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5-{[benzyl(methyl)amino]methyl}-N-(dicyclopropylmethyl)-N-methyl-1,2-oxazole-3-carboxamide
1-[1-(1-ethyl-1H-1,3-benzodiazol-2-yl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]cyclopropane-1-carboxamide
3-(dimethyl-1,2-oxazol-4-yl)-N-{2-[(pyridin-3-yl)amino]ethyl}propanamide
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)naphthalene-1-carboxamide
5-(3-{[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}propyl)-1,3,4-thiadiazol-2-amine
ethyl 4-({[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}amino)piperidine-1-carboxylate
2-(3-hydroxypropyl)-9-[2-(3-methylphenoxy)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
(1R,5S)-8-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}-3,8-diazabicyclo[3.2.1]octane
7-chloro-2-({[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl)amino}methyl)-4H-pyrido[1,2-a]pyrimidin-4-one
1-(methoxymethyl)-N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}cyclobutane-1-carboxamide
2-(2-ethoxyphenyl)-4-{[2-(2-methoxyphenyl)pyrrolidin-1-yl]methyl}-5-methyl-1,3-oxazole
4-{[3-methyl-4-(propan-2-yl)piperazin-1-yl]methyl}-2-(propan-2-yl)pyrimidine
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}[4-(1H-indol-3-yl)butan-2-yl]amine
1-(2-{5-acetyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-oxoethyl)-1,2-dihydropyridin-2-one
1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]ethan-1-one
methyl 3-[1-(pyridin-2-ylmethyl)-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propanoate
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
N-cyclohexyl-2-ethyl-7-(2-methoxybenzamido)-1-methyl-1H-1,3-benzodiazole-5-carboxamide
methyl 2-[2-({4-[(2-methylphenyl)methyl]piperazin-1-yl}methyl)phenoxy]acetate
N-{2-[2-(cyclohex-1-en-1-yl)acetyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}-2-(2-fluorophenyl)acetamide
2-[(2E)-3-phenylprop-2-en-1-yl]-8-[2-(pyrrolidin-1-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
6-(4-methoxypiperidin-1-yl)-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
2-(4-{5-methylthieno[2,3-d]pyrimidin-4-yl}-1H-pyrazol-1-yl)-N-(2-propyl-2H-1,2,3-triazol-4-yl)acetamide
5-{[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-2-(methylsulfanyl)pyrimidine
4-[(1-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}pyrrolidin-3-yl)methyl]benzoic acid
1-(oxan-4-yl)-4-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}piperazine
N2,N2-dimethyl-N4-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-5,6,7,8-tetrahydroquinazoline-2,4-diamine
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
2-amino-8-[4-(3,4-dimethylphenoxy)phenyl]-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
2-({[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)-N-methylacetamide
N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}-2-(2-oxopyrrolidin-1-yl)acetamide
1-(1-{[1-(2-amino-9H-purin-6-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
5-[4-(4-methoxybutyl)piperazine-1-carbonyl]-2-phenylpyrimidin-4-ol
9-{[4-(benzyloxy)-2-hydroxyphenyl]methyl}-1,4,9-triazaspiro[5.5]undecan-5-one
1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-2-[2-(pyrrolidin-1-yl)ethyl]piperidine
N-{[6,7-dimethoxy-2-(3-methoxyphenyl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)thiophene-2-carboxamide
(1R,3S)-N1,N1,2,2,3-pentamethyl-N3-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)cyclopentane-1,3-dicarboxamide
2-[4-(3-cyanopyrazin-2-yl)piperazin-1-yl]-N-(1,3-thiazol-2-yl)propanamide
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
N-(1-cycloheptylpiperidin-3-yl)-3-fluoro-4-methoxybenzamide
1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-3-propoxypiperidine
N-(2-methoxyethyl)-2-(2-methyl-5-oxopyrrolidin-1-yl)-N-(thiophen-2-ylmethyl)acetamide
3-(3-fluoropyridin-4-yl)-N-propylbenzamide
6-[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-2,3,4,9-tetrahydro-1H-carbazole
methyl 4-{[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]methyl}thiophene-2-carboxylate
2-(3-cyclopropanecarbonyl-1H-indol-1-yl)-1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}ethan-1-one
5-(methoxymethyl)-N-{2-[2-(propan-2-yloxy)phenyl]ethyl}thiophene-2-carboxamide
[1-({1-[(trimethylpyrazin-2-yl)methyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]methanol
2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}acetamide
3-[(3S,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-fluorophenyl)urea