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1-[(5-methylfuran-2-yl)methyl]-N3-[1-(naphthalen-1-yl)ethyl]-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
3-{[methyl(pyridin-3-ylmethyl)amino]methyl}-N-(1-methyl-1H-indazol-5-yl)benzamide
1-(2-chloro-4-fluorobenzoyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
1-[(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinolin-2-yl]isoquinoline
4-(4-chlorophenyl)-1-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]butan-1-one
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-6-(methoxymethyl)-N,1-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1'-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
methyl (1S,3R,3aR,6aS)-5-ethyl-3-(oxan-4-yl)-4,6-dioxo-1-phenyl-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
3-methanesulfonyl-N-[(3R,4S)-4-(propan-2-yl)-1-(pyridin-2-ylmethyl)pyrrolidin-3-yl]propanamide
N-benzyl-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-cyclohexaneamido-N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-1-(2-methoxyethyl)-1H-1,3-benzodiazole-7-carboxamide
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-4-methylpyrimidin-2-amine
3-(2-chlorophenyl)-N-[(4-hydroxyazepan-4-yl)methyl]-5-methyl-1,2-oxazole-4-carboxamide
N-ethyl-N-(2-methylprop-2-en-1-yl)-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
2-{5-[(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)methyl]-3-methyl-1H-1,2,4-triazol-1-yl}ethan-1-ol
3-hydroxy-1-methyl-3-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}piperidin-2-one
1-[2-({[(4-fluorophenyl)methyl](methyl)amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
2-{6-[(2-methoxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidin-4-amine
10-methoxy-5-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
(1S,5R)-6-methyl-3-{2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]acetyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
[(3R,4S)-4-(morpholin-4-ylmethyl)-1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-3-yl]methanol
4-[4-(methylamino)-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl]-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
1-{1-[(5-chloro-2-hydroxyphenyl)methyl]piperidin-3-yl}-N-cyclopentyl-1H-1,2,3-triazole-4-carboxamide
N-[3-(cyclohexylsulfanyl)propyl]-3-(4-hydroxyphenyl)-1H-pyrazole-5-carboxamide
1-(1-benzothiophen-2-ylmethyl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
4-(1-ethyl-1H-imidazol-2-yl)-1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]piperidine
2-[4-({4-[2-(methylsulfanyl)propyl]-1H-1,2,3-triazol-1-yl}methyl)-1,3-thiazol-2-yl]pyrazine
(2R)-1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-cyclohexyl-2-hydroxyethan-1-one
N-tert-butyl-2-(4-{[3-(2-hydroxypropan-2-yl)piperidin-1-yl]methyl}phenoxy)acetamide
{1-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]-3-methylbutan-2-yl}dimethylamine
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(isoquinolin-5-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-N-[3-(1H-pyrazol-1-yl)propyl]piperidin-4-amine
N,4-dimethyl-1-(6-methyl-4-oxo-4H-pyran-2-carbonyl)piperidine-4-carboxamide
(4aR,7aS)-1-(3-methylbut-2-en-1-yl)-4-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
8-[2-(pyridin-4-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
4-(1-{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}piperidine-3-carbonyl)morpholine
N-{[6,7-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)oxolane-2-carboxamide
1-[(3-methoxyphenyl)methyl]-4-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperazin-2-one
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-6-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
5-{4-[(3-cyclopropyl-1H-pyrazol-5-yl)methyl]-6-hydroxy-1,4-diazepane-1-carbonyl}-2,3-dihydro-1H-pyrazol-3-one
1-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}-2-{5-[4-(prop-2-en-1-yloxy)phenyl]-2H-1,2,3,4-tetrazol-2-yl}ethan-1-one
propan-2-yl 7-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfamoyl]-1,2,3,4-tetrahydroisoquinoline-2-carboxylate
1-benzyl-8-(cyclohex-3-en-1-ylmethyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-methyl-4-{3-[1-(pyridin-3-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyridine
4-ethyl-1-methyl-3-({1-[(3R)-1,2,3,4-tetrahydroisoquinoline-3-carbonyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1,5-dimethyl-4-{[methyl({[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl})amino]methyl}-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
2-{1-[(4-ethylphenyl)methyl]-5-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-1,2,4-triazol-3-yl}acetamide
4-(5-methoxypyridin-3-yl)benzamide
(3R,4R)-4-amino-1-[4-methoxy-3-(morpholin-4-yl)benzoyl]piperidin-3-ol
1-(2-methyl-5-{2-methyl-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl}phenyl)imidazolidin-2-one