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dimethyl({[(1R,5S,6S)-3-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl})amine
1-(cyclopropylmethyl)-2-(propan-2-yl)-4-[4-(4H-1,2,4-triazol-4-yl)benzoyl]-1,4-diazepane
1-ethyl-N-[3-(4-fluorophenyl)propyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
1-{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}-4-(propan-2-yl)piperazine
[1-({[6-(piperidin-3-yl)pyrimidin-4-yl]amino}methyl)cyclobutyl]methanol
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}thian-4-amine
2-(azocan-1-yl)-1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
2-(2H-1,3-benzodioxol-5-yl)-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]acetamide
3-({4-[(4-tert-butyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}methyl)-N-methylpyridin-2-amine
3-[2-(2,6-difluorophenyl)ethyl]-1-[5-(methoxymethyl)furan-2-carbonyl]piperidine
(1R,6S)-9-methyl-3-(5-methylpyrazine-2-carbonyl)-3,9-diazabicyclo[4.2.1]nonane
4-(piperidin-1-ylmethyl)-N-[(1-propyl-1H-pyrazol-4-yl)methyl]benzamide
ethyl 3-[(2,4-difluorophenyl)methyl]-1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidine-3-carboxylate
1-methyl-4-(1-phenylpiperidin-4-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
[(3R,4R)-1-[3-(5-methylfuran-2-yl)benzoyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(1S,5R)-3-[(4-fluorophenyl)methanesulfonyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[(dimethylamino)methyl]-1-[(5-ethylpyridin-2-yl)methyl]piperidin-3-ol
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-(6-phenoxypyridin-3-yl)-1-(pyridin-3-ylmethyl)piperidine-2-carboxamide
2-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-3-carboxamide
N-[2-(1-methylpyrrolidin-2-yl)ethyl]-2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2,5-dimethyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
3-(1-{[4-(difluoromethoxy)phenyl]methyl}piperidin-4-yl)-N-[2-(dimethylamino)ethyl]propanamide
1-{2-[(1-methylpiperidin-4-yl)oxy]phenyl}-5-oxopyrrolidine-3-carboxylic acid
3-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)piperidin-2-one
N-(pyridin-2-ylmethyl)-3-{[1-(pyridin-4-yl)piperidin-4-yl]oxy}benzamide
1'-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
8-fluoro-N-methyl-4-oxo-N-(2-phenoxyethyl)-1,4-dihydroquinoline-3-carboxamide
N,N-dimethyl-6-oxo-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decane-2-sulfonamide
[4-(3-chloro-4-fluoro-1-benzothiophene-2-carbonyl)-1,4-oxazepan-6-yl]methanol
5-{2-[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-7-yl]-2-oxoethyl}-3,4-dihydropyrimidin-4-one
(1S,5R)-3-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(3-acetylphenyl)-1-methyl-2-oxo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-carboxamide
2-(dimethylamino)-N,4-dimethyl-N-[1-(pyridin-3-yl)pentyl]pyrimidine-5-carboxamide
1-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-1H-pyrazole-4-carbonyl)-4-(furan-2-carbonyl)piperazine
4-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]-1-(1H-indazol-5-yl)piperazin-2-one
N-[(4-methoxyphenyl)methyl]-2,6-dimethyl-N-(oxolan-2-ylmethyl)pyridine-4-carboxamide
methyl 9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-7-oxo-3-{[4-(propan-2-yloxy)phenyl]methyl}-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-[1-(3-methylbutyl)-8-[1-(methylsulfanyl)propan-2-yl]-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanamide
2-(pyridin-3-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]pyrimidine-5-carboxamide
2-{5-[(N-cyclohexylacetamido)methyl]-1,2,3,6-tetrahydropyridin-1-yl}propanamide
2-methyl-4-{[(prop-2-en-1-yl)(pyridin-3-ylmethyl)amino]methyl}phenol
N-({5-[6-(dimethylamino)pyrazin-2-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
4-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-methyl-5-propylpyrimidine
1-{2-[2-(2,3-dimethoxyphenyl)-1H-imidazol-1-yl]propyl}-1H-1,2,4-triazole
N3-cyclohexyl-N5-cyclopropyl-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[1-(1,3-thiazol-2-yl)propyl]-1H-pyrazole-3-carboxamide