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N-[3-(2-oxopyrrolidin-1-yl)propyl]-4-(1H-pyrazol-3-yl)benzamide
5-({4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl}methyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{2-[(benzylsulfamoyl)amino]ethyl}-3-methylpyridin-2-amine
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-5-(1H-pyrazol-1-ylmethyl)furan-2-carboxamide
N-[3-(1H-imidazol-1-yl)propyl]-N-(pyridin-3-ylmethyl)-2-(trimethyl-1H-pyrazol-1-yl)acetamide
5-[2-(benzenesulfonyl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
1-[(1S,5R)-6-(2-phenoxyethanesulfonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-ethyl-6-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)pyridine-3-carboxamide
4-{[1-cyclohexyl-5-(1H-1,2,3-triazol-1-ylmethyl)-1H-1,2,4-triazol-3-yl]methyl}-1-methylpiperidine
1-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-2-(pyrrolidin-1-yl)propan-1-one
5-(2-{3,9-diazaspiro[5.5]undecan-3-yl}-2-oxoethyl)-2-ethyl-6-methyl-3,4-dihydropyrimidin-4-one
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-2-methylpropanamide
(2R,6S)-4-[1-(4-chloro-2-fluorobenzoyl)piperidin-4-yl]-2,6-dimethylmorpholine
N-(1-benzyl-1H-pyrazol-3-yl)-2-[4-(6-methylpyridazin-3-yl)-1H-pyrazol-1-yl]acetamide
1-{2-[2-(3-methoxyphenyl)azetidin-1-yl]-2-oxoethyl}pyrrolidin-2-one
2-methyl-N-[2-(3-phenylpropoxy)phenyl]-3-(1H-1,2,4-triazol-1-yl)propanamide
N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-5-[(methylsulfanyl)methyl]furan-2-carboxamide
[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl](methyl)[2-(methylamino)ethyl]amine
N-[(3R,4S)-4-cyclopropyl-1-methanesulfonylpyrrolidin-3-yl]-4-phenylbutanamide
(3S)-N,N-dimethyl-1-[1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carbonyl]azepan-3-amine
3-(2-{7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
2-methoxy-1-[1'-(1-methyl-1H-pyrrole-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]-2-(4-methoxyphenoxymethyl)-1,3-oxazole
4-[(1R,5S,8S)-8-methoxy-3-azabicyclo[3.2.1]octane-3-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
(2S,4S)-1-[(3-chlorophenyl)methyl]-4-{[(2,4-dimethoxy-3-methylphenyl)methyl]amino}-N-[2-(2-fluorophenyl)ethyl]pyrrolidine-2-carboxamide
8-(3,6-dimethylpyrazin-2-yl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
N-benzyl-2-({[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-N-methyl-2,3-dihydro-1H-inden-2-amine
3-{[2-(3-fluorophenyl)-8-methoxy-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}-4H-chromen-4-one
3-(1-methyl-1H-imidazol-2-yl)-6-[4-(propan-2-yloxy)phenyl]pyridazine
ethyl 5-(cyclohex-3-en-1-ylmethyl)-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-5-[4-(trifluoromethyl)phenyl]-1,2,4-triazin-3-amine
7-(cyclobutylmethyl)-2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-2,7-diazaspiro[4.5]decane
6-[4-(cyclopropylamino)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl]-2,3-dihydropyridazin-3-one
2-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyrazine
3-(1-methyl-1H-pyrazol-4-yl)-1-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)propan-1-one
N-[(2S,4R,6S)-2-benzyl-6-[2-(methylamino)pyridin-3-yl]oxan-4-yl]acetamide
1-[2-(4-methoxyphenyl)ethyl]-4-[(6-methyl-2-propylpyrimidin-4-yl)amino]pyrrolidin-2-one
8-fluoro-2-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}quinoline
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-1H-1,2,3-benzotriazole-5-carboxamide
2-{2-[(6-methoxypyrimidin-4-yl)amino]ethyl}-1,2,3,4-tetrahydrophthalazine-1,4-dione
3-(1,4-diazepane-1-sulfonyl)-N-(1-phenylethyl)benzamide
1-{1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carbonyl}-N,N-diethylpyrrolidin-3-amine
3-(4-methanesulfonylphenyl)-6-methoxypyridazine
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-3-phenoxypropanamide
N-(2-methylphenyl)-3-{[5-(oxolan-2-yl)thiophen-2-yl]formamido}propanamide
(3S,5S)-N-(cyclohexylmethyl)-1-(2,3-dihydro-1H-inden-2-yl)-5-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)pyrrolidin-3-amine
(2S,4S)-4-amino-1-[(5-phenylthiophen-2-yl)methyl]pyrrolidine-2-carboxylic acid
N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-5-oxo-2,5-dihydro-1H-pyrazole-3-carboxamide
3-[1-(cyclohex-3-en-1-ylmethyl)-1H-pyrazol-5-yl]-1-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]urea
3-{3-[3-(piperidine-1-carbonyl)-5-(1,2,5-thiadiazole-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-1-yl]propyl}pyridine