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methyl 2-(3-methylphenyl)-2-[(thian-4-yl)amino]acetate
6-(piperidin-3-yl)-2-(4,5,6,7-tetrahydro-1-benzothiophen-3-yl)-3,4-dihydropyrimidin-4-one
(4-{5-[(3-methyl-1,2-oxazol-5-yl)methyl]-1,2,4-oxadiazol-3-yl}phenyl)methanol
2-{[3-(1H-pyrazol-5-yl)piperidin-1-yl]methyl}benzoic acid
methyl 2-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-sulfonyl}benzoate
1-[3-(3-{[methyl(1-methylpiperidin-4-yl)amino]methyl}phenoxymethyl)piperidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
2,6-dimethoxy-4-({[(2-methylphenyl)methyl](prop-2-en-1-yl)amino}methyl)phenol
2-amino-N-{2-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]ethyl}-5,6,7,8-tetrahydroquinazoline-4-carboxamide
1-[3-(aminomethyl)phenyl]-3-{2-[(trifluoromethyl)sulfanyl]ethyl}urea
3-(2,5-dioxoimidazolidin-4-yl)-N-[1-(3-methylphenyl)piperidin-4-yl]propanamide
2-fluoro-N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylbenzamide
N-[2-(4-methyl-1H-imidazol-2-yl)ethyl]-5-(4-methylphenyl)-1H-pyrazole-3-carboxamide
1-{1-[(4-hydroxy-3-methylphenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
N-[cyclopropyl(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
(2S,4S)-4-amino-1-(2,3-dimethyl-1H-indole-5-carbonyl)-N-methylpyrrolidine-2-carboxamide
2-[3-(2-hydroxyethyl)-4-[(4-methylphenyl)methyl]piperazin-1-yl]-6-methylpyridine-3-carbonitrile
2-[4-(2-amino-6-methylpyrimidin-4-yl)-1H-pyrazol-1-yl]-N-(1-cyclohexyl-1H-pyrazol-5-yl)acetamide
ethyl({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)[3-(1H-pyrazol-1-yl)propyl]amine
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyloxane-4-carboxamide
N-(furan-2-ylmethyl)-N-methyl-5-{[methyl(2-phenylethyl)amino]methyl}-1,2-oxazole-3-carboxamide
2-(2-chloro-6-methoxyphenyl)-5-fluoro-N-methylpyrimidin-4-amine
7-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}-2-oxa-7-azaspiro[4.5]decan-8-one
3-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-6-yl}-1-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]urea
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-[3-(methylsulfanyl)propyl]piperidine-3-carboxamide
N-[2-(2-ethylphenoxy)ethyl]-N,2-dimethyl-2,8-diazaspiro[4.5]decane-3-carboxamide
2-methyl-6-{2-[2-(pyridin-4-yl)-1H-imidazol-1-yl]propyl}pyridine
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-7-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}thian-4-amine
4-(4-methoxyphenyl)-N-methyl-4-oxo-N-[1-(2-phenylethyl)piperidin-3-yl]butanamide
7-(1,3-benzothiazol-2-yl)-4-[(4-ethoxyphenyl)methyl]-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(2-methoxyethoxy)piperidine
N-[6-(dimethylamino)-1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl]-2-(thiophen-2-yl)azetidine-1-carboxamide
6-{2-[3-(dimethylamino)propyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}pyridine-2-carboxylic acid
(1R,3S,5S)-8-{[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-8-azabicyclo[3.2.1]octan-3-ol
[(5-methylthiophen-2-yl)methyl](pyridin-4-ylmethyl)(1,3-thiazol-2-ylmethyl)amine
N-{[1-(dimethylamino)cyclohexyl]methyl}-5-ethylpyrimidin-2-amine
5-(4-benzylpiperidine-1-carbonyl)-1-(cyclohexylmethyl)-N,N-dimethyl-4-oxo-1,4-dihydropyridine-3-carboxamide
(4aS,7aR)-1-cycloheptanecarbonyl-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[7-chloro-2-(4-hydroxypiperidin-1-yl)quinolin-3-yl]methyl}-N-[2-(4-fluorophenyl)ethyl]-1,3-dimethyl-1H-pyrazole-5-carboxamide
5-propyl-N-{1-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
5-methoxy-2-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}-4H-pyran-4-one
3-[2-(1,2-oxazinan-2-yl)-2-oxoethyl]-4-[(3-phenoxyphenyl)methyl]piperazin-2-one
[(2S)-1-{5-[3-(trifluoromethyl)phenoxymethyl]-1H-pyrazole-3-carbonyl}pyrrolidin-2-yl]methanol
2-(2-methoxyphenyl)-1-[4-(1H-pyrazol-5-yl)phenyl]-1H-imidazole
4-methoxy-N-(2-{7-[(2,3,6-trifluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
N-{[2-(4-fluorophenyl)-6-methylquinolin-3-yl]methyl}cyclopropanamine
3-(2,3-dimethoxyphenyl)-1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}pyrrolidine
3-(4-chloro-2-methylbenzoyl)-1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidine
5-[methyl(2-phenylethyl)amino]-2-[2-(1H-1,2,4-triazol-1-yl)ethyl]-2,3-dihydropyridazin-3-one
4-{[4-(3-benzoylpiperidine-1-carbonyl)furan-2-yl]methyl}morpholine