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methyl 4-[5-(2-fluoro-6-methoxyphenyl)-4-phenyl-1H-imidazol-1-yl]butanoate
2-(4-benzyl-2-oxopyrrolidin-1-yl)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methylacetamide
5-(1,3-benzothiazol-6-yl)-1,2,3,4-tetrahydroisoquinoline
N-(1-{4-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]phenyl}-1H-pyrazol-4-yl)oxane-4-carboxamide
6-(2,5-dimethylfuran-3-yl)-7-methyl-2-(1,4-oxazepane-4-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
(2R)-2-amino-1-{4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}propan-1-one
2-[4-(2-aminopyrimidin-4-yl)-1H-pyrazol-1-yl]-N-(3-methyl-1-phenyl-1H-pyrazol-5-yl)acetamide
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-6-(hydroxymethyl)-1,4-oxazepane-4-carboxamide
ethyl 4-[(3-fluorophenyl)methyl]-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxylate
N-(2-{[methyl({[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl})amino]methyl}quinolin-6-yl)acetamide
2-(methylamino)-N-[(3-methylphenyl)(thiophen-2-yl)methyl]acetamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
(1s,4s)-4-{4-[1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-1H-1,2,3-triazol-1-yl}cyclohexan-1-amine
8-[(5-ethylpyridin-2-yl)methyl]-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
3,6,7-trimethyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1-benzofuran-2-carboxamide
4-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]benzene-1-sulfonamide
2-(cyclohex-1-en-1-yl)-N-{[7-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
(3R)-1-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}pyrrolidin-3-ol
4-methyl-1-[(2-methylphenyl)methyl]-1,4-diazepan-5-one
ethyl 4-{[(1-cyclopentylpiperidin-4-yl)methyl]amino}piperidine-1-carboxylate
1-methyl-2-oxo-8-(pyridin-3-ylmethyl)-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)benzamide
2-(4-methoxyphenyl)-1-[3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]ethan-1-one
ethyl 1-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]piperidine-2-carboxylate
2,2,3,3-tetramethyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}cyclopropane-1-carboxamide
N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-1-(4-fluorophenyl)cyclopropane-1-carboxamide
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-6-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
8-(2-amino-6-methylpyrimidin-4-yl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
7-(isoquinoline-5-carbonyl)-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-(3-methoxyphenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
(2S,4S)-4-amino-N-(propan-2-yl)-1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}pyrrolidine-2-carboxamide
2-[3-(4-phenylpiperazin-1-yl)piperidine-1-carbonyl]pyrazine
1-{[(3R,4R)-4-(hydroxymethyl)-1-(2-methyl-5-propylpyrimidin-4-yl)pyrrolidin-3-yl]methyl}piperidin-4-ol
methyl 3-(2-methoxyacetamido)-1-(3-phenylpropyl)-5-(propylamino)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
dimethyl(1-{3-[3-(methylsulfanyl)-1H-1,2,4-triazol-5-yl]phenyl}ethyl)amine
4-ethyl-3-{[1-(6-methyl-2-propylpyrimidin-4-yl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[2-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-oxoethyl]piperazin-2-one
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-{2,8-diazaspiro[4.5]decan-2-yl}-2-(dimethylamino)-2-(3-methylphenyl)ethan-1-one
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-(1H-1,2,4-triazol-1-yl)benzamide
4-{1-benzyl-3-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-2,1,3-benzoxadiazole
(1S,5R)-3-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(furan-2-ylmethyl)-2-(4-methyl-1,4-diazepan-1-yl)-N-(2-methylpropyl)acetamide
6-[1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)piperidin-3-yl]-2-methylpyrimidin-4-ol
N-[2-(furan-2-ylmethyl)-3-hydroxypropyl]-2-(2-oxopiperidin-1-yl)acetamide
2-[4-(4-methoxyphenyl)-2-methyl-3-oxopiperazin-1-yl]-N-(pyridin-2-ylmethyl)acetamide
1-cyclopropyl-N-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
N-[(2-aminopyrimidin-5-yl)methyl]-N-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide