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2-[1-(furan-2-ylmethyl)-4-{[5-(1H-pyrazol-5-yl)furan-2-yl]methyl}piperazin-2-yl]ethan-1-ol
9-(oxan-4-yl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decane
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
methyl 3-(4-{[4-(3-methylphenoxy)piperidin-1-yl]methyl}-1H-pyrazol-1-yl)propanoate
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-ethyl-N-methylacetamide
(2S)-2-[(1,7-dimethyl-1H-indol-2-yl)formamido]-3-phenylpropanamide
3-(2-methoxyethyl)-1-(2-methoxyphenyl)-5-[1-(1H-1,2,4-triazol-1-yl)ethyl]-1H-1,2,4-triazole
1-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-methylpropan-1-one
1-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-3-(pyrazin-2-yl)propan-1-one
propan-2-yl 4-{[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]amino}piperidine-1-carboxylate
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-2-oxo-1-oxaspiro[4.4]nonane-4-carboxamide
2-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}-1-(prop-2-en-1-yl)pyrrolidine
1-{2-[1-(4-chloro-2-methylphenyl)-3-methyl-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,2,3,4-tetrazole
4-{[1-(4-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1,5-dimethyl-1H-pyrazole
2-(4-chlorophenyl)-1-{4-[2-(oxolan-2-yl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}ethan-1-one
7-[(2S)-2-methoxy-2-phenylacetyl]-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-[2-(trifluoromethyl)morpholin-4-yl]pyrimidin-4-amine
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-2,4-dimethyl-1,3-thiazole-5-carboxamide
3-[3-methyl-1-(2-methylpropyl)-1H-pyrazol-5-yl]-1-[(5-methylfuran-2-yl)methyl]urea
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-3-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
methyl 5-[(2,2-dimethylpropyl)amino]-1-(2-methoxyethyl)-3-(3-methylbutanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(2,6-difluoro-3-methoxyphenyl)methyl]-2-(1H-pyrazol-1-yl)butanamide
[3-(1H-imidazol-1-yl)propyl][(3-methyl-1H-pyrazol-5-yl)methyl](pyridin-3-ylmethyl)amine
N,3,6-trimethyl-N-(quinolin-5-ylmethyl)-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
N,3,4,7-tetramethyl-N-(thian-4-yl)-1H-indole-2-carboxamide
1-(1-benzofuran-2-ylmethyl)-4-[3-(pyrrolidine-1-carbonyl)phenoxy]piperidine
N-[2-(1-methylpiperidin-3-yl)ethyl]-1-(morpholin-4-yl)cyclohexane-1-carboxamide
3-[1-(2-benzyl-1,3-thiazole-4-carbonyl)pyrrolidin-2-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(cyclopentylcarbamoyl)-4-(3-fluorophenoxy)piperidine-4-carboxylic acid
1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-6-azaspiro[2.5]octane
2-({2-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
2-(5-chloro-1H-1,3-benzodiazol-2-yl)-1-[(3S)-3-(dimethylamino)azepan-1-yl]ethan-1-one
(1S,5R)-3-benzyl-6-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
9-(cyclopropylmethyl)-4-(3-methoxypropyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
methyl 2-(benzylsulfamoyl)-6-[2-(cyclohex-1-en-1-yl)acetyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(3S,4R)-4-(4-fluorophenyl)-1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]pyrrolidine-3-carboxylic acid
(2R,3R,6R)-3-phenyl-5-(quinolin-2-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N,N-dimethyl-2-[(1S,5R)-6-[1-(4-methylphenyl)cyclopropanecarbonyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]-1-(1-methyl-1H-pyrrole-2-carbonyl)piperidine
4-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-7-(2,3-dimethoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(5-ethyl-1,3-oxazole-4-carbonyl)-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
N-(2-hydroxyethyl)-5-methoxy-N-[(2E)-3-phenylprop-2-en-1-yl]-1H-indole-2-carboxamide
1-(2-oxo-2-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethyl)pyrrolidin-2-one
4-(3,5-dimethyl-1H-pyrazol-1-yl)-1-{4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}butan-1-one
ethyl 1-(2,1,3-benzoxadiazol-4-ylmethyl)-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylate
5-(4-chloro-3,5-dimethylphenoxymethyl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1,2-oxazole-3-carboxamide
9-[4-(3-hydroxypiperidin-1-yl)pyrimidin-2-yl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
1,3-dimethyl-2,6-dioxo-N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)-2,3-dihydro-1H-indene-1-carboxamide