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N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-2,3-dimethylquinoxaline-6-carboxamide
1-{3-[3-(hydroxymethyl)piperidin-1-yl]propyl}-3-(2,4,5-trifluorophenyl)urea
1-({5-[1-(3-fluoropyridin-4-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)azepane
1-(2-{[(1-ethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-4-methylpyrimidin-5-yl)ethan-1-one
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
methyl 3-[2-oxo-6-(pyridin-4-ylmethoxy)-4-(quinoline-6-carbonyl)-1,4-diazepan-1-yl]propanoate
N,N-dimethyl-4-[(1E)-3-{4-[2-(oxolan-2-yl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}prop-1-en-1-yl]aniline
4-{4-[4-(2,4-dimethylphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-[1-(1,3-thiazol-2-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
4-methoxy-6-{3-[1-(2-methoxyethyl)-1H-pyrazol-3-yl]phenyl}pyrimidine
(3S,4R)-1-(benzenesulfonyl)-3-benzyl-4-methylpiperidin-4-ol
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N,3,5-trimethyl-1H-indole-2-carboxamide
N-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}methyl)-3-{imidazo[1,2-a]pyridin-2-yl}propanamide
(2S)-4-(methylsulfanyl)-2-{[2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}butan-1-ol
3-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-1-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]urea
1-[(2,6-difluorophenyl)methyl]-N-ethyl-N-[2-(pyrrolidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}methyl)-2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carboxamide
{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)amine
2-(2,4-dimethoxyphenyl)-3-(piperidine-1-carbonyl)pyridine
2-(furan-2-yl)-5-({2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}methyl)pyrimidine
2,3-dimethyl-6-(1-{thieno[3,2-d]pyrimidin-4-yl}piperidin-4-yl)-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
N-[(5-methyl-2-{3-[3-(pyridin-3-yl)propanamido]phenyl}-1,3-oxazol-4-yl)methyl]-2,3-dihydro-1,4-benzodioxine-6-carboxamide
5-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-9-carbonyl]-1,2-dihydropyridin-2-one
2-(3,4-dimethylphenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-1-yl]ethan-1-one
3-(1-benzofuran-2-yl)-4-{1H-imidazo[4,5-b]pyridin-2-yl}-1H-pyrazole
(2S,4S)-N-ethyl-4-[(6-ethyl-2-methylpyrimidin-4-yl)amino]-1-(pyridin-2-ylmethyl)pyrrolidine-2-carboxamide
(3aR,6aR)-2-(2-methyl-1H-pyrrole-3-carbonyl)-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-({[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}amino)butan-1-ol
(3aS,6aS)-2-cyclohexyl-5-[(4-methyl-1,3-thiazol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-methoxy-3-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]pyrazine
2-[2-(2H-1,3-benzodioxol-5-yloxy)acetyl]-2,7-diazaspiro[4.5]decan-6-one
{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}(thiophen-2-ylmethyl)amine
N-(2,3-dihydro-1H-inden-2-yl)-2-(methylamino)-N-propylpyridine-4-carboxamide
N-(3-hydroxypropyl)-N-[(5-methylthiophen-2-yl)methyl]-1,3-benzothiazole-6-carboxamide
2-(dimethylamino)-2-(2-methylphenyl)-1-[3-(pyridin-2-yl)azetidin-1-yl]ethan-1-one
4-(3,4-difluorobenzoyl)-1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidine
N-ethyl-2-(1H-indol-3-yl)-N-[(2E)-3-phenylprop-2-en-1-yl]acetamide
1-[3-(4-phenoxybenzoyl)piperidin-1-yl]ethan-1-one
2-[3-cyclopropyl-5-({[(3,5-dimethylphenyl)methyl]sulfanyl}methyl)-1H-1,2,4-triazol-1-yl]acetic acid
5-oxo-1-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrrolidine-3-carboxylic acid
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-8-[5-(trifluoromethyl)pyridin-2-yl]-1,8-diazaspiro[4.5]decane
(3aR,5R,6S,7aS)-2-(4-chloro-2-methoxybenzoyl)-octahydro-1H-isoindole-5,6-diol
4-(morpholin-4-yl)-N-[1-(3-phenylpropyl)piperidin-3-yl]benzamide
9-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
1,3-dimethyl-5-{2-oxo-2-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]ethyl}imidazolidine-2,4-dione
N-(1,2-oxazol-3-ylmethyl)-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
2,2-dimethyl-1-{4-[3-(1-methylpiperidin-2-yl)propanoyl]piperazin-1-yl}propan-1-one
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(4-methyl-1H-pyrazol-1-yl)propanamide
N2-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-N4-methylpyrimidine-2,4-diamine
2-methyl-3-[3-(naphthalene-2-carbonyl)piperidine-1-carbonyl]pyridine
1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-3-(2-fluorophenoxymethyl)piperidine