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3-({[2-(dimethylamino)ethyl]amino}methyl)-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxypiperidin-2-one
4-(4-methylphenoxy)-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)piperidine-4-carboxamide
[1-(1-benzofuran-2-ylmethyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
3-{4-methyl-6H,7H,8H-cyclopenta[g]quinazolin-2-yl}-3,9-diazaspiro[5.6]dodecan-10-one
benzyl({[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl})ethylamine
4-[6-amino-5-cyano-4-(pyridin-3-yl)pyridin-2-yl]benzoic acid
2-[benzyl(methyl)amino]-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
N-[2-(ethylsulfanyl)ethyl]-6-methoxy-1-methyl-1H-indole-2-carboxamide
N-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}-3-{2-[(4-methylphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
2-(1-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}piperidin-2-yl)acetic acid
2-(4-chloro-2-methylphenoxy)-N-methyl-N-{2-[4-(4-methylpiperazine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}propanamide
3-(3-hydroxy-3-methylbutyl)-N-[2-(4-hydroxyphenyl)ethyl]benzamide
N-[(1R,3R)-3-aminocyclopentyl]-2-(1,1-dioxo-1λ6-thiomorpholin-4-yl)benzamide
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-2-(dimethylamino)-2-(2-methylphenyl)acetamide
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-1,3-dimethyl-1H-pyrazole-4-carboxamide
6-amino-N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methylpyridine-2-carboxamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine-2-carboxamide
methyl (2R,4S)-1-{[2,4-dimethyl-5-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-4-hydroxypiperidine-2-carboxylate
4-methyl-1-(2-{[3-(trifluoromethyl)phenyl]methyl}morpholin-4-yl)pentane-1,2-dione
3-(2H-1,3-benzodioxol-5-ylmethyl)-1-(furan-3-carbonyl)-3-methylpiperidine
3-({4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)phenol
(2S,4S)-N-cyclopropyl-1-[(2,5-dimethoxyphenyl)methyl]-4-[(4-fluorophenyl)sulfanyl]pyrrolidine-2-carboxamide
methyl 3-({2-[(2-fluorophenyl)methyl]-1,3-benzoxazol-6-yl}formamido)propanoate
N-[2-(1-methanesulfonylpiperidin-2-yl)ethyl]pyrimidin-4-amine
3-{[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]methyl}-1H-indole
5-(2H-1,3-benzodioxol-5-yl)-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1,2,4-triazin-3-amine
4-methyl-2-(methylsulfanyl)-6-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}pyrimidine
2-ethyl-4-methyl-5-{3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-1,3-oxazole
6-(6-aminopyridin-3-yl)-N-cyclopentylpyridazin-3-amine
4-{[(3S,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]methyl}benzonitrile
methyl (1R,3S,3aR,6aS)-1-[(4-hydroxyphenyl)methyl]-5-methyl-4,6-dioxo-3-(1,3-thiazol-2-yl)-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)(1H-pyrazol-5-ylmethyl)amine
N-(4-fluorophenyl)-1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-amine
N-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]acetamide
5-[({[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]-N,N-dimethyl-1,3-thiazol-2-amine
N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
(4aR,7aS)-1-[2-(dimethylamino)acetyl]-4-[2-(propylsulfanyl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-methyl-1-(3-methylphenyl)-4-[3-(pyridin-3-yl)propanoyl]piperazin-2-one
8-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
(1S,6R)-3-(1,3-benzothiazol-2-ylmethyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-3-oxopiperazine-1-carboxamide
2-[methyl({4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenyl})amino]ethan-1-ol
3-{5-butyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1-(4-hydroxypiperidin-1-yl)propan-1-one
methyl 3-{[4-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-7-oxo-1,4-diazepan-1-yl]methyl}benzoate
1-(4-{6-amino-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-6-hydroxy-1,4-diazepan-1-yl)propan-1-one
2-(2,3-dihydro-1H-inden-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N-[1-(3-methylbutanoyl)azepan-3-yl]-3-(pyridin-3-yl)propanamide
N-[2-(5,7-difluoro-2-methyl-1H-indol-3-yl)ethyl]-2-(2,5-dioxoimidazolidin-1-yl)acetamide
3-[(1-acetylpiperidin-4-yl)oxy]-N-[2-(3-chlorophenyl)ethyl]-4-methoxybenzamide