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N-[(3R,4R)-3-hydroxypiperidin-4-yl]-4-(2-methylphenyl)benzamide
2-(3-methylthiophen-2-yl)-4-(3,3,3-trifluoropropyl)pyrimidine
(1S,5R)-6-(cyclopropylmethyl)-3-{[3-(morpholin-4-yl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane
N-{4-[3-(methoxymethyl)pyrrolidine-1-carbonyl]phenyl}ethane-1-sulfonamide
4-[4-(pyrrolidin-1-ylmethyl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
N-{[7-(1,3-benzothiazol-2-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}oxolane-2-carboxamide
7-(furan-3-ylmethyl)-N-[2-(pyridin-4-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
[(4-ethyl-5-{1-[3-(trifluoromethyl)pyridin-2-yl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
N-cyclopropyl-3-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propanamide
5-[1-(2-aminoacetyl)pyrrolidin-2-yl]-N-(2-phenoxyethyl)thiophene-2-carboxamide
4-{[1-(3-methylfuran-2-carbonyl)piperidin-4-yl]oxy}-N-(2-phenylethyl)benzamide
(3-{2-[1-(3,5-difluoropyridine-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
5-cyclopentyl-3-({4-[5-(oxan-2-yl)furan-2-yl]-1H-1,2,3-triazol-1-yl}methyl)-1,2,4-oxadiazole
2-ethoxy-3-{5-methylthieno[2,3-d]pyrimidin-4-yl}pyridine
1-{1'-[(4-methyl-1H-imidazol-2-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
4-(4-chlorophenyl)-N-methyl-N-(quinoxalin-6-ylmethyl)butanamide
4-ethyl-3-[1-(5-phenyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(oxolan-3-yl)-5-[2-(1H-pyrazol-1-yl)phenyl]-1,2,4-oxadiazole
3-{1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl}-N-(2-fluorophenyl)propanamide
1-[2-fluoro-5-(4H-1,2,4-triazol-4-yl)phenyl]-3-[2-(N-methylmethanesulfonamido)ethyl]urea
N-[(1R,3R)-3-aminocyclopentyl]-2-(1-benzylpiperidin-4-yl)acetamide
5-[4-(difluoromethoxy)phenyl]-1-propyl-1H-1,2,4-triazole
N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
2-methyl-N-[(2-methylphenyl)methyl]-2,8-diazaspiro[4.5]decane-8-carboxamide
3-(3,5-dimethylphenyl)-N-[(3-methyl-1H-pyrazol-5-yl)methyl]propanamide
N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}cyclopentanamine
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,3-dimethoxybenzamide
methyl 3-cyclopropaneamido-6-{[4-(2-ethoxyphenyl)piperazin-1-yl]methyl}thieno[2,3-b]pyridine-2-carboxylate
N-[(3R,4S)-1-(carbamoylmethyl)-4-phenylpyrrolidin-3-yl]-2-(2-oxopiperidin-1-yl)acetamide
9-[4-(aminomethyl)benzoyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
2-chloro-4-({[3-(4-methyl-1H-pyrazol-1-yl)propyl]carbamoyl}amino)-N-(propan-2-yl)benzamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methylacetamide
2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]acetamide
5-benzoyl-1-(cyclopropylmethyl)-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(4-{6-hydroxy-4-[2-(1H-pyrazol-4-yl)ethyl]-1,4-diazepan-1-yl}piperidin-1-yl)ethan-1-one
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-(hydroxymethyl)furan-2-carboxamide
N-[(5-methyl-2-{3-[3-(pyridin-3-yl)propanamido]phenyl}-1,3-oxazol-4-yl)methyl]furan-3-carboxamide
2-(2-propyl-1,3-thiazole-4-carbonyl)-2,7-diazaspiro[4.5]decane
9-(4-chloro-3-fluorobenzoyl)-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
2-(1-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)ethan-1-ol
3-(1-methyl-1H-pyrazol-4-yl)-N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)propanamide
1-benzyl-N3-cyclopropyl-4-oxo-N5-[1-(thiophen-3-yl)propan-2-yl]-1,4-dihydropyridine-3,5-dicarboxamide
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-1-methyl-1H-pyrazole-4-carboxamide
2-[1-(2-methoxypyridine-3-carbonyl)-4-(pyrrolidin-1-ylmethyl)piperidin-4-yl]-5-methylpyridine
5-[(3,3-diphenylpiperidin-1-yl)methyl]-N-methyl-1,2,4-oxadiazole-3-carboxamide
4-(2-methyl-1H-imidazol-1-yl)-1-(4-methyl-1H-imidazole-5-carbonyl)piperidine-4-carboxylic acid
(2E)-N-{[6-(dimethylamino)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-N-(oxolan-2-ylmethyl)-3-(thiophen-2-yl)prop-2-enamide
4-(2-methylpropyl)-1-[1-(methylsulfanyl)propan-2-yl]-1,4-diazepan-5-one
(3S,4R)-4-(2-methylphenyl)-1-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}pyrrolidine-3-carboxylic acid
4-chloro-N,N-dimethyl-5-{[methyl({[4-(1H-pyrazol-1-yl)phenyl]methyl})amino]methyl}-1,3-thiazol-2-amine