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4-[(1-cyclopropyl-1H-imidazol-2-yl)methyl]-1-methyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
3-[(3-cyclopropyl-1H-1,2,4-triazol-5-yl)methyl]-4,6-dimethyl-2,3-dihydro-1H-indol-2-one
2-(4-{[4-(2-methylphenyl)phenyl]methyl}-1-(1-methylpiperidin-4-yl)piperazin-2-yl)ethan-1-ol
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(methylamino)pyridine-4-carboxamide
1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-3-(3-methoxypropyl)piperidine
N-methyl-5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]-N-[2-(oxan-4-yl)ethyl]pyridin-2-amine
N-[2-(dimethylamino)ethyl]-5-methoxy-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)furan-2-carboxamide
2-(4-methyl-1H-pyrazol-1-yl)-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}propanamide
1-(3-chloro-4-methoxyphenyl)-N-[2-(ethylsulfanyl)ethyl]-5-oxopyrrolidine-3-carboxamide
3-[(2R,3R,6R)-5-(4-methylbenzoyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
(2S,4R)-1-benzyl-4-{[(4-methoxy-2,5-dimethylphenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
3-(4-methyl-1H-pyrazol-1-yl)-1-[(1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
2-(2,4-difluorophenyl)-5-(thiolan-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
6,7-dimethoxy-2-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}-1,2,3,4-tetrahydroisoquinoline
methyl 4-[4-(1H-indole-6-carbonyl)piperazin-1-yl]benzoate
N-cyclopropyl-3-[1-({4-[methyl(phenyl)amino]phenyl}methyl)piperidin-3-yl]propanamide
5-{4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}pyrimidine
(3S,4S)-4-[(dimethylamino)methyl]-1-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-3-ol
1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-(2-{2-[(2-chlorophenyl)methyl]morpholin-4-yl}-2-oxoethyl)-1,2,3-oxadiazol-3-ium-5-olate
2-({3-[4-(2,5-difluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-6-methoxyphenol
(3S,4S)-1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-(naphthalen-2-yl)piperidin-3-ol
3-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N-(propan-2-yl)propanamide
2-[({1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}oxy)methyl]pyridine
2-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)acetamide
N-[(3R,4S)-4-cyclopropyl-1-(pyridazin-3-yl)pyrrolidin-3-yl]-2-(3-methyl-2,5-dioxoimidazolidin-1-yl)acetamide
N-methyl-2-[methyl({[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl})amino]propanamide
1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
N-(5-methanesulfonamido-2-methylphenyl)-3-(3-methylphenoxy)azetidine-1-carboxamide
1-cyclopropyl-4-{4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}pyrrolidin-2-one
N-({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)cyclopentanecarboxamide
4-{[2-(3-methylphenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}morpholine-2-carboxamide
N4-[(5,6-dimethylpyridin-3-yl)methyl]-N2-(2-methoxyethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
2-{4-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]piperidin-1-yl}pyrimidine
6-{[2-(pyridin-4-yl)ethyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-2-methylbenzamide
2-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}-N-(pyridin-2-ylmethyl)acetamide
4-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl}pyrrolidin-2-one
1-methyl-2-(2-{2-[2-(propan-2-yl)pyrimidin-4-yl]-1H-imidazol-1-yl}ethyl)-1H-1,3-benzodiazole
7-(piperidin-3-ylmethyl)-N-[2-(1H-pyrazol-4-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-({3-benzyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-3-methyl-5-phenyl-1,2-oxazole
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(2-methoxyethyl){[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amine
N-[(4-cyanophenyl)methyl]-6-ethyl-1,5-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-(4-{[3-(2-hydroxyethyl)-4-[(5-methylfuran-2-yl)methyl]piperazin-1-yl]methyl}thiophen-2-yl)ethan-1-one
N4-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)-N2,6-dimethylpyrimidine-2,4-diamine
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(6-methoxypyrimidin-4-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(4-fluorophenyl)-1-{[2-(2-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
N-[(1-cyclopropanecarbonylpiperidin-3-yl)methyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
2-(furan-2-yl)-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzoyl]azepane
2-(3-acetyl-1H-indol-1-yl)-N-(pyridin-3-ylmethyl)butanamide