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1-[2-(4-methoxyphenyl)ethyl]-6-oxo-N-[3-(pyridin-4-yl)propyl]piperidine-3-carboxamide
9-{[5-(oxan-2-yl)furan-2-yl]methyl}-6-oxa-9-azaspiro[4.5]decane
2-{2-[4-phenyl-5-(3-phenyl-1,2,4-oxadiazol-5-yl)-1H-imidazol-1-yl]ethoxy}ethan-1-ol
3-{2-[4-(3-methylpyridin-2-yl)piperazin-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
5-({2-[(2-chlorophenyl)methyl]morpholin-4-yl}methyl)-2-hydroxybenzoic acid
methyl 3-{[(2-methylphenyl)formamido]methyl}-5-(quinoline-8-sulfonamido)benzoate
2-{4-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]morpholin-3-yl}acetic acid
1-(furan-2-yl)-2-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]ethane-1,2-dione
1-(1H-imidazol-4-ylmethyl)-N-[4-(3-methoxyphenyl)phenyl]pyrrolidine-2-carboxamide
1-(diethylamino)-3-[2-methoxy-4-({[2-(pyrazin-2-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
ethyl 1-(2-hydroxy-6-methylpyridine-3-carbonyl)-3-(3-phenylpropyl)piperidine-3-carboxylate
3-({2-[3-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}methyl)-1,2,4-oxadiazole-5-carboxamide
4-(6-ethylpyrimidin-4-yl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-[(3R,4S)-1-{6-methylthieno[2,3-d]pyrimidin-4-yl}-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
1-(1,3-benzothiazol-2-ylmethyl)-1-methyl-3-(trimethyl-1H-pyrazol-4-yl)urea
ethyl 1-[(3-acetylphenyl)methyl]-4-[(2-chlorophenyl)methyl]piperidine-4-carboxylate
8-methyl-5-{[(2R)-2-methylpiperazin-1-yl]methyl}quinoline
1-{1-[(2,4-dimethylphenyl)methyl]piperidin-3-yl}-N-(2-hydroxyethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
2-[1-(3-methylphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetamide
(1R,7S)-6-(4-ethylpiperazine-1-carbonyl)-3-(2-phenoxyethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
1-(2-ethoxyethyl)-4-phenyl-5-[5-(1H-pyrazol-5-yl)thiophen-2-yl]-1H-imidazole
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-{[1-(pyrimidin-4-yl)ethyl]sulfamoyl}benzamide
3-phenyl-3-({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propan-1-ol
1-{[1-(morpholin-4-yl)cyclohexyl]methyl}-5-{2-[(pyridin-3-ylmethyl)amino]ethyl}pyrrolidin-2-one
N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-3,5-dimethyl-1H-indole-2-carboxamide
8-[(4Z)-hept-4-en-1-yl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
(4aR,7aS)-1-benzyl-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[1-(1-methylpiperidine-2-carbonyl)azetidin-3-yl]pyridine
(4aS,8aR)-1-(2-aminoethyl)-6-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-decahydro-1,6-naphthyridin-2-one
1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-8-(pyrimidin-2-yl)-1,8-diazaspiro[4.5]decane
7-(2-amino-3-cyclopentylpropanoyl)-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(1R,5R)-6-(cyclobutylmethyl)-3-[4-(pyrrolidin-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
1-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-5-oxopyrrolidine-3-carboxylic acid
3-[5-(1-acetylpiperidin-4-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-N-cyclopropylpropanamide
N-[2-(dimethylsulfamoyl)ethyl]-2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
3-(1-methyl-1H-imidazole-2-carbonyl)-1-(1-methyl-1H-pyrrole-2-carbonyl)piperidine
methyl (2S)-1-(1-{2-[(2-chlorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-3-carbonyl)pyrrolidine-2-carboxylate
5-[1-(4-methyl-1,3-oxazole-5-carbonyl)piperidin-4-yl]-5-(3-methylbutyl)-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
1-(4-{1-[(5-methylfuran-2-yl)methyl]-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenyl)-1H-imidazole
1-{imidazo[1,2-a]pyridine-3-carbonyl}-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-methanesulfonyl-1,5-diazatricyclo[5.2.2.02,6]undecane
1-{3-[4-(1H-pyrrole-2-carbonyl)piperazine-1-carbonyl]piperidin-1-yl}propan-1-one
5-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
4-(2-methoxy-5-methylphenyl)-5-methylthieno[2,3-d]pyrimidine
2-{1-[3-(morpholin-4-yl)propyl]-1H-1,2,3-triazol-4-yl}-1H-1,3-benzodiazole
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(oxan-4-ylmethyl)acetamide
1-[(5-chlorofuran-2-yl)methyl]-N-methylpyrrolidine-3-carboxamide
3-[2-(3-fluorophenyl)ethyl]-1-(prop-2-ene-1-sulfonyl)piperidine
2-methyl-5-(3-{[(2-methyl-5-propylpyrimidin-4-yl)amino]methyl}pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
5-acetyl-N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N,2,4-trimethyl-1H-pyrrole-3-carboxamide