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2-(3-fluorophenyl)-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1,3-benzoxazole-5-carboxamide
2-(4-ethylphenoxy)-1-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]ethan-1-one
N-(1H-imidazol-2-ylmethyl)-3-(3-methoxyphenyl)-N-methyl-1H-pyrazole-4-carboxamide
5,6-dimethyl-N-[1-(thiophene-2-carbonyl)piperidin-3-yl]pyridine-3-carboxamide
4-fluoro-2-{[2-(1-methyl-1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]methyl}phenol
7-methyl-3-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-3,7,11-triazaspiro[5.6]dodecan-12-one
2-benzyl-8-[2-(2-fluorophenyl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
1-ethyl-3-{3-[(2-fluorophenyl)methoxy]azetidine-1-carbonyl}-3-methylpiperidine
1-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)-4-(piperidine-1-sulfonyl)-1,4-diazepane
2-(1-benzyl-4-{[2-(naphthalen-1-yl)pyrimidin-5-yl]methyl}piperazin-2-yl)ethan-1-ol
9-[(1-methyl-1H-indol-2-yl)methyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]piperidin-3-amine
2,6-difluoro-N-[(3R,4S)-1-(3-hydroxypropyl)-4-propylpyrrolidin-3-yl]-3-methoxybenzamide
(3aR,6aR)-2-(cyclobutylmethyl)-5-[2-(3,5-difluorophenyl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[3-(4-fluorophenyl)oxolan-3-yl]-5-{1-methyl-1H-pyrazolo[1,5-a]imidazol-7-yl}-1,2,4-oxadiazole
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[2-(1H-indol-3-yl)ethyl]benzamide
4-[4-(benzenesulfonyl)phenyl]benzamide
2-ethoxy-1-{3-[2-(quinolin-6-yl)pyridin-4-yl]pyrrolidin-1-yl}ethan-1-one
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-(2-methoxyethyl)pyrrolidine-3-carboxylic acid
4-(4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-1-yl)-2-[1-(thiophen-2-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
N-(propan-2-yl)-1-[(1s,4s)-4-{[(2,4,5-trimethoxyphenyl)methyl]amino}cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1-(2-{2-[4-(propan-2-yl)phenyl]-1H-imidazol-1-yl}ethyl)-1H-1,2,3-triazole
(2S)-N2-(2-methylpropyl)-N2-(pyridin-4-ylmethyl)pyrrolidine-1,2-dicarboxamide
2-[(1S,5R)-6-(cyclopropylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N-[2-(4-fluorophenyl)ethyl]acetamide
(2R,6R)-4-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-{[5-(3-methoxyphenyl)-1,2-oxazol-3-yl]methyl}-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
1-[4-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazin-1-yl]ethan-1-one
N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-3-(2-methylphenyl)-3-phenylpropanamide
1-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-(1-methyl-1H-pyrrol-2-yl)propan-1-one
1,3-dimethyl-6-({5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-(3-methoxypropyl)piperidine-3-carboxylic acid
1-{4-[({[(1R,9aR)-1-hydroxy-octahydro-1H-quinolizin-1-yl]methyl}amino)methyl]phenyl}pyrrolidin-2-one
N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
[(3R,4R)-1-(4-fluorobenzoyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
1-(5-ethyl-1,3-oxazole-4-carbonyl)-4-[(3-fluorophenyl)methyl]piperazine
N-[(3R,4R)-3-hydroxy-1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidin-4-yl]pyrazine-2-carboxamide
N-(furan-3-ylmethyl)-1-(oxan-4-yl)piperidine-3-carboxamide
1-[(2E)-3-phenylprop-2-en-1-yl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N,N-dimethyl-2-[(4-oxo-4-phenylbutanamido)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
2-{2-[2-(4-fluorophenyl)azetidin-1-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
4-[4-(2-methylpyrrolidine-1-carbonyl)phenoxy]-1-(2-phenylethyl)piperidine
4-{1-[(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl]pyrrolidin-2-yl}-3,5-dimethyl-1,2-oxazole
5-[4-(1-hydroxy-3-phenylpropyl)piperidine-1-carbonyl]-2-methyl-3,4-dihydropyrimidin-4-one
1-[1-(1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidin-4-yl)ethyl]-4-methylpiperazine
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(thiophen-2-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
3-{[1-(hydroxymethyl)cyclobutyl]methyl}-3-methyl-1-(2,4,5-trifluorophenyl)urea
8-[(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)methyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-{[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]sulfonyl}benzonitrile
1-(1,4-dioxan-2-ylmethyl)-3-(3-fluorophenyl)urea
4-(1,3-benzothiazole-6-carbonyl)-1-butylpiperazin-2-one