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1-[3-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
1-{2-oxo-2-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]ethyl}imidazolidine-2,4-dione
N-cyclopropyl-2-{[6-(2-fluorophenyl)imidazo[2,1-b][1,3]thiazol-3-yl]formamido}acetamide
5-({3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}methyl)isoquinoline
4-ethyl-3-methyl-5-({2-[5-(1-methyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}sulfanyl)-4H-1,2,4-triazole
2-(4-methoxy-2-methylphenyl)-2-[4-(pyridin-4-yl)piperazin-1-yl]acetic acid
1-[2-(difluoromethoxy)benzoyl]-4-(2-methylpyridin-4-yl)-1,4-diazepane
(2E)-1-[4-(4-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}phenoxy)piperidin-1-yl]-3-(thiophen-2-yl)prop-2-en-1-one
N-{[7-(1,3-benzothiazol-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-5-(methoxymethyl)furan-2-carboxamide
(1R,5R)-3-methanesulfonyl-6-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
1-[2-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)ethyl]-2-methyl-1H-indole
3-(1,3-benzothiazol-2-yl)-1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
2-(furan-2-yl)-N-methyl-N-(pyrazin-2-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-[(1S,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]-3,6-dimethyl-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline
ethyl 4-benzyl-1-[(4-hydroxyquinolin-2-yl)methyl]piperidine-4-carboxylate
(1R,3S)-3-(2-aminoethoxy)-7-(4-chloro-1H-pyrazole-3-carbonyl)-7-azaspiro[3.5]nonan-1-ol
5-acetyl-N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
(4aR,7aS)-1-cyclobutanecarbonyl-4-(3-methyl-1H-pyrazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(4-fluorophenyl)-1-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}-1,2,3,6-tetrahydropyridine
2-({[(3R,4R)-1-[(2,6-dimethylphenyl)methyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
2-(3-fluorophenyl)-N-[1-(3-methylpyridin-2-yl)propan-2-yl]-1,3-benzoxazole-5-carboxamide
N-[(2-fluorophenyl)methyl]-3-{1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]piperidin-3-yl}propanamide
N-{[2-(4-acetylpiperazin-1-yl)-5,8-dimethoxyquinolin-3-yl]methyl}-3-methyl-N-(oxolan-2-ylmethyl)thiophene-2-carboxamide
N-(2-hydroxyethyl)-6,6-dimethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-5-oxothiomorpholine-3-carboxamide
1,3,6-trimethyl-5-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{2-[4-(methoxymethyl)piperidin-1-yl]-4-(morpholin-4-yl)pyrimidin-5-yl}-2-methylpropanoic acid
N-cyclopentyl-N-[(5-methylthiophen-2-yl)methyl]-3-(1H-1,2,4-triazol-1-yl)propanamide
(3R,5S)-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
1-{1-[2-(1H-indazol-3-yl)acetyl]-1,2,3,6-tetrahydropyridin-4-yl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-[(5-acetylthiophen-3-yl)methyl]piperidine-3-carbonitrile
4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperidine
(3S,4S)-1-(4-cyclopentylpyrimidin-2-yl)-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
1-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
{[2-(4-cyclohexylpiperazine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}(2-methoxyethyl)(propan-2-yl)amine
N-butyl-2-(cyclopropylmethyl)-4-oxo-1,3,8-triazaspiro[4.5]dec-1-ene-8-carboxamide
1-[3-({3-[(3-chlorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}methyl)phenyl]ethan-1-one
N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-2-(1-propylpiperidin-4-yl)acetamide
2-[4-(4-cyclopentylpyrimidin-2-yl)-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl]ethan-1-ol
5-acetyl-N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}thiophene-2-carboxamide
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-1-[4-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
N-[3-(6-methyl-1,3-benzoxazol-2-yl)propyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-[(3R,4R)-3-hydroxy-1-(2-methylquinolin-4-yl)piperidin-4-yl]pyrazine-2-carboxamide
2-(adamantan-1-yl)-N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-4-hydroxypyrimidine-5-carboxamide
(3S,4S)-1-(benzenesulfonyl)-4-[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]pyrrolidin-3-ol
3-[1-(1,1-dioxo-1λ6-thian-4-yl)piperidin-4-yl]-1-(2-ethylphenyl)urea
4-[1-benzyl-5-(cyclopropylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
(3R,4R)-1-(2-ethoxy-5-methylbenzenesulfonyl)-3,4-dimethylpyrrolidin-3-ol
N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-5-(2-fluorophenoxymethyl)-N-methyl-1H-pyrazole-3-carboxamide
2-(pyridin-2-yl)-N-[1-(thiophen-3-yl)propan-2-yl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine