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6-[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidine-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(dimethyl-1,3-thiazol-5-yl)-N-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}acetamide
3-(4-cyclohexylphenyl)-1-{2-[(pyridin-3-yl)amino]ethyl}urea
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-1-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}propan-1-one
2-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]thiophene-3-sulfonamide
5-ethyl-N-{3-[(pyridin-3-yl)amino]propyl}-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
11-(morpholin-4-yl)-4-{[3-(trifluoromethyl)phenyl]methyl}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
7-(5-chloropyridin-2-yl)-4-[(3-ethyl-1H-pyrazol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[7-(3,6-dimethylpyrazin-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
1-ethyl-N-[(4-fluorophenyl)methyl]-7-methyl-4-oxo-N-(prop-2-en-1-yl)-1,4-dihydro-1,8-naphthyridine-3-carboxamide
N-{[1-(1,3-thiazole-5-carbonyl)piperidin-3-yl]methyl}naphthalene-1-carboxamide
N-({1-[(3-acetylphenyl)methyl]piperidin-3-yl}methyl)thiophene-2-carboxamide
4-[2-(1-benzyl-3-oxopiperazin-2-yl)acetyl]-1,4-diazepan-2-one
N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}-2,3-dihydro-1-benzofuran-5-carboxamide
5-(2-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-2-oxoethyl)-2,6-dimethyl-3,4-dihydropyrimidin-4-one
6-(2-methylpropyl)-4-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1,2-dihydropyrimidin-2-one
4-{3-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]phenyl}-4H-1,2,4-triazole
1,3-dimethyl-5-({[4-(1H-pyrazol-1-yl)butan-2-yl]amino}methyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
5-cyclopropanecarbonyl-1'-(pyridine-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-butyl-N-[(4-fluorophenyl)methyl]-2-(pyrrolidin-1-yl)propanamide
1-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(furan-2-carbonyl)-1,4-diazepane
1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{3-[(6-hydroxy-6-methylheptan-2-yl)amino]butyl}phenol
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carboxamide
(3aS,6aR)-5-(3-chloropyridin-2-yl)-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-{[1-(ethoxymethyl)cyclobutyl]methyl}-1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-4-amine
(1R,2R,6S,7S)-4-(2-methoxypyridine-4-carbonyl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane
N-butyl-N-(furan-2-ylmethyl)-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-[2-({[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]amino}methyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]ethan-1-one
4-[4-(benzyloxy)piperidine-1-carbonyl]-1-cyclopentylpyrrolidin-2-one
2-(4-cyclopropanecarbonylpiperazin-1-yl)-4-(propan-2-yl)-6-(trifluoromethyl)pyrimidine
5-[(4-hydroxypiperidin-1-yl)methyl]-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1,2-oxazole-3-carboxamide
6-(6-methoxypyridin-3-yl)-N2-(4-methylphenyl)-1,3,5-triazine-2,4-diamine
4-methyl-1-{4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}pentan-1-one
2-methylpropyl 4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.5]undecane-9-carboxylate
N-cyclopentyl-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}-5-methylthiophene-2-carboxamide
1-methyl-1'-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-N,4-dimethyl-1H-imidazole-2-carboxamide
N-(1-methoxypropan-2-yl)-5-methyl-4-{[3-(2-oxopyrrolidin-1-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
1-(3,4-dihydro-2H-1,4-benzoxazin-4-yl)-2-{2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}ethan-1-one
ethyl 2-[3-oxo-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-8-yl]propanoate
N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-2,3-dihydro-1-benzothiophene-2-carboxamide
(2S,4R)-4-[(adamantan-2-yl)amino]-1-[(4-chlorophenyl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
(3S,4S)-4-cyclopropyl-1-(1H-indole-6-carbonyl)pyrrolidine-3-carboxylic acid
3-{[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}imidazolidine-2,4-dione
N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-1-(propan-2-yl)piperidine-4-carboxamide
8-methoxy-2-{[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]methyl}quinoline
N-(3-hydroxy-3-phenylpropyl)-N-methyl-3-(1-methylpiperidin-4-yl)propanamide
6-[methyl(pyridin-3-ylmethyl)amino]-N-[2-(1-methylpiperidin-2-yl)ethyl]pyridine-3-carboxamide
1-{4-[4-(1-hydroxycyclopentyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-3-(1-methylpiperidin-4-yl)propan-1-one