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4-(2-ethyl-4-methyl-1,3-oxazole-5-amido)-N-phenylpiperidine-1-carboxamide
7-({cyclopropyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)-4-methyl-2H-chromen-2-one
2-[(1-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}piperidin-4-yl)oxy]pyrimidine
N-[2-(dimethylamino)-3-methylbutyl]-2,5-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
1-[(4-chlorophenyl)methyl]-4-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperazine
1-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]-2-(2-methylphenyl)ethan-1-one
4-(2-oxo-1,3-oxazolidin-3-yl)-N-[3-(pyridin-3-yl)phenyl]piperidine-1-carboxamide
4-ethyl-3-[1-(2-methyloxolane-2-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[4-(4-methoxyphenyl)-1H-imidazol-2-yl]-1-(propan-2-yl)pyrrolidin-2-one
1-methyl-4-[3-(2-phenylethyl)-5-[2-(1H-1,2,3,4-tetrazol-1-yl)ethyl]-1H-1,2,4-triazol-1-yl]piperidine
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-1-cyclopentanecarbonylpiperidine-4-carboxamide
dimethyl({2-[2-(5-methylpyridin-3-yl)phenoxy]ethyl})amine
3-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1-(5,6,7,8-tetrahydronaphthalen-1-yl)urea
4-[3-(methanesulfonylmethyl)piperidin-1-yl]-6-(propan-2-yl)pyrimidin-2-amine
N-(1,1-dioxo-1λ6-thian-4-yl)-N,2,6-trimethylquinoline-4-carboxamide
methyl 4-(5-{[(2-hydroxypropyl)(methyl)amino]methyl}-1,2,4-oxadiazol-3-yl)benzoate
3-[(3S,5S,9R)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]-1-(5-fluoro-2-methylphenyl)urea
(1S,5R)-3-({7-chloro-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(2-phenylethyl)-5-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazol-5-yl]-1H-1,2,4-triazole
5-[4-(2-methoxyethoxy)phenyl]-2-(4H-1,2,4-triazol-4-yl)pyridine
{4-[(4-chlorophenyl)methyl]-1-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl}methanol
(3R,9aR)-8-(3-fluoro-4-methylbenzoyl)-3-(hydroxymethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[3-(pyrrolidin-1-yl)propyl]amine
1'-(3,5-difluoropyridine-2-carbonyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-{1-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]piperidin-3-yl}benzoic acid
5-[4-(benzyloxy)piperidine-1-carbonyl]-4-methyl-2-(propan-2-yl)pyrimidine
N-{[2-(azepan-1-yl)-7-chloroquinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]oxolane-2-carboxamide
2-(1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-2-yl)-1H-1,3-benzodiazole
[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl](ethyl)[(1-ethyl-1H-pyrazol-4-yl)methyl]amine
2-methyl-1-({4-[2-oxo-2-(piperidin-1-yl)ethoxy]phenyl}methyl)-1,4-diazepan-5-one
3-ethyl-8-[2-(oxan-2-ylmethoxy)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]-3-[(oxolan-3-yl)sulfamoyl]benzamide
N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-1-(pyridin-4-ylmethyl)piperidine-3-carboxamide
7-(3-chlorophenyl)-4-(1,3-thiazol-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
ethyl 5-[2-(dimethyl-1H-1,2,4-triazol-1-yl)acetyl]-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-{3-[(dimethylsulfamoyl)amino]phenyl}urea
N-[2-(4-hydroxy-6-methylpyrimidin-2-yl)ethyl]-2-(thiophen-3-yl)acetamide
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-3-oxo-3,4-dihydro-2H-1,4-benzoxazine-7-carboxamide
ethyl 1-{2-[3-(2-fluorophenyl)-1-(2-methoxyethyl)-2,5-dioxopyrrolidin-3-yl]acetyl}piperidine-3-carboxylate
4-{2-methyl-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl}-1,2-dihydrophthalazin-1-one
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)pentanamide
3-(6-{[2-(dimethylamino)ethyl]amino}-1H-pyrrolo[2,3-b]pyridin-4-yl)-5-hydroxybenzoic acid
N-(1-methyl-1H-1,3-benzodiazol-6-yl)-4-(2-phenoxyethyl)piperazine-1-carboxamide
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-4,6-dimethylpyrimidin-2-amine
3-methyl-8-[3-(piperidin-3-yl)benzoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
6-methoxy-4-{6-oxa-9-azaspiro[4.5]decane-9-carbonyl}-1,2,3,4-tetrahydroquinolin-2-one
N-cyclopropyl-3-methyl-N-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)thiophene-2-carboxamide
(1S,5R)-6-[2-(methylsulfanyl)pyrimidine-5-carbonyl]-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
2-methyl-N-[2-methyl-2-(pyrrolidin-1-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-[3-({[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amino}methyl)phenyl]ethan-1-one