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N-[(1-ethylpyrrolidin-2-yl)methyl]-3-[1-(2-methylpyrimidine-5-carbonyl)piperidin-4-yl]propanamide
1-(2-methoxyethyl)-8-[(1-methyl-1H-indol-3-yl)methyl]-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[4-(oxolan-3-ylmethyl)piperazin-1-yl]pyridine-3-carboxamide
2-cyclohexyl-5-{[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methyl}pyrimidine
3-{[5-(4-methanesulfonylphenyl)-4-phenyl-1H-imidazol-1-yl]methyl}-1,2-oxazole
N-[3-(3-methylphenyl)phenyl]-1-(1H-pyrazol-3-ylmethyl)piperidine-3-carboxamide
1-[(1-benzyl-1H-imidazol-2-yl)methyl]-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
4-(4-chlorophenyl)-N-[2-hydroxy-2-(pyridin-2-yl)ethyl]butanamide
3-(5-hydroxyadamantan-2-yl)-3H,4H-pyrido[3,4-d]pyrimidin-4-one
1-(3-{[(oxan-4-yl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
(3aS,6aS)-2-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)thiophene-2-sulfonamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-benzyl-4-{[(2-methoxynaphthalen-1-yl)methyl]amino}pyrrolidine-2-carboxamide
1-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-2-ethylpiperidine
2-amino-4-(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(pyridin-2-yl)pyridine-3-carbonitrile
1-ethyl-N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1H-pyrazole-5-carboxamide
(1S,5R)-6-(2-methoxyethyl)-3-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(5-cyclopropyl-1-{8-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-1H-pyrazole-4-carbonyl)-N,N-diethylpyrrolidin-3-amine
N-{1-[1-(1-carbamoylcyclopropanecarbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
1-(6-ethyl-2-methylpyrimidin-4-yl)-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]piperidin-4-amine
N-(2-fluorophenyl)-3-(1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)propanamide
2-[1-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-4-yl]-1,2,3,4-tetrahydroisoquinoline
5-(2-methyl-1-benzofuran-5-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
4-({4-methyl-5-[({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)piperidine
N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(pyridin-3-yl)acetamide
2-(2,2-dimethylpropanoyl)-N-(thiophen-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
2-(2-hydroxy-4-methylpentanoyl)-N-(5-methyl-1,2-oxazol-3-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
2-{4-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidine-1-carbonyl]piperidin-1-yl}acetamide
4-(1H-imidazol-1-yl)-N-{[4-(oxolan-2-ylmethoxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)benzamide
N-(8-methylquinolin-5-yl)-2-oxo-1-oxa-3,8-diazaspiro[4.6]undecane-8-carboxamide
N,6-dimethyl-N-[3-(pyrrolidin-1-yl)butyl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
3-(6-chloro-1H-1,3-benzodiazol-2-yl)phenol
4-benzyl-1-[(4-methylphenyl)methyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(4,7-dimethylquinazolin-2-yl)-N-(propan-2-yl)azepan-4-amine
2-methyl-2-phenyl-1-[3-(1H-pyrazol-5-yl)piperidin-1-yl]propan-1-one
7-methoxy-3-[1-methyl-5-(thiophen-2-yl)-1H-pyrazole-3-carbonyl]-2,3,4,5-tetrahydro-1H-3-benzazepine
2-(1H-imidazol-1-yl)-1-[2-(2-phenylethyl)piperidin-1-yl]ethan-1-one
5-(2,3-dihydro-1H-isoindole-2-carbonyl)-2-(4-methylphenyl)pyrimidin-4-ol
N-(3-methoxyphenyl)-1-[2-(2-methylpropanamido)ethyl]-1H-1,2,3-triazole-4-carboxamide
[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl][(dimethyl-1,2-oxazol-4-yl)methyl]methylamine
9-(2-methylfuran-3-carbonyl)-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
(2E)-3-(3,4-dimethoxyphenyl)-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}prop-2-enamide
1-{[1-(3-cyanopyridin-2-yl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
N-[(3S,4R)-1-(3-cyano-6-methylpyridin-2-yl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
1-(2-methylpropyl)-2-({4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}methyl)-1H-1,3-benzodiazole
N-(3-fluoro-2-methylphenyl)-2-[2-(3-fluorophenyl)-3-oxopiperazin-1-yl]acetamide
2-(3,5-dimethoxyphenyl)-1-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}ethan-1-one
N-[1-(adamantan-1-yl)propyl]-3-[5-(5-methyl-1,2-oxazol-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
5-{3-[1-(dimethylamino)ethyl]phenyl}pyridine-3-carboxylic acid