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2,3-difluoro-N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)benzamide
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-[(6-methylpyridin-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
6-(2,3-dihydro-1H-inden-2-yl)-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
3-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-N-(3-methoxypropyl)benzene-1-sulfonamide
2-(3-{[4-(pyridin-4-yl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
6-{[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperazin-2-yl}ethan-1-ol
(2S)-2-amino-3-hydroxy-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-3-phenylprop-2-yn-1-one
methyl N-{4-[4-chloro-3-(methylcarbamoyl)phenyl]phenyl}carbamate
3-methyl-8-{[5-(1-methyl-1H-1,3-benzodiazol-2-yl)furan-2-yl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(4-methoxyphenyl)methyl]-1-(5-oxopyrrolidine-2-carbonyl)piperidine-4-carboxamide
3-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-methyl-N-[2-(oxan-4-yl)ethyl]benzamide
2-{[methyl(2,2,6,6-tetramethylpiperidin-4-yl)amino]methyl}quinolin-8-ol
{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[(8-methoxyquinolin-5-yl)methyl]methylamine
1-methyl-3-(2-methylpropyl)-N-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]-1H-pyrazole-5-carboxamide
4-(2,4-dichlorophenyl)-6-methoxypyrimidine
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
5-cyclopropanecarbonyl-1'-(thiophen-2-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-phenyl-N-[4-(4-{[(4-phenyl-1,3-thiazol-5-yl)methyl]amino}piperidin-1-yl)phenyl]propanamide
N-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)-2-[4-(morpholin-4-yl)-6-oxo-1,6-dihydropyridazin-1-yl]acetamide
N-[(1R,2R,4S)-bicyclo[2.2.1]heptan-2-yl]-5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
2,5-dimethyl-3-{4-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}pyrazine
2-[2-ethoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]-3-methoxypyrazine
N-(2-{[3-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]methyl}quinolin-6-yl)acetamide
2-(4-methyl-1H-1,3-benzodiazol-2-yl)-N-(1-propyl-1H-1,2,3-triazol-4-yl)pyrrolidine-1-carboxamide
2-{7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}pyridine-3-carboxamide
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1H-pyrazole-3-carboxamide
3-(2-fluorophenyl)-N-(furan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-1H-pyrazole-5-carboxamide
1-{4-[(2,2-dimethylmorpholin-4-yl)methyl]phenoxy}-3-(4-methylpiperazin-1-yl)propan-2-ol
1-(4-{1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-1H-pyrazole-4-carbonyl}piperazin-1-yl)ethan-1-one
4-[1-(2-methoxyphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]butanamide
5-(2-chloro-4-methoxyphenoxymethyl)-N-[2-(cyclohex-1-en-1-yl)ethyl]-1,2-oxazole-3-carboxamide
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-2-(2-methylphenoxy)ethan-1-one
2-[4-(dimethylamino)phenyl]-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-[(3R,4S)-1-(carbamoylmethyl)-4-cyclopropylpyrrolidin-3-yl]-6-methoxy-2,3-dihydro-1H-indene-5-carboxamide
(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-2-(1H-pyrazole-3-carbonyl)-decahydroisoquinoline
3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepin-3-yl)butan-1-one
{3-[(2-methylphenyl)methyl]-1-[1-(2-phenylethyl)piperidin-4-yl]piperidin-3-yl}methanol
2-(2-methoxyethoxy)-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
1-[4-(4-methoxyphenoxy)piperidin-1-yl]-2-(morpholin-4-yl)butan-1-one
6-(2-chlorophenyl)-7-(cyclopropylmethyl)-N-ethyl-8-oxo-N-propyl-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-(8-chloroquinolin-5-yl)-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane-4-carboxamide
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)[2-(pyridin-4-yl)ethyl]amine
4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}butanamide
N-{[1-(1H-indol-2-ylmethyl)pyrrolidin-3-yl]methyl}-2-methoxy-2-methylpropanamide
1-methyl-5-[methyl(thiophen-3-ylmethyl)amino]-N-[2-(piperidin-1-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5-(methoxymethyl)-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
N-[(2-chloropyridin-3-yl)methyl]-N-methyl-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
5-[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione