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N,N-dimethyl-5-{[(3-methylphenyl)methyl]amino}-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
7-methyl-N-[(3-methylphenyl)methyl]-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
5-(4-cyclopentylpiperazin-1-yl)-1-ethyl-N-(furan-3-ylmethyl)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-[2-(aminomethyl)-5-chloro-2,3-dihydro-1-benzofuran-7-yl]-N-(propan-2-yl)benzamide
5-methyl-14-(5-propylfuran-2-yl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
6-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-N-ethyl-N-methylpyridine-3-carboxamide
ethyl 1-{2-[bis(propan-2-yl)amino]ethyl}-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylate
5-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-methyl-2-(4H-1,2,4-triazol-4-yl)pyridine
N'-(3-chloro-2-methylphenyl)-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}propanediamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
2-(3-fluorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-1-yl]ethan-1-one
N-[(3-ethoxyphenyl)methyl]-N-methyl-2-{8-methyl-3-oxo-2,8-diazaspiro[4.5]decan-2-yl}acetamide
8-{[3-(morpholin-4-yl)phenyl]methyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
(3S,4S)-1-(1-benzothiophen-2-ylmethyl)-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-2-methoxy-5-sulfamoylbenzamide
N-[(5-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
(2S)-4-methyl-2-[4-(pyrimidin-5-yl)-1H-1,2,3-triazol-1-yl]pentan-1-ol
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-2-[methyl(pyridin-4-ylmethyl)amino]acetamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[2-(cyclohex-1-en-1-yl)ethyl]-N-propylacetamide
(3S,4S)-1-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]-4-cyclopropylpyrrolidine-3-carboxylic acid
N,2-dimethyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}imidazo[1,2-a]pyrimidine-3-carboxamide
1-[(2-{[(benzylsulfamoyl)amino]methyl}phenyl)methyl]pyrrolidin-2-one
N-methyl-4-sulfamoyl-N-[1-(thiophen-2-yl)ethyl]butanamide
4-[2-(2-hydroxyethyl)-3-oxo-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridine-6-carbonyl]-1,2-dihydroquinolin-2-one
N-cyclopropyl-N-[(2-ethoxyphenyl)methyl]but-3-enamide
3-cyclopropyl-5-[(2,3,4-trifluorophenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2-(5-fluoro-2-methylphenyl)-1-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]ethan-1-one
3-ethyl-N-(2-hydroxyethyl)-N-[(2-methoxyphenyl)methyl]-4-methyl-1H-pyrazole-5-carboxamide
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-(1,2-oxazole-3-carbonyl)piperazine
dimethyl({[4-methyl-5-(1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}piperidin-3-yl)-4H-1,2,4-triazol-3-yl]methyl})amine
N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}-2,4-dimethyl-1,3-thiazole-5-carboxamide
N-[2-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-5-methylthiophene-2-carboxamide
N-[2-(furan-2-ylmethyl)-3-hydroxypropyl]-4-(1H-imidazol-1-yl)benzamide
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(2H-1,2,3,4-tetrazol-2-yl)ethan-1-one
2-(2,4-dichlorophenoxy)-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}acetamide
7-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-sulfonyl}-2,3,4,5-tetrahydro-1,5-benzothiazepin-4-one
1-methyl-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}piperidine-2-carboxamide
4-({[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]carbamoyl}amino)-N,N,3-trimethylbenzamide
N-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]-3-(1-methylpiperidin-3-yl)propanamide
4-(4-methylphenoxy)-1-(1H-pyrazole-4-carbonyl)piperidine
4,6-dimethyl-2-[4-({4-[(methylamino)methyl]-1H-1,2,3-triazol-1-yl}methyl)piperidin-1-yl]pyridine-3-carbonitrile
N-[(4-fluorophenyl)methyl]-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-[4-(6-ethyl-2-methylpyrimidin-4-yl)-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol
N-cyclopropyl-1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}piperazine-2-carboxamide
4-[4-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]-6-[(3-methoxyphenyl)methoxy]-1-(2-methylpropyl)-1,4-diazepan-2-one
1-{4-[1-(3-fluorophenyl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]-1H-pyrazol-3-yl}-1H-1,2,3,4-tetrazole
2-benzyl-4-(2-hydroxy-5-methoxyphenyl)-3-methyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
5-{[4-(1-benzyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}-N,N-dimethylfuran-2-carboxamide
3-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-3-ethyl-1-(4-fluorophenyl)urea
2-{[(2,1,3-benzothiadiazol-5-ylmethyl)(methyl)amino]methyl}benzoic acid