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N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-5-phenyl-1,2-oxazole-3-carboxamide
N-[2-(azepan-1-yl)ethyl]-N-methyl-2,3-dihydro-1H-indene-1-carboxamide
(1R,7S)-N-methyl-3-[2-(4-methylphenyl)ethyl]-4-oxo-N-(pyridin-2-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-[5-(methoxymethyl)pyrazolo[1,5-a]pyrimidin-7-yl]-4-(thiophene-2-carbonyl)piperazine
1-[4-(4-{[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]amino}piperidin-1-yl)phenyl]pyrrolidin-2-one
3-(dimethyl-1,2-oxazol-4-yl)-1-[4-(thian-4-yl)piperazin-1-yl]propan-1-one
1-{3-[2-(pyridin-4-yl)pyridin-4-yl]pyrrolidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
N-methyl-N-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}oxan-4-amine
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-[(3-methoxyphenyl)methyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2R,6S)-2,6-dimethyl-4-{[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}morpholine
(4aR,8aR)-2-cyclobutanecarbonyl-7-{[4-(difluoromethoxy)phenyl]methyl}-decahydro-2,7-naphthyridin-4a-ol
4-methyl-2-[4-(4-methylpyrimidine-5-carbonyl)piperazin-1-yl]-6-(trifluoromethyl)pyrimidine
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-2-(1-methyl-1H-indol-3-yl)acetamide
7-(2-methoxyethyl)-2-(1-methyl-1H-pyrazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}thiophene-3-carboxamide
1-(cyclopropylmethyl)-5-(5-ethyl-1,2-oxazole-3-carbonyl)-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-2,3-dimethoxy-N-(oxolan-2-ylmethyl)benzamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-[(2-methylphenyl)sulfanyl]-N-[(1-methylpiperidin-3-yl)methyl]acetamide
2-({4-[(4-methylpiperazin-1-yl)methyl]piperidin-1-yl}methyl)quinoline
6-{3-[(4-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}-N,N-dimethylpyrazine-2-carboxamide
N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
3-(2-methyl-1H-indol-1-yl)-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}propanamide
1-[(3-methylthiophen-2-yl)methyl]-4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-[3-(prop-2-en-1-yloxy)benzoyl]piperidin-3-amine
1-{4-[3-(4-fluorophenoxy)propyl]piperazin-1-yl}-2-(morpholin-3-yl)ethan-1-one
{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]methylamine
1-{2-[(3S,4R)-3-cyclopropyl-4-[(pyrimidin-2-yl)amino]pyrrolidin-1-yl]-2-oxoethyl}piperidin-2-one
N-cyclohexyl-3-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)propanamide
2-[4-(1H-pyrazol-5-yl)phenyl]pyridine-3-carbonitrile
3-(2H-1,3-benzodioxole-5-carbonyl)-N-benzylpiperidine-1-carboxamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)acetamide
N-[(4-hydroxyphenyl)methyl]-N-(pyridin-3-ylmethyl)spiro[2.2]pentane-1-carboxamide
1-cyclobutyl-4-[4-(piperidine-1-carbonyl)phenoxy]piperidine
N,1-dibenzyl-N-(3-hydroxy-2-methylpropyl)-5-methyl-1H-1,2,3-triazole-4-carboxamide
1-[5-(4-aminoazepane-1-carbonyl)-2-methylphenyl]imidazolidin-2-one
{2-methyl-6-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]pyrimidin-4-yl}methanamine
2-{5-[4-(aminomethyl)phenyl]-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl}acetic acid
4-(hydroxymethyl)-1-[4-(1,3-oxazol-5-yl)benzenesulfonyl]azepan-4-ol
2-ethyl-8-[2-(2-hydroxyphenoxy)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
2-[1-(4-fluorophenyl)-1H-pyrazol-4-yl]-1H-1,3-benzodiazole-5-carbonitrile
3-(1-benzyl-3-methyl-1H-pyrazol-5-yl)-1-[(2S)-pyrrolidin-2-ylmethyl]urea
N-methyl-N-[2-(oxan-2-yl)ethyl]quinoxaline-6-carboxamide
N-{1-[1-(1-benzofuran-2-carbonyl)piperidin-4-yl]-2-phenylethyl}-N-methylpyridine-2-carboxamide
6-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N,N-dimethylpyrazine-2-carboxamide
4-[1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]-1-(2-methylbenzoyl)piperidine
2-(5-chloro-6-methyl-1-benzofuran-3-yl)-1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
5-(2-fluorophenyl)-N-{[1-(morpholin-4-yl)cycloheptyl]methyl}-1,2,4-triazin-3-amine
2-ethoxy-6-{[3-(2-hydroxyethyl)-4-[(3-methoxyphenyl)methyl]piperazin-1-yl]methyl}phenol
2-{1-[(2-fluorophenyl)methyl]-4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol