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(3R,5S)-5-[4-(3,4-dichlorophenyl)piperazine-1-carbonyl]pyrrolidin-3-ol
N-({7-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)oxolane-3-carboxamide
2-(4-{[3-(3-methoxyphenoxy)azetidin-1-yl]methyl}-3,5-dimethyl-1H-pyrazol-1-yl)ethan-1-ol
2-(2,5-dimethylphenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]ethan-1-one
3-[1-(2-hydroxyethyl)-3-(phenoxymethyl)-1H-1,2,4-triazol-5-yl]-1,2-dihydroquinolin-2-one
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
2-(4-fluorophenyl)-1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
1-methyl-2-(1-{[1-(2-methylphenyl)pyrrolidin-3-yl]methyl}-1H-imidazol-2-yl)-1H-imidazole
3-(3-fluorophenyl)-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
N-(2-methoxypyridin-3-yl)-2-(pyrrolidin-3-yl)benzamide
1-(2-methoxyethyl)-6-oxo-N-[(4-phenyloxan-4-yl)methyl]piperidine-3-carboxamide
2-[(3R,4S)-3-(4-cyanobenzenesulfonamido)-4-cyclopropylpyrrolidin-1-yl]acetamide
(propan-2-yl)({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)amine
4-methoxy-N-(2-methoxyethyl)-2-({1-[1-(methylsulfanyl)propan-2-yl]piperidin-4-yl}oxy)benzamide
1-cyclohexyl-5-(4-fluorophenoxymethyl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-6-methylpyridine-3-carboxamide
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-(furan-2-yl)-7-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[2-(pyridin-3-yl)ethyl]amine
4-(4-methyl-1H-pyrazol-1-yl)-6-(1H-pyrazol-3-yl)pyrimidine
3-(2-ethyl-1H-imidazol-1-yl)-N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
3-(2-methyl-1H-imidazol-1-yl)-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]propan-1-one
4-[5-(3-methyl-3-phenylpiperidine-1-carbonyl)-1H-pyrazol-3-yl]pyridine
1-(3-hydroxy-2,2-dimethylpropyl)-N-[3-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
(4aR,8aR)-2-cyclobutanecarbonyl-7-[(3-fluoro-4-methylphenyl)methyl]-decahydro-2,7-naphthyridin-4a-ol
6-ethoxy-2-{[3-(morpholin-4-yl)azetidin-1-yl]methyl}quinoline
(2R,6R)-4-(2-amino-6-methylpyrimidin-4-yl)-10-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
(2S,4R)-4-amino-N-ethyl-1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)sulfonyl]pyrrolidine-2-carboxamide
5-methoxy-1,2-dimethyl-N-[2-(2-methylpropanesulfonyl)ethyl]-1H-indole-3-carboxamide
methyl({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}){[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
3-propyl-5-[3-(1H-pyrazol-1-yl)phenyl]-1,2,4-oxadiazole
2-[benzyl(methyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
4-[3-(azetidine-1-carbonyl)piperidin-1-yl]-1-(2,3-dihydro-1H-inden-2-yl)piperidine
N-[(4-chlorophenyl)methyl]-N-(3-hydroxypropyl)-2-(1H-imidazol-2-yl)benzamide
4-[(5-chloro-2,3-dimethoxyphenyl)methyl]-1-(3-methoxyphenyl)piperazin-2-one
1,3-dimethyl-5-{2-[4-(2-methylphenyl)-1,4-diazepan-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-cyclopropyl-N-(thiophen-3-ylmethyl)-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
(4aS,7aR)-1-[(2-ethylphenyl)methyl]-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{3-[ethyl(pyridin-4-ylmethyl)amino]piperidine-1-carbonyl}pyridin-2-ol
{7-[6-(azepan-1-yl)pyridazin-3-yl]-5-fluoro-2,3-dihydro-1-benzofuran-2-yl}methanamine
5-[2-(methylamino)ethyl]-1-{[3-(trifluoromethoxy)phenyl]methyl}pyrrolidin-2-one
5-fluoro-N,N-dimethyl-2-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}pyrimidin-4-amine
2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}pyridine-3-carboxylic acid
N3-methyl-N3-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-N5-{[3-(trifluoromethoxy)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
2-{4-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-yl]piperidin-1-yl}-4,6-dimethylpyrimidine
3-{4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl}propanamide
N-[(3,4-dimethoxyphenyl)methyl]-2-[4-hydroxy-4-(hydroxymethyl)azepan-1-yl]acetamide
N-{5-[2-(pyridin-2-yl)-1H-imidazol-1-yl]pyridin-2-yl}methanesulfonamide
methyl 2-[(3,5-dimethylphenyl)sulfamoyl]-6-(pyrazine-2-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(3aS,6aS)-2-[(5-chlorofuran-2-yl)methyl]-5-(dimethylcarbamoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{2-oxo-2-[2-(pyridin-3-yl)pyrrolidin-1-yl]ethyl}piperidine-4-carboxamide