorpholine
3-{2-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
4-fluoro-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)benzene-1-sulfonamide
1-phenyl-4-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]butane-1,4-dione
5-methyl-N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-(1-{1-[(5-acetylthiophen-3-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methylbenzamide
(1R,5R)-6-benzyl-3-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-1,3,6-trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[3-(furan-2-yl)benzoyl]-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
N-cyclopropyl-3-hydroxy-N-(naphthalen-1-ylmethyl)propanamide
5-cyclobutanecarbonyl-1'-(pyridin-4-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
methyl[(2-methylpyridin-4-yl)methyl]{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}amine
methyl 6-[(4-ethoxyphenyl)methyl]-2-[ethyl(2-methylprop-2-en-1-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-(2-chloro-6-fluoro-3-methylbenzoyl)-1-(3-methoxyphenyl)piperazin-2-one
1-{1-[2-(2-chloro-6-fluorophenyl)acetyl]piperidin-4-yl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
5-(2,6-difluorophenoxymethyl)-N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-1,2-oxazole-3-carboxamide
N-(5-{[(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)carbamoyl]amino}-2-methylphenyl)cyclopentanecarboxamide
ethyl 1-[(2H-1,3-benzodioxol-5-yl)carbamoyl]-3-benzylpiperidine-3-carboxylate
N-ethyl-8-methyl-2-(2-methylpyrimidin-5-yl)-N-(pentan-2-yl)quinoline-4-carboxamide
4,6-dimethyl-2-oxo-N-[1-(piperidin-1-ylmethyl)cyclohexyl]-1,2,3,4-tetrahydropyrimidine-5-carboxamide
8-methoxy-4-methyl-2-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}quinoline
3-{[8-(2-methoxyethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]methyl}benzonitrile
2-(cyclohexylmethyl)-4-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]morpholine
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-1-(4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidin-1-yl)propan-1-one
(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-6-[3-(prop-2-en-1-yloxy)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
(4aR,7aS)-1-benzyl-4-(1-methyl-1H-imidazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(2-propyl-1H-1,3-benzodiazol-1-yl)-1-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]propan-1-one
3-({[(3,4-dimethylphenyl)methyl]amino}methyl)-3-hydroxy-1-(2-phenylethyl)piperidin-2-one
5-methyl-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)-1,3,4-oxadiazol-2-amine
2-(2-hydroxyphenoxy)-1-[3-(2-methylphenoxymethyl)piperidin-1-yl]ethan-1-one
N-[(3R,4S)-4-cyclopropyl-1-(oxan-4-yl)pyrrolidin-3-yl]-2-(2,5-dioxoimidazolidin-1-yl)acetamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-1-phenyl-1H-1,2,3-triazole-5-carboxamide
2-(5,6-dimethoxy-1-oxo-1,2-dihydroisoquinolin-2-yl)-N-(1,4-dioxan-2-ylmethyl)-N-methylacetamide
4-cyclopropyl-6-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}pyrimidine
2-cyclopropyl-4-hydroxy-N-[(2-methylphenyl)(pyridin-4-yl)methyl]pyrimidine-5-carboxamide
3-(2-amino-1,3-thiazol-4-yl)-1-[3-(4-fluorophenoxymethyl)piperidin-1-yl]propan-1-one
1-(4-{2-[(3S)-3-(dimethylamino)azepan-1-yl]-2-oxoethoxy}phenyl)propan-1-one
1-{[4-(pyridin-3-yl)phenyl]methyl}-4-(pyridin-3-ylmethyl)-1,4-diazepane
3-[3-(piperidine-1-carbonyl)phenyl]-1-[2-(pyridin-2-ylsulfanyl)ethyl]urea
5-(3-{[2-(4-methoxy-2,3-dimethylphenyl)-1H-imidazol-1-yl]methyl}phenyl)-1H-1,2,3,4-tetrazole
(3S,4R)-N,N-dimethyl-4-(propan-2-yl)-1-(quinoline-6-carbonyl)pyrrolidin-3-amine
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-[2-(pyridin-4-yl)-1,3-thiazole-4-carbonyl]pyrrolidin-3-yl]methanol
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-7-acetamido-2-(2-methoxyphenyl)-N,1-dimethyl-1H-1,3-benzodiazole-5-carboxamide
2-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
N,3,6-trimethyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
2-(5-{4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine-1-carbonyl}-1H-pyrazol-3-yl)phenol
N-[(3-fluorophenyl)methyl]-9-methoxy-3-(1-methylazepane-2-carbonyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide