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4-[(3-fluorophenyl)methyl]-1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-1,4-diazepan-5-one
2-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}-4-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidine
3-(1-{[1-(cyclohex-3-ene-1-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-1-ol
ethyl 1-benzyl-5-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-(5-amino-1H-1,2,4-triazol-3-yl)-1-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]propan-1-one
2-amino-4-[1-(propan-2-yl)-1H-pyrazol-4-yl]-5H,7H,8H-pyrano[4,3-b]pyridine-3-carbonitrile
1-cyclopentyl-N-[3-(3-methylphenyl)propyl]-5-oxopyrrolidine-3-carboxamide
3-({3-azaspiro[5.5]undecan-9-yl}amino)-N-(4-fluorophenyl)propanamide
2-[3-(3-chlorophenyl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
N-[(2S)-1-methoxypropan-2-yl]-3-[methyl(pyrazin-2-ylmethyl)sulfamoyl]benzamide
N-[4-(1-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-1H-1,2,3-triazol-4-yl)phenyl]acetamide
2-{4-[(2-chlorophenyl)methyl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
1-[1'-(quinoline-8-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-1-[3-(1H-pyrazol-1-yl)phenyl]piperidin-4-amine
N-ethyl-2-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-(2-ethylpyrimidine-5-carbonyl)pyrrolidin-3-yl]methanol
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-5-phenyl-1H-pyrrole-2-carboxamide
(1R,5R)-6-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}(methyl)[(2-methylpyridin-4-yl)methyl]amine
5-(2-methyloxolan-2-yl)-3-(2-phenylethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
4-({2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}methyl)phenol
4-(cyclopropylmethyl)-1-{2-[methyl(piperidin-4-yl)amino]acetyl}-3-(propan-2-yl)-1,4-diazepan-5-one
6-[8-(cyclopropylmethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-2-carbonitrile
1-[3-(2-ethoxyphenyl)propyl]-2-(oxolan-3-yl)-1H-imidazole
1-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)-4-(thiophen-2-ylmethyl)piperazine
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(3-chlorophenyl)methyl]-4-(cyclooctylamino)pyrrolidine-2-carboxamide
4-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}-1-(2-methyloxolane-2-carbonyl)piperidine
6-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-1-yl]-2,4-dimethylpyridine-3-carbonitrile
1-(2-methyl-1,3-thiazole-4-carbonyl)-4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidine
3-(1-methyl-1H-pyrazol-4-yl)-1-[3-(4-phenoxybenzoyl)piperidin-1-yl]propan-1-one
8-[(6-chloropyridin-3-yl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
5-[1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1H-1,2,3-triazol-4-yl]-3-(2-methoxyethyl)-1,2,4-oxadiazole
4-(dimethyl-1,2-oxazol-4-yl)-3-(1-methyl-5-oxopyrrolidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{2-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}cyclopentan-1-one
4-(3-fluorophenoxy)-1-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]piperidine
2,5-dioxo-6-{pyrazolo[1,5-a]pyridin-3-ylmethyl}-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
4-methyl-N-(1,2-oxazol-3-ylmethyl)-2-(pyridin-3-yl)pyrimidine-5-carboxamide
(3R,9aR)-3-[(1S)-1-hydroxyethyl]-8-{[3-(methylsulfanyl)phenyl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-[(6-fluoro-4-oxo-1,4-dihydroquinolin-2-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
3-{5-[3-(dimethylsulfamoyl)propyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
4-(3-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}phenyl)morpholine
3-methyl-3-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl}piperidine
3-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
N-[(2S,4R,6R)-2-(5-tert-butyl-1H-pyrazol-3-yl)-6-cyclohexyloxan-4-yl]acetamide
(2S)-2-[2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamido]propanamide
4-benzyl-3-[1-(pyridine-3-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
ethyl 4-[2-(4-benzyl-2-oxopyrrolidin-1-yl)acetyl]piperazine-1-carboxylate
(1R,5R)-6-(2-hydroxy-4-methylbenzoyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide