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N-{3-[7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-3-oxopropyl}-N-methylmethanesulfonamide
5-cyclobutanecarbonyl-1'-(oxan-4-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
[2-(1-cyclopentylpiperidin-4-yl)ethyl](1-methoxypropan-2-yl)amine
2-(furan-2-ylmethyl)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane
(4aS,8aR)-6-(2-amino-4-methyl-1,3-thiazole-5-carbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
4-ethyl-1-methyl-3-({1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-methyl-4-{5-[3-(3-methylbutanoyl)piperidine-1-carbonyl]pyridin-2-yl}piperazin-2-one
N-cyclohexyl-N-(2-hydroxyethyl)-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
6-(2,5-dimethylfuran-3-yl)-2-(3-hydroxypiperidine-1-carbonyl)-7-methyl-7H,8H-imidazo[1,2-a]pyrazin-8-one
(2S,4S)-1-(5-acetylthiophene-3-carbonyl)-4-amino-N,N-diethylpyrrolidine-2-carboxamide
3-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1-(4-fluoro-2-methylphenyl)-3-(propan-2-yl)urea
2-(dimethyl-1,2-oxazol-4-yl)-N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)acetamide
3-[ethyl({[3-(5-methylfuran-2-yl)phenyl]methyl})amino]-1λ6-thiolane-1,1-dione
5-butyl-1-(3-chlorophenyl)-4-(4-methyl-1H-imidazole-2-carbonyl)piperazin-2-one
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-(2-methoxyacetyl)-N-[4-(3-methoxyphenyl)phenyl]piperidine-3-carboxamide
[5-({1-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]piperidin-4-yl}methyl)-4-methyl-4H-1,2,4-triazol-3-yl]methanol
N-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-3-(4-methylpiperazine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-(1,4-dioxan-2-ylmethyl)-2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
N-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
9-(5-ethyl-2-methylpyrimidin-4-yl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
(3aS,7aR)-5-methyl-2-[2-(2,2,3,3-tetrafluoropropoxy)acetyl]-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
2-methyl-1-[3-({2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-imidazol-1-yl}methyl)piperidin-1-yl]propan-1-one
methyl(propyl)[(5-{[4-(pyridin-3-yl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]amine
N'-(3-chloro-4-fluorophenyl)-N-(2-hydroxy-3-methoxypropyl)butanediamide
6-(morpholin-4-yl)-N4-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]pyrimidine-2,4-diamine
3-(2,5-dioxoimidazolidin-4-yl)-N-[(5-ethylpyridin-2-yl)methyl]-N-methylpropanamide
N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-decahydro-2,7-naphthyridine-2-carboxamide
(2S,4S)-4-amino-1-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)pyrrolidine-2-carboxylic acid
1-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N-(3-chloro-4-fluorophenyl)-N'-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N'-(pyridin-3-ylmethyl)propanediamide
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
6-methyl-3-{[methyl({[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl})amino]methyl}-1,2-dihydroquinolin-2-one
5-[5-(furan-3-yl)-1,2,4-oxadiazol-3-yl]-6-methyl-2-[(2S)-1-methylpyrrolidine-2-carbonyl]-1,2,3,4-tetrahydro-2,7-naphthyridine
1-{2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxybenzoyl}pyrrolidin-3-amine
2-[(5-methylpyrazin-2-yl)methyl]-9-(1H-pyrazole-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
3-hexyl-8-[(1s,4s)-4-hydroxycyclohexanecarbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(azepane-1-carbonyl)-5-(piperidin-1-yl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole
3-benzyl-4-{8-methylimidazo[1,2-a]pyridine-2-carbonyl}piperazin-2-one
3-(5-cyano-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl)-N-(5-cyclopropyl-1,3,4-thiadiazol-2-yl)propanamide
1-(4-{[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}phenyl)pyrrolidine
2-[(3S,4R)-4-amino-1-(5-tert-butyl-1,3,4-oxadiazol-2-yl)pyrrolidin-3-yl]ethan-1-ol
2-[5-(1,3-benzoxazol-2-yl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
5-(2,4-dichlorophenoxymethyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
3-methoxy-5-[2-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]pyridine
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-1-(propan-2-yl)piperidine-4-carboxamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-{methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}pyridine-3-carboxamide
N-[(2-methylphenyl)methyl]-2-[(1S,5R)-7-oxo-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-{imidazo[1,2-a]pyridin-3-yl}acetamide