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1-[(3S,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
(2R,3R)-3-(dimethylamino)-1'-(5-methoxyfuran-2-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
dimethyl(3-{2-[1-(6-methylpyridine-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)amine
2-[(3-methoxyphenyl)methyl]-8-(pyrazin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
(1S,2S)-2-{4-[(2,3-dimethoxyphenyl)methyl]piperazin-1-yl}cyclohexan-1-ol
1-(1,2,3,4-tetrahydronaphthalen-2-yl)-4-(1,3-thiazole-4-carbonyl)piperazine
1-methyl-3-{[6-oxo-4-(piperazin-1-yl)-1,6-dihydropyridazin-1-yl]methyl}-1,2-dihydroquinolin-2-one
2-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-N-(propan-2-yl)propanamide
5-{2-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-3,6-dimethyl-[1,2]oxazolo[5,4-d]pyrimidine
(4S)-1-(4-chloro-2-hydroxybenzoyl)-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
1-(cyclohexylmethyl)-N-methyl-6-oxo-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-3-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-N-{1-[(3-fluorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}acetamide
(2S,4S)-4-amino-1-{2-[3-chloro-2-oxo-5-(trifluoromethyl)-1,2-dihydropyridin-1-yl]acetyl}pyrrolidine-2-carboxylic acid
3-({4-[3-(4-fluorophenoxy)propyl]piperazin-1-yl}methyl)pyrrolidin-3-ol
(1,3-benzothiazol-2-ylmethyl)(methyl){4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}amine
2-[4-(hydroxymethyl)-4-(2-phenylethyl)piperidin-1-yl]pyridine-3-carbonitrile
2-{1-[(2-fluorophenyl)methyl]-4-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperazin-2-yl}ethan-1-ol
8-{[3-(pyridin-2-ylmethoxy)phenyl]methyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
5-{[3-(aminomethyl)pyrrolidin-1-yl]methyl}-N-benzylpyrimidin-2-amine
N-[2-(1-{[3-(trifluoromethoxy)phenyl]methyl}piperidin-2-yl)ethyl]acetamide
1-methyl-5-(4-phenylpiperidin-1-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-4-propylpyrimidine-5-carboxamide
1-[(5-{[2-(methoxymethyl)piperidin-1-yl]methyl}-2,4-dimethylphenyl)methyl]-4-methylpiperazine
N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
4-(1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}azetidin-3-yl)morpholine
1-{2-[(3-fluorophenyl)methyl]morpholin-4-yl}-2-(2-methoxyethoxy)ethan-1-one
2-{[4-(pyridin-4-yl)-1,4-diazepan-1-yl]methyl}pyridine-3-carboxylic acid
N-(2-phenylethyl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-4-carboxamide
(1R,4S)-1,7,7-trimethyl-4-[1-phenyl-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-2-oxabicyclo[2.2.1]heptan-3-one
3-amino-1-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}pyrrolidine-3-carboxylic acid
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}thian-4-amine
N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamide
(3S,4R)-1-[(2-methoxypyridin-3-yl)methyl]-4-(3-methylthiophen-2-yl)piperidin-3-ol
(1S,5R)-6-benzyl-3-[4-(1H-1,2,3,4-tetrazol-1-yl)butanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(cyclohexylmethyl)-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[4-(3-methylpyridin-4-yl)piperazin-1-yl]-4-(piperidin-1-yl)butan-1-one
1-(oxane-4-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
2-(2-chloro-4-fluorophenyl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}acetamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}({[3-(methylsulfanyl)phenyl]methyl})amine
1-(3-chlorophenyl)-4-(2-methoxy-5-methylbenzoyl)-5-methylpiperazin-2-one
N-[3-(4-fluorophenyl)phenyl]-1-[2-(1H-imidazol-2-yl)ethyl]piperidine-3-carboxamide
4-({[(5-methoxy-1H-indol-2-yl)methyl]amino}methyl)-2,6-dimethylphenyl acetate
1-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]cyclopropan-1-amine
dimethyl(3-{2-[1-(pyrazin-2-yl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)amine
2-[5-(methanesulfonylmethyl)pyridin-2-yl]-1-methyl-1H-indole
4-[1-(carbamoylmethyl)-1H-imidazol-2-yl]-N-cyclohexylpiperidine-1-carboxamide
N-(1-{1-[(2Z)-2-fluoro-3-phenylprop-2-enoyl]piperidin-4-yl}-2-phenylethyl)-N,1,3-trimethyl-1H-pyrazole-5-carboxamide