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(1R,5R)-6-(1-benzofuran-2-ylmethyl)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
7-methyl-2-(2-methyl-1-benzofuran-7-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-(1H-pyrazol-1-yl)butanamide
4-(cyclopropylmethyl)-1-[2-(2,5-difluorophenyl)acetyl]-1,4-diazepan-5-one
N'-(3-chloro-4-methylphenyl)-N-[2-(pyrrolidin-1-yl)ethyl]propanediamide
5-{[3-(azepane-1-carbonyl)-1,2-oxazol-5-yl]methoxy}-2-methyl-1,3-benzothiazole
1-{4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidin-1-yl}-2-(2-phenyl-1H-imidazol-1-yl)ethan-1-one
3-(2-cyclopentylethyl)-3,4-dihydropteridin-4-one
(1R,5R)-6-benzyl-3-[5-(methoxymethyl)thiophene-2-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
6-(piperidin-1-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]pyrimidin-4-amine
3-{[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]amino}-N-(pyridin-3-yl)propanamide
N-cyclopropyl-3-{[1-(3-methylpyridin-2-yl)propan-2-yl]sulfamoyl}benzamide
N-[(3S,4R)-1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
2-benzyl-8-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
N-(1H-imidazol-2-ylmethyl)-2-{[(3-methylthiophen-2-yl)methyl]amino}benzamide
2-(morpholin-4-yl)-3-{[3-(1H-pyrazol-5-yl)piperidin-1-yl]methyl}quinoline
N,2,6,8-tetramethyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]quinoline-4-carboxamide
(2S)-1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-4-methyl-2-phenylpiperazine
2-ethoxy-3-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine-1-carbonyl)pyridine
4-{2-[4-(methylsulfanyl)phenyl]acetyl}-1-(oxan-4-ylmethyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
6-[4-(2-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-[2-({4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}methyl)phenoxy]acetic acid
(1R,2S)-N1-butyl-N2-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]cyclohexane-1,2-dicarboxamide
N-(2-chlorophenyl)-4-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]morpholine-2-carboxamide
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-2-hydroxy-3-methylbutanamide
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetamide
N-[2-(diethylamino)ethyl]-5-(methoxymethyl)-N-methyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
2-[({1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}amino)methyl]-6,8-dimethylquinolin-4-ol
methyl 4-(5-{[4-(1,3-benzoxazol-2-yl)piperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
1-cyclobutanecarbonyl-N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]piperidine-4-carboxamide
N-methyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-5-propyl-1,3,4-oxadiazole-2-carboxamide
{2-[4-(2-methylphenyl)-1,4-diazepan-1-yl]-1,3-thiazol-4-yl}methanol
1-[3-(1,3-oxazol-5-yl)phenyl]-3-[1-(thian-4-yl)piperidin-4-yl]urea
7-methyl-2-[2-(2-oxoazepan-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
N-(2-fluoro-5-methylphenyl)-2-{[2-(4-hydroxypiperidin-1-yl)ethyl]amino}acetamide
N-(1-methoxypropan-2-yl)-15-methyl-13-oxo-9-(pyridin-3-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
N-[4-({[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]amino}methyl)phenyl]acetamide
6-[(prop-2-en-1-yl)amino]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
N-{[(3S,4S)-3-hydroxy-1-[(5-hydroxy-2-methoxyphenyl)methyl]piperidin-4-yl]methyl}pyrrolidine-1-carboxamide
3-{[1-(3-acetamidothiophene-2-carbonyl)pyrrolidin-3-yl]methyl}benzamide
ethyl 4-[2-(2-oxo-4-phenylpyrrolidin-1-yl)acetyl]piperazine-1-carboxylate
4-{4-[(2-hydroxyphenyl)methyl]piperazin-1-yl}-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
(4aR,7aS)-4-[(2-methoxyphenyl)methyl]-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
5-[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonane-7-carbonyl]-1,2-dihydropyridin-2-one
ethyl 4-[4-(6-carbamoylpyrazin-2-yl)piperazin-1-yl]piperidine-1-carboxylate
N-butyl-2-(2,6-dioxo-1,3-diazinan-1-yl)-N-[(5-methylthiophen-2-yl)methyl]acetamide
1-[1-(4-ethylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(pyrazin-2-yl)propan-1-one
1-[2-(3-fluorophenyl)ethyl]-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-6-oxopiperidine-3-carboxamide
6-methyl-N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)pyridazin-3-amine
1-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]-2-[2-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazole