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5-hydroxy-6-(4-hydroxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-2-(4-methylphenyl)-2,3-dihydropyridazin-3-one
N-cyclopentyl-5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
6-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane-4-carbonyl}-2,3,4,5-tetrahydropyridazin-3-one
(3S,4S)-1-(benzenesulfonyl)-4-[(2-hydroxyethyl)(thiophen-2-ylmethyl)amino]pyrrolidin-3-ol
4-ethyl-3-[1-(3-methylquinolin-2-yl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-[2-(thiophen-2-yl)pyrimidine-5-carbonyl]-3,9-diazaspiro[5.6]dodecan-10-one
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-[2-(dimethylamino)acetyl]piperidine-4-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
(5-{[3-(2-chlorophenyl)pyrrolidin-1-yl]methyl}furan-2-yl)methanol
1-ethyl-4-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperazin-2-one
1-(4-methylpiperazin-1-yl)-3-{1-[3-(prop-2-en-1-yloxy)benzoyl]piperidin-3-yl}propan-1-one
3-(furan-2-yl)-2-[5-(1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]propanoic acid
N-(2,4-dimethoxyphenyl)-3-{1-[2-(methylsulfanyl)benzoyl]piperidin-4-yl}propanamide
N-ethyl-5-(3-fluorophenoxymethyl)-N-[(1-methylpyrrolidin-3-yl)methyl]-1H-pyrazole-3-carboxamide
4-{4-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methoxy]-3-methoxyphenyl}butan-2-one
ethyl 4-{[3-methyl-1-(pyridin-3-yl)butyl]amino}piperidine-1-carboxylate
ethyl 3-{[5-(2,5-dimethylphenoxymethyl)-1,2-oxazol-3-yl]formamido}-4-methylpentanoate
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(methylamino)pyridine-4-carboxamide
1-(2,4-dimethylphenyl)-5-[2-(ethanesulfinyl)ethyl]-3-(propan-2-yl)-1H-1,2,4-triazole
1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
4-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-4-yl}-5-(3-methylphenyl)-2-(pyridin-4-yl)pyrimidine
3-{[1-(hydroxymethyl)cyclopentyl]methyl}-3-methyl-1-{3-[(E)-2-(pyridin-2-yl)ethenyl]phenyl}urea
(3S,7S,8aS)-3-(4-aminobutyl)-7-{[(4-methylphenyl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
8-[2-(4-chlorophenoxy)ethyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-3-(3-hydroxyquinoxalin-2-yl)propanamide
2-[3-(pyrrolidine-1-carbonyl)piperazin-1-yl]quinoxaline
3-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-5-(2,6-difluorophenoxymethyl)-1,2-oxazole
N-[2-(1-cyclopentylpiperidin-4-yl)ethyl]pyrimidin-2-amine
2-[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]-5-(1H-1,2,3,4-tetrazol-1-yl)-1H-1,3-benzodiazole
2-[2-(3-phenoxyphenyl)-1H-imidazol-1-yl]ethan-1-ol
5-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridine-6-carbonyl]-1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole
1'-(2,5-dimethylfuran-3-carbonyl)-5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-chloro-N,N-dimethyl-5-{[3-(pyrrolidin-1-yl)piperidin-1-yl]methyl}-1,3-thiazol-2-amine
5-cyclopropyl-N-methyl-N-[(4-phenoxyphenyl)methyl]-1,3-oxazole-4-carboxamide
[(3R,5S)-5-(hydroxymethyl)-1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-3-yl]methanol
2-(cyclopent-2-en-1-yl)-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)acetamide
2-{3-[3-(pyrazin-2-yl)phenyl]-1H-pyrazol-1-yl}-N-(1,3-thiazol-2-yl)propanamide
7-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-oxa-7-azaspiro[4.5]decan-8-one
N-ethyl-N-[2-(4-methoxyphenoxy)ethyl]-2,6-dimethylpyrimidine-4-carboxamide
1-(2-{[(2-chloro-4-fluorophenyl)methyl](methyl)amino}ethyl)cyclopentan-1-ol
2-[6-(piperidin-1-yl)pyridin-3-yl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetic acid
1-[(3-chloro-2-fluorophenyl)methyl]-4-(hydroxymethyl)azepan-4-ol
5-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1-ethylpiperidin-2-one
3-hydroxy-1-(3-phenylpropyl)-3-[(propylamino)methyl]piperidin-2-one
N-[(2-chlorophenyl)methyl]-3-[1-(4,4,4-trifluorobutyl)piperidin-3-yl]propanamide
3,5-difluoro-2-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
2-{[2-(morpholin-4-ylmethyl)piperidin-1-yl]methyl}-1H-1,3-benzodiazole
N,N-dimethyl-4-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]piperazine-1-carboxamide
2-[(4-chlorophenyl)methyl]-N-(2-hydroxy-2-phenylethyl)-N-methyl-1,3-benzoxazole-5-carboxamide
N-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1-(morpholine-4-carbonyl)piperidin-4-amine