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1-(3-{[1-methyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}propyl)pyrrolidin-2-one
1-benzyl-N-ethyl-5-[methyl(2-methylpropyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-4-ol
2-[(3-aminopyrrolidin-1-yl)methyl]-6-fluoroquinolin-4-ol
N-[2-(6-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
1-methyl-4-(1-{1-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperidin-4-yl}piperidine-3-carbonyl)piperazine
4-amino-N-[(1-benzyl-1H-pyrazol-4-yl)methyl]pyridine-2-carboxamide
4-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-1-(4-methoxyphenyl)-3-methylpiperazin-2-one
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-(methoxymethyl)furan-2-carboxamide
4-[(4aS,8aR)-decahydroisoquinolin-2-yl]-N-[3-(1H-imidazol-1-yl)propyl]pyridine-2-carboxamide
4-chloro-N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-2-hydroxybenzamide
(3S,4S)-1-(2-hydroxypyridine-3-carbonyl)-4-propylpyrrolidine-3-carboxylic acid
1-{3-oxo-3-[2-(2-phenylethyl)morpholin-4-yl]propyl}piperidin-2-one
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-methyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-{[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-3,5-dimethyl-1-(propan-2-yl)-1H-pyrazole
(5S)-5-[({[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(pyridin-2-ylmethyl)amino)methyl]pyrrolidin-2-one
2-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}benzonitrile
N-[(2-fluorophenyl)methyl]-3-[1-(4-phenylbutanoyl)piperidin-3-yl]propanamide
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methoxyethyl)-N-(propan-2-yl)acetamide
6-methyl-2-[(2-{[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)amino]-3,4-dihydropyrimidin-4-one
7-hydroxy-6-methoxy-4-[5-(1H-pyrazol-3-yl)thiophen-2-yl]-1,2,3,4-tetrahydroquinolin-2-one
2-ethyl-4-({4-[(3-methylphenyl)methyl]piperazin-1-yl}methyl)pyrimidine
N-methyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
(1R,9aR)-1-(2,6-difluorophenoxymethyl)-octahydro-1H-quinolizine
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
3-[2-(4-ethylpiperazin-1-yl)ethyl]-8-(oxolan-3-ylmethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(1S,5R)-3-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(2-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}-1H-pyrrol-1-yl)pyrimidine
2-{[4-(8-methoxyquinolin-5-yl)phenyl]sulfanyl}acetamide
2-{4-[(2-methyl-1,3-thiazol-5-yl)methyl]-1-[(4-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-2-phenyl-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N-(1-benzothiophen-2-ylmethyl)-2-methoxy-N,2-dimethylpropanamide
3-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyridin-2-ol
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-5-phenyl-1,2-oxazole-3-carboxamide
3-[2-(4-fluorophenyl)ethyl]-1-(4-methyl-1,3-thiazole-5-carbonyl)piperidine
3-chloro-4-{[1-(4-hydroxy-4-methylpentan-2-yl)piperidin-4-yl]oxy}-N-(2-methoxyethyl)benzamide
1-(5-propylpyrimidin-4-yl)-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}piperidin-4-amine
2-(2,3-difluorophenyl)-1-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-1H-imidazole
N-[(1-propyl-1H-pyrazol-4-yl)methyl]-3-sulfamoylbenzamide
1-[(4-methoxyphenyl)methyl]-4-[2-(methylamino)pyridine-3-carbonyl]piperazin-2-one
1-cyclobutanecarbonyl-N-methyl-N-(quinolin-2-ylmethyl)piperidin-4-amine
N-[3-(furan-2-yl)phenyl]-1-[2-(pyridin-3-yl)acetyl]piperidine-4-carboxamide
5-(1H-imidazol-1-ylmethyl)-N-methyl-N-[(3-methylthiophen-2-yl)methyl]furan-2-carboxamide
N-(2,1,3-benzoxadiazol-4-ylmethyl)-N-[(3-ethoxyphenyl)methyl]cyclopropanamine
(2R,3R)-1'-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-3-(pyrrolidin-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
4-ethyl-3-{[1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]methyl}-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}propanamide
5-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-2-(propan-2-yl)-3,4-dihydropyrimidin-4-one
N-methyl-2-[methyl({[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl})amino]propanamide
4-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}morpholine