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N-methyl-N-[2-(pyrrolidin-1-yl)ethyl]-5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,2-oxazole-3-carboxamide
1-(2-methoxyethyl)-3-(2-methylphenyl)-3-{2-oxo-2-[4-(pyridin-4-ylmethyl)piperazin-1-yl]ethyl}pyrrolidine-2,5-dione
4-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-methyl-1-(2-methylpropyl)piperazin-2-one
4-[(1S,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]-7,8-dimethyl-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline
3-{[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}pyridine
3-fluoro-4-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
(1-{2-[(6,7-dimethoxy-4-methylquinolin-2-yl)amino]ethyl}piperidin-3-yl)methanol
N-[(3S,7S,8aS)-3-[(1R)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]naphthalene-2-carboxamide
2-[(4aR,7aS)-4-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
7-[(3-methoxyphenyl)methyl]-6-oxo-N-(prop-2-en-1-yl)-2,7-diazaspiro[4.5]decane-2-carboxamide
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methylpropyl)acetamide
methyl 4-{[3-(2-hydroxyethyl)-4-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-1-yl]methyl}benzoate
2-chloro-6-methoxy-4-{[methyl({[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}phenol
2-(1-methyl-1H-pyrazol-4-yl)-5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridine
1-[9-methoxy-7-(8-methoxy-4-methylquinolin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(3,4,5-trimethoxyphenyl)ethan-1-one
4-{[4-methyl-5-({[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}sulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine
2-[4-(3-methoxypyrazin-2-yl)-1-(3-phenylpropyl)piperazin-2-yl]ethan-1-ol
3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-4-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}-1H-pyrazole
4-(4-chlorophenoxy)-N-[(3-fluorophenyl)methyl]piperidine-4-carboxamide
2,3-dimethyl-N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]quinoxaline-6-carboxamide
8-(2-hydroxybenzoyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
3-({4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)phenol
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-2-(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
4-[2-(2-oxoimidazolidin-1-yl)ethyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methyl-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
5-{3-[2-(2,4-difluorophenyl)ethyl]piperidine-1-carbonyl}-2-(propan-2-yl)-3,4-dihydropyrimidin-4-one
methyl 3-[(2E)-3-(3-fluorophenyl)prop-2-enamido]-6-{[(furan-2-ylmethyl)(methyl)amino]methyl}thieno[2,3-b]pyridine-2-carboxylate
(1-{[2-(naphthalen-1-yl)pyrimidin-5-yl]methyl}pyrrolidin-3-yl)methanamine
N-(2-{[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]methyl}quinolin-5-yl)acetamide
3-{[7-(2-methyl-1,3-thiazole-4-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}pyridine
[(3S,5R)-1-[(3-phenyl-1,2-oxazol-5-yl)methyl]-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
(1S,5R)-N6-(3,4-difluorophenyl)-N3,N3-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3,6-dicarboxamide
2-[(5-methylpyrazin-2-yl)methyl]-8-(1,3-thiazol-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
4-{1,3,6-trimethyl-1H-pyrazolo[3,4-b]pyridine-4-carbonyl}piperazine-2-carboxylic acid
(2S,4R)-4-amino-N-ethyl-1-(2-methoxypyridine-4-carbonyl)pyrrolidine-2-carboxamide
4-[2-amino-3-cyano-6-(5-methylpyridin-2-yl)pyridin-4-yl]benzamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
9-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}-3-oxa-9-azaspiro[5.5]undecane
7-[(2,3-difluorophenyl)methyl]-2-(2-methylpropanoyl)-2,7-diazaspiro[4.5]decan-6-one
8-(1,3-benzothiazol-2-ylmethyl)-3-(2-methoxyethyl)-1-[2-(4-methoxyphenyl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methyl-N-[(5-phenyl-1H-pyrazol-3-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
(2-{methyl[(2-phenyl-1,3-thiazol-4-yl)methyl]amino}-1,3-thiazol-4-yl)methanol
8-methyl-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(4-chlorophenyl)ethyl]-2-(1H-imidazol-2-yl)benzamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(4-propylpyrimidine-5-carbonyl)piperidin-3-ol
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperazine
1-[4-(1,3-benzoxazol-2-yl)piperazin-1-yl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
4-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-9-methoxy-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-2-(propan-2-yl)-1,3-thiazole
5-acetyl-N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]thiophene-2-carboxamide