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1-(cyclopropylmethyl)-5-[2-(2-methoxyphenoxy)acetyl]-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-(5-phenyl-1,2,4-oxadiazol-3-yl)pyrrolidin-3-yl]acetamide
({4-cyclopropyl-5-[1-(pyridin-4-ylmethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
3-{[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]methyl}pyridine
5-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-2-methoxyphenol
1-methyl-3-phenyl-4-{pyrazolo[1,5-a]pyrimidin-3-yl}-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
6-[(3-methoxyphenyl)methoxy]-1-(2-methylpropyl)-4-(1,2,3-thiadiazole-4-carbonyl)-1,4-diazepan-2-one
2-methoxy-5-{1-[(2-methylphenyl)methyl]-4-phenyl-1H-imidazol-5-yl}pyrimidine
[(2-methoxypyrimidin-5-yl)methyl](methyl)[1-(pyridin-3-yl)ethyl]amine
1-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-3-[(dimethylamino)methyl]piperidin-3-ol
3-methyl-1-[(3-methylphenyl)methyl]-5-[(2,2,3,3-tetrafluoropropoxy)methyl]-1H-1,2,4-triazole
N-{[4-(6-amino-4-methylpyridin-3-yl)phenyl]methyl}acetamide
6-ethoxy-4-methyl-2-{4-[4-(pyridin-2-ylmethyl)piperazin-1-yl]azepan-1-yl}quinazoline
(2,3-dihydro-1-benzofuran-5-ylmethyl)(ethyl)[2-(1H-pyrazol-1-yl)ethyl]amine
7-fluoro-N-{[3-(methylsulfanyl)phenyl]methyl}-2-oxo-1,2-dihydroquinoline-4-carboxamide
(3R,4R)-1-[6-ethyl-2-(piperidin-1-yl)pyrimidin-4-yl]-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
1-(4-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}piperazin-1-yl)ethan-1-one
8-[(3-methoxyphenyl)methyl]-1-(3-methylbutyl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-benzyl-4-[(1H-imidazol-2-ylmethyl)sulfamoyl]benzamide
2-[5-(4-methoxy-2-methylphenyl)-3-methyl-1H-1,2,4-triazol-1-yl]acetic acid
3-methyl-N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)-5,6-dihydro-1,4-dioxine-2-carboxamide
1-[2-(1-{[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethyl]pyrrolidin-2-one
N-(2-fluoro-5-methylphenyl)-3-{[(3R)-pyrrolidin-3-yl]sulfamoyl}benzamide
(2R,6R)-4-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-triene-6-carboxylic acid
N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N,1-dimethyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-{2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl}-3-(4-methyl-1,3-thiazol-5-yl)propanamide
N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
1-(4-fluorophenyl)-4-[9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]butane-1,4-dione
N-cyclopropyl-1-{1-[(2-fluorophenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
N-benzyl-3-{1-[(2E)-3-(1H-imidazol-4-yl)prop-2-enoyl]piperidin-4-yl}-N-methylpropanamide
1-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)-3-(1H-1,2,4-triazol-1-yl)propanamide
1-(4-{[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]methoxy}phenyl)propan-1-one
(1R,5R)-3-(6-methoxy-1-methyl-1H-indole-2-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane
(2S,4R)-1-[(2,6-dichloro-3,4-dimethoxyphenyl)methyl]-4-(dimethylamino)pyrrolidine-2-carboxylic acid
N-cyclooctyl-2-methylpyrimidine-5-carboxamide
1-[(2-methoxyphenyl)methyl]-6-oxo-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}piperidine-3-carboxamide
2-[2-(4-chloro-2-methylphenoxy)acetyl]-2,7-diazaspiro[4.5]decan-6-one
9-(2-amino-6-methylpyrimidin-4-yl)-2-cyclopropyl-2,9-diazaspiro[5.5]undecan-3-one
[4-(2-phenoxyethyl)-1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-4-yl]methanol
3-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)butane-1-sulfonamide
[(1-ethyl-1H-pyrazol-4-yl)methyl](methyl)[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]amine
2-methyl-8-[2-(phenylamino)pyrimidine-5-carbonyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
3-{[2-(piperidin-1-ylmethyl)-1,4-oxazepan-4-yl]methyl}pyridin-2-amine
5-{[({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)(propan-2-yl)amino]methyl}pyrrolidin-2-one
2-ethyl-9-(2-methylpyridin-4-yl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
N-(1,4-dioxan-2-ylmethyl)-5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
2-[(4-fluorophenyl)methyl]-4-[(2,4,5-trimethoxyphenyl)methyl]morpholine