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4-{4-[4-(2-methoxyphenyl)piperidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
2-methyl-5-[4-(oxolan-3-ylmethyl)piperazin-1-yl]-2,3-dihydropyridazin-3-one
[3-(prop-2-en-1-yl)-1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl]methanol
(isoquinolin-5-ylmethyl)(pyridin-3-ylmethyl)(thiophen-3-ylmethyl)amine
6-(3,4-diethoxybenzoyl)-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
1-[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-4-(pyridin-4-yl)-1,4-diazepane
2-methyl-8-[4-methyl-2-(piperidin-1-yl)pyrimidine-5-carbonyl]-2,8-diazaspiro[4.5]decane
1-[4-(2-methoxy-5-{[methyl(propan-2-yl)amino]methyl}phenoxy)piperidin-1-yl]pent-4-en-1-one
3-({[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)amino)propane-1,2-diol
N-ethyl-N-[2-(3-methylphenoxy)ethyl]-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
1-{2-[1-(4-methoxyphenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}piperidine
(4aS,8aR)-6-(1-benzofuran-5-ylmethyl)-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
2-[(3,5-difluorophenyl)methyl]-8-[2-(methylsulfanyl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
5-chloro-2-(4-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyrimidine
(2S,4R)-4-amino-N-ethyl-1-[3-(4-methylphenyl)benzoyl]pyrrolidine-2-carboxamide
[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](methyl){[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amine
N-{2-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)amino]ethyl}pyridine-3-carboxamide
2-({3-[(3-fluorophenyl)amino]piperidin-1-yl}methyl)-3-methoxyphenol
1-[3-(5-methylfuran-2-yl)butyl]-4-[(4-phenyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
N3-[(3-fluorophenyl)methyl]-N5-methyl-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
2-(4-{[5-(methoxymethyl)furan-2-yl]methyl}-1-[(2-methylphenyl)methyl]piperazin-2-yl)ethan-1-ol
(1R,3S)-3-amino-N-[(4-methoxyphenyl)methyl]-N-(pyridin-2-ylmethyl)cyclohexane-1-carboxamide
[3-(2-phenoxyethyl)-1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidin-3-yl]methanol
2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)-1-[(3S,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]ethan-1-one
5-acetyl-N-[2-(1,3-benzoxazol-2-ylsulfanyl)ethyl]-2,4-dimethyl-1H-pyrrole-3-carboxamide
2-butyl-8-[2-(morpholin-4-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
8-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
N-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)-3-(pyridin-4-yl)propanamide
6-cyclopentyl-1-methyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[1-(1H-imidazol-2-yl)ethyl]-1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-(2-phenyl-1H-imidazol-1-yl)ethan-1-one
methyl(quinolin-8-ylmethyl)[(3-{2-[1-(1,3-thiazole-5-carbonyl)piperidin-2-yl]ethoxy}phenyl)methyl]amine
(2S,4R)-4-amino-1-(4-phenylbutanoyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
(3E)-1-{3-methyl-3,9-diazaspiro[5.6]dodecan-9-yl}pent-3-en-1-one
2-phenyl-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-5,6,7,8-tetrahydroquinazolin-5-amine
1-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-3-propoxypiperidine
(2S)-2-[({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amino]propanamide
(3aS,6aS)-2-cyclopentanecarbonyl-5-(1,3-thiazol-2-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-{1-[(4-phenylbutan-2-yl)amino]ethyl}adamantan-1-ol
6-(aminomethyl)-2-methyl-N-[2-(4,5,6,7-tetrahydro-1H-indazol-3-yl)ethyl]pyrimidin-4-amine
3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]propanamide
3-(furan-2-yl)-1-[4-(2-methoxyphenoxy)piperidin-1-yl]propan-1-one
1-(2-fluoro-5-methanesulfonamidophenyl)-3-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}urea
N-[(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-3-yl)methyl]-1H-indazole-3-carboxamide
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-[5-(pyrimidin-5-yl)-1H-indol-1-yl]acetamide
1-[(3-carboxy-1H-pyrazol-4-yl)methyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-1-ethyl-5-oxopyrrolidine-3-carboxamide
1-(4-fluorophenyl)-2,2-dimethyl-N-[(5-methylpyrazin-2-yl)methyl]cyclopropane-1-carboxamide
(2S,4S)-4-amino-N,N-diethyl-1-(2-methoxyacetyl)pyrrolidine-2-carboxamide
2-ethoxy-4-(1-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1H-imidazol-2-yl)phenol