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2,2-dimethyl-5-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]thiomorpholin-3-one
[(3-chloro-4-methoxyphenyl)methyl](methyl)[(3-methyl-1H-pyrazol-4-yl)methyl]amine
N-[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]-2-(6-oxo-1,6-dihydropyrimidin-5-yl)acetamide
5-(2,3-difluorobenzoyl)-3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
(1S,5R)-3-benzyl-6-[(3,4-dimethoxypyridin-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-2-(pyridin-4-yl)pyrimidine-5-carboxamide
6-(2-chlorophenyl)-N-methyl-N-(2-methylpropyl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)-2-(pyrrolidin-1-yl)ethan-1-one
N-[2-(4-methylpiperazin-1-yl)butyl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
1-(4-methoxybenzoyl)-4-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperazine
1-(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carbonyl)piperidin-4-ol
4-[1-(4-chlorophenyl)-1H-pyrazol-4-yl]-N-[(1-methylpyrrolidin-3-yl)methyl]pyrimidin-2-amine
N-(3-hydroxypropyl)-2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]acetamide
9-[(2,5-dimethylphenyl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(3-fluorophenoxymethyl)-N-[(4-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1,3-oxazole-4-carboxamide
1-(4-methoxyphenyl)-3-methyl-4-(pyrrolidine-1-carbonyl)piperazin-2-one
3-{[1-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-1H-1,2,3-triazol-4-yl]methyl}-2,3-dihydro-1,3-benzoxazol-2-one
6-methyl-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxamide
5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-2-(pyridin-4-yl)pyrimidine
({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)[2-(diethylamino)ethyl]methylamine
2-(3,4-dichlorophenyl)-4-(6-methylpyrimidin-4-yl)morpholine
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-(pyridin-3-ylmethoxy)-4-[(2,4,5-trimethoxyphenyl)methyl]-1,4-diazepan-2-one
methyl (2S,4R)-4-(dimethylamino)-1-(4-acetamidobenzenesulfonyl)pyrrolidine-2-carboxylate
[(3R,4R)-1-[(5-ethylpyridin-2-yl)methyl]-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
1-({1-[4-(propan-2-yl)phenyl]-1H-pyrazol-4-yl}methyl)piperidine-4-carbonitrile
N-(pyridin-2-ylmethyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
4-(4-{[3-(2-oxopyrrolidin-1-yl)propyl]amino}piperidin-1-yl)-N-(1-phenylethyl)benzamide
methyl 3-benzamido-6-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)thieno[2,3-b]pyridine-2-carboxylate
N-methyl-N-{3-[(4-methylphenyl)sulfanyl]propyl}-2-oxo-1,2-dihydroquinoline-4-carboxamide
5-[4-(2-methoxyethyl)piperazine-1-carbonyl]-N-(propan-2-yl)pyrimidin-2-amine
1'-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
1-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-(5-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
1-{4-[3-({[(5-chlorothiophen-2-yl)methyl]amino}methyl)pyridin-2-yl]piperazin-1-yl}ethan-1-one
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[2-(morpholin-4-yl)ethyl]benzamide
1-[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one
N-({4-[(2-chloroprop-2-en-1-yl)oxy]phenyl}methyl)-N-(pyridin-3-ylmethyl)acetamide
4-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}-5,6,7,8-tetrahydroquinazolin-2-amine
2-methoxy-5-{[4-(propan-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyrimidine
N-(3-benzamido-4-methoxyphenyl)-4-methyl-1,2,3-thiadiazole-5-carboxamide
N-[2-methyl-2-(morpholin-4-yl)propyl]-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
1-(2,3,5,6-tetramethylbenzoyl)piperidine-4-carboxylic acid
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine
4-{3-[2-(2,6-difluorophenyl)ethyl]piperidine-1-carbonyl}-1-methylpiperidine
3-[1-(2,6-dimethylpyrimidine-4-carbonyl)piperidin-4-yl]-N-[(4-fluorophenyl)methyl]propanamide
1-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
(3R,4R)-4-ethyl-1-(5-phenyl-1,2-oxazole-4-carbonyl)piperidine-3,4-diol
5-methanesulfonyl-2-methyl-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]pyrimidin-4-amine
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-{[methyl({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl})amino]methyl}-4H-chromen-4-one
N-[1-(3-fluoro-4-hydroxyphenyl)ethyl]-3,4-dimethyl-5-sulfamoylbenzamide