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N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-2-(furan-2-yl)-2-oxoacetamide
1-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]-2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
3-({1-[4-(morpholin-4-yl)butanoyl]pyrrolidin-3-yl}methyl)benzamide
(2R,6R)-4-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(ethanesulfonyl)ethan-1-one
(2E)-N-{[7-(3,6-dimethylpyrazin-2-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(4-methoxyphenyl)prop-2-enamide
1-(oxolane-2-carbonyl)-N-[(3-propyl-1,2-oxazol-5-yl)methyl]piperidin-4-amine
3-[(2R,3R,6R)-5-cyclopentanecarbonyl-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
dimethyl({4-[(7-methyl-2-phenyl-1H-indol-3-yl)methyl]-1,4-oxazepan-6-yl}methyl)amine
ethyl 1-[6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidine-3-carboxylate
1-cyclobutanecarbonyl-4-{3-[(2-methylphenyl)methoxy]azetidine-1-carbonyl}piperidine
1-{2-[2-(pyridin-4-yl)-1H-imidazol-1-yl]ethyl}imidazolidin-2-one
1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-2-(5-methyl-1,2-oxazol-3-yl)piperidine
1'-[4-methyl-6-(2-methylpropyl)pyrimidin-2-yl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,3'-pyrrolidine]
2-{[4-(5-methylfuran-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}quinolin-8-ol
2-amino-4-{2-[(oxolan-2-ylmethyl)amino]pyrimidin-5-yl}-6-phenylpyridine-3-carbonitrile
1-[(3-chlorophenyl)methyl]-N-phenylpiperidin-3-amine
N,1-dibenzyl-N-(2-hydroxyethyl)-2-methyl-5-(2-methylpropanamido)-1H-1,3-benzodiazole-7-carboxamide
2-(2,5-dimethoxyphenyl)-1-[7-({methyl[2-(pyridin-2-yl)ethyl]amino}methyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
1-{2-[methyl({[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]pyrimidin-4-yl}piperidin-3-ol
[1-(3,4-dimethylphenyl)ethyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N,2,3,5-tetramethylpyrazolo[1,5-a]pyrimidin-7-amine
6-fluoro-2-[4-(1-methylpiperidin-4-yl)piperazine-1-carbonyl]-1H-1,3-benzodiazole
1-({3-[(3-fluorophenyl)methoxy]-4-methoxyphenyl}methyl)piperidine-3-carbonitrile
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-[4-(methylsulfanyl)benzoyl]pyrrolidin-3-yl]methanol
6-butyl-2-[4-(piperazin-1-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
ethyl 4-[(4-methoxyphenyl)methyl]-1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]piperidine-4-carboxylate
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-N,N-dimethylaniline
4-{[4-methyl-5-({[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}sulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine
4-[4-(6-methoxypyridin-2-yl)benzenesulfonyl]thiomorpholine
ethyl 2-[1-(2,5-difluorobenzenesulfonyl)piperidin-2-yl]acetate
8-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(5-methyl-1,2-oxazol-3-yl)-1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidine
(1R,2R,6S,7S)-N-{3-[(2-methoxyethyl)carbamoyl]-2-methylphenyl}-4-azatricyclo[5.2.1.02,6]decane-4-carboxamide
N-({1-[(1,4-dimethylpiperidin-4-yl)methyl]pyrrolidin-3-yl}methyl)-2-(pyrrolidin-1-yl)acetamide
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N,1-dimethyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(3S,4R)-1-(3,4-dimethylbenzoyl)-4-(3-methylthiophen-2-yl)piperidin-3-ol
N-[(4-fluorophenyl)(pyridin-4-yl)methyl]-5-methyl-1,3,4-oxadiazol-2-amine
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-(morpholin-4-yl)butanamide
methyl 1-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-2-carboxylate
5-{4-[3-(morpholin-4-ylmethyl)phenyl]phenyl}-1H-imidazol-2-amine
2-(5-chloropyridin-2-yl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
4-methoxy-N-[2-(1-methylpyrrolidin-2-yl)ethyl]-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
2-hydroxy-2-(4-methoxyphenyl)-N-[3-(pyridin-3-yl)propyl]acetamide
3-(2-ethylbutyl)-8-[2-(methylamino)-1,3-thiazole-4-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[2-(2-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-3-(methoxymethyl)piperidine
8-chloro-4-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-2-methylquinoline
2-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]-3,4-dihydroquinazolin-4-one
[(3R,5R)-1-(2,5-dimethylfuran-3-carbonyl)-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
7-(3-phenylpropyl)-2-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decane