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N-[2-(dimethylsulfamoyl)ethyl]-1-oxo-1,2-dihydroisoquinoline-4-carboxamide
(3S,4R)-4-phenyl-1-[3-(pyridin-2-yl)propanoyl]pyrrolidine-3-carboxylic acid
9-(2-amino-6-methylpyrimidin-4-yl)-2-(cyclopropylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-(2-butylpyrrolidine-1-carbonyl)-2-methoxyphenol
3-[1-methyl-5-(pyrrolidine-1-sulfonyl)-1H-1,3-benzodiazol-2-yl]-N-(oxolan-3-yl)propanamide
8-{[3-(furan-2-yl)phenyl]methyl}-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
3-[2-(4-ethylpiperazin-1-yl)ethyl]-8-(1-methylcyclopropanecarbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(2,1,3-benzothiadiazol-5-ylmethyl)-5-(2,6-dimethoxyphenyl)-1,2,4-triazin-3-amine
1-[(2-phenyl-1,3-thiazol-5-yl)methyl]-4-(thian-4-yl)piperazine
1'-(2,2-dimethyloxane-4-carbonyl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-(pyrrolidin-3-ylmethyl)piperidine-4-carboxamide
3-(3-hydroxy-3-methylbutyl)-N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)benzamide
(2S)-1-(3,5-dichloro-4-methylbenzoyl)-2-(methoxymethyl)pyrrolidine
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-2-(3-phenylpropyl)-1,3-benzoxazole-5-carboxamide
N-methyl-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
(but-2-yn-1-yl)({[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl})(furan-2-ylmethyl)amine
2-(3-phenylpropyl)-8-(pyridin-4-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
N-[(3-methylphenyl)methyl]-2,3-dioxo-N-(propan-2-yl)-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
3-(pyridin-4-yl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1H-pyrazole-5-carboxamide
3-(4-chlorophenyl)-1-(1,3-thiazol-4-ylmethyl)piperidine
methyl({[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl})(oxan-2-ylmethyl)amine
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-[3-(dimethylamino)propyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
N-{[4-(3-bromophenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl]methyl}-N-methylmethanesulfonamide
N-(3,4-difluorophenyl)-1-({4-[2-(pyrimidin-5-yl)ethynyl]phenyl}methyl)piperidin-3-amine
6-methyl-5-(prop-2-en-1-yl)-N4-{[4-(pyrrolidine-1-carbonyl)phenyl]methyl}pyrimidine-2,4-diamine
1-{4-[(furan-2-ylmethyl)sulfanyl]phenyl}-3-methyl-3-(thian-4-yl)urea
N-ethyl-5-(4-methanesulfonylphenyl)furan-2-carboxamide
N-[4-({4-[(2-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenyl]acetamide
2-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]acetic acid
1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-4-(prop-2-en-1-yl)-1,4-diazepan-5-one
3-[(1S,4S)-5-(2-methoxy-5-phenylphenyl)-6-oxo-2,5-diazabicyclo[2.2.1]heptan-2-yl]propanamide
5-fluoro-2-methoxy-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}benzamide
2-{[(5-ethylpyridin-2-yl)methyl](pyridin-2-ylmethyl)amino}butan-1-ol
N-{3-[6-(propan-2-yloxy)pyridazin-3-yl]phenyl}acetamide
3-methyl-6-{5-[(1S)-1-(1H-1,2,3,4-tetrazol-1-yl)ethyl]-1,2,4-oxadiazol-3-yl}pyridazine
4-ethyl-N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]benzamide
2-methanesulfonyl-1-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]ethan-1-one
4-[5-(3-methoxyphenyl)furan-2-carbonyl]-N,N-dimethylpiperazine-1-carboxamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-(5,6,7,8-tetrahydroquinoxalin-5-yl)acetamide
2-(5-acetylthiophen-3-yl)-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}acetamide
4-({[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}carbamoyl)pyridin-1-ium-1-olate
1-(diphenylmethyl)-N-methyl-N-(pyrazin-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-{1-[(1-benzylpyrrolidin-3-yl)methyl]-1H-imidazol-2-yl}-1-ethyl-1H-imidazole
3-(3-fluorophenoxymethyl)-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidine
2-(5-{[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]methyl}furan-2-yl)benzonitrile
3-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-1,1,1-trifluoropropan-2-ol
2-amino-4-methyl-N-{2-[2-(trifluoromethyl)phenyl]ethyl}-1,3-benzothiazole-6-carboxamide
1-{[1-(4-fluorophenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]methyl}-3-methyl-1H-pyrazol-5-amine
(2S,4S)-N-ethyl-4-(2-hydroxy-4-methoxybenzamido)-1-[(2E)-2-methylbut-2-en-1-yl]pyrrolidine-2-carboxamide
(3R,4R)-4-amino-1-[(2-cyclohexylpyrimidin-5-yl)methyl]piperidin-3-ol