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{1-[1-(2-ethyl-4-methyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methanol
2-amino-1-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
N-(1-cycloheptylpiperidin-3-yl)-2-methylpyridine-3-carboxamide
(2S,4S)-1-benzyl-4-{[(3,4-difluorophenyl)methyl]amino}-N-[2-(2-fluorophenyl)ethyl]pyrrolidine-2-carboxamide
methyl 2-(ethylsulfamoyl)-6-[(4-methoxynaphthalen-1-yl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-{[4-(1H-imidazol-1-yl)phenyl]methyl}-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
N-(2-hydroxyethyl)-N-(1,3-thiazol-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-{2-[3-(trifluoromethyl)phenyl]ethyl}acetamide
2-acetyl-8-(2-methyl-2-phenylpropanoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-{2-[2-(3-phenyl-1,2-oxazol-5-yl)-1H-imidazol-1-yl]ethyl}pyridine
2-[4-(isoquinolin-5-ylmethyl)-1-(thiophen-3-ylmethyl)piperazin-2-yl]ethan-1-ol
2-{4-[1-(1,3-thiazole-4-carbonyl)pyrrolidin-3-yl]piperidin-1-yl}pyrimidine
N-methyl-4-(morpholine-4-carbonyl)-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]pyridin-2-amine
2-methyl-5-propyl-4-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
2-[4-(2H-1,3-benzodioxol-5-ylmethyl)-3-oxopiperazin-1-yl]pyridine-3-carboxamide
N-[(4-methoxyphenyl)methyl]-2-(2-oxo-1,2-dihydropyrimidin-1-yl)-N-(pyridin-2-ylmethyl)acetamide
N,6-dimethyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
4-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}-1-(2-methylpentyl)piperidine
3-[1-(5,6-dimethylpyridine-3-carbonyl)piperidin-3-yl]benzoic acid
1-[1-(2-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(1,2-oxazinan-2-yl)propan-1-one
3-[2-(2-fluorophenyl)acetyl]-9-methoxy-N-methyl-7-oxo-N-(1,3-thiazol-4-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-(2-methoxyphenyl)-1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]propan-1-one
4-[(2,6,6-trimethylcyclohex-1-en-1-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-[(2,6-difluorophenyl)methyl]-4-(oxolan-3-yl)-1H-1,2,3-triazole
(3S,4R)-1-[(2-cyclohexylpyrimidin-5-yl)methyl]-N,N-dimethyl-4-propylpyrrolidin-3-amine
methyl (2R)-2-({5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)propanoate
1-methyl-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]azepane-2-carboxamide
3-{4-[2-(pyridin-2-yl)pyrimidin-5-yl]-1H-1,2,3-triazol-1-yl}propane-1,2-diol
9-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1-methyl-1H,2H,3H,6H,7H,8H,9H-[1,4]oxazino[3,2-g]quinoline-2,7-dione
2-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]pyridine-3-carboxylic acid
2-cyclopropyl-9-[2-(4-methyl-1H-pyrazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(3-methoxyphenyl)-3-[1-(3-phenylprop-2-ynoyl)piperidin-4-yl]propanamide
7-fluoro-N-(2-methanesulfonylethyl)-3-methyl-1H-indole-2-carboxamide
(3S,4S)-4-cyclopropyl-1-[(dimethyl-1,2-oxazol-4-yl)methyl]pyrrolidine-3-carboxylic acid
1-cyclohexyl-6-hydroxy-4-(thiolan-3-yl)-1,4-diazepan-2-one
1-{[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
(2R,3R,6R)-3-phenyl-5-(1,3-thiazol-2-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-({4-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-6-methylpyrimidin-2-yl}amino)phenol
6-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidine
1-[4-(4-methoxybenzoyl)piperazin-1-yl]-3-(pyridin-2-yl)propan-1-one
N-[3-(4-hydroxyphenyl)propyl]-3-(1H-pyrazol-1-yl)benzamide
4-[5-({[(5-methylpyrazin-2-yl)methyl]amino}methyl)-1,2,4-oxadiazol-3-yl]benzoic acid
N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-(3-hydroxy-3-methylbut-1-yn-1-yl)benzamide
1-ethyl-N-(3-hydroxy-3-phenylpropyl)-N-methyl-2-oxo-1,2-dihydropyridine-4-carboxamide
methyl[(3-phenyl-1H-pyrazol-4-yl)methyl]{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
1-[(6-methoxypyridin-3-yl)methyl]-4-(pyrrolidine-1-sulfonyl)-1,4-diazepane
N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-(1,2-oxazinan-2-yl)propanamide
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}({1-[2-(1H-pyrazol-1-yl)phenyl]ethyl})amine
(2S,3R)-2-{[6-(4-ethylphenyl)imidazo[2,1-b][1,3]thiazol-3-yl]formamido}-3-hydroxybutanamide