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3-chloro-N-[2-(dimethylamino)ethyl]-4-{[1-(oxane-4-carbonyl)piperidin-4-yl]oxy}benzamide
2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)-1-[(3R,5S)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]ethan-1-one
3-(2,2-dimethylpropyl)-5-{pyrazolo[1,5-a]pyridine-2-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2-amino-6-(2-amino-4-methyl-1,3-thiazol-5-yl)-4-(1H-indol-3-yl)pyridine-3-carbonitrile
1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
3-benzyl-5-(2,3-dihydro-1-benzofuran-7-yl)-1H-1,2,4-triazole
[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]({[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl})methylamine
(2S)-2-[(5,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)formamido]-4-methanesulfonylbutanoic acid
N-(2-methoxyethyl)-4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]-N-[(4-methylphenyl)methyl]benzamide
4-{[4-(3-methylphenyl)-4H-1,2,4-triazol-3-yl]methyl}morpholine
N-(oxolan-2-ylmethyl)-2-(pyridin-4-yl)-N-(thiophen-3-ylmethyl)pyrimidine-5-carboxamide
(2R,6S)-4-(1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)-2,6-dimethylmorpholine
(4aS,8aR)-1-(3-aminopropyl)-6-[(4-chlorophenyl)methyl]-decahydro-1,6-naphthyridin-2-one
7,8-dimethyl-3-{2-[1-(propan-2-yl)piperidin-2-yl]ethyl}-3,4-dihydroquinazolin-4-one
1-(4-methyl-1,2,5-oxadiazol-3-yl)-4-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazine
3-ethyl-N-[3-(4-methoxyphenoxy)propyl]-N,4-dimethyl-1H-pyrazole-5-carboxamide
4,4-difluoro-1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}piperidine
9-[(1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
4-[(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-methylpyrrolidine-3-carbonyl]piperazin-2-one
N-[(1-ethylpyrrolidin-2-yl)methyl]-2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carboxamide
2-amino-4-[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]-6-(thiophen-2-yl)pyridine-3-carbonitrile
[(dimethyl-1,2-oxazol-4-yl)methyl](methyl){[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]methyl}amine
2-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
4-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-6-methoxypyrimidine
4-[(dimethylamino)methyl]-1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}azepan-4-ol
N-(3-methoxy-2,2-dimethylpropyl)-3-oxo-3,4-dihydroquinoxaline-2-carboxamide
2-(3-{[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]methyl}phenoxy)acetamide
methyl 3-(1-{3,3-dimethyl-2-methylidenebicyclo[2.2.1]heptane-1-carbonyl}piperidin-4-yl)propanoate
N3-cycloheptyl-1-cyclopropyl-N5-(furan-2-ylmethyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-(2-ethoxyethyl)-4-[(3-hydroxyazetidin-1-yl)sulfonyl]benzamide
1-(4-{[2-(3-methoxyphenyl)azetidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
2,2-dimethylpropyl (2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxylate
N-({5-[(2,6-difluoro-4-methoxyphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
4-{[4-(1-hydroxy-3-methylbutyl)piperidin-1-yl]methyl}-1,5-dimethyl-1H-pyrrole-2-carbonitrile
N-cyclopropyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]oxane-2-carboxamide
1-[(5-methylthiophen-2-yl)methyl]-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
{4-[(2-chlorophenyl)methyl]-1-[(6-methoxy-2H-chromen-3-yl)methyl]piperidin-4-yl}methanol
N-methyl-1-(2-phenylethyl)-N-[2-(pyridin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
7-[2-amino-6-(thiophen-2-ylsulfanyl)pyrimidin-4-yl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
(4aR,7aS)-1-(pyrimidin-2-yl)-4-[3-(4H-1,2,4-triazol-4-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[(3-ethyl-1,2-oxazol-5-yl)methyl][(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]methylamine
N-(1-phenylethyl)-4-{4-[(propan-2-yl)amino]piperidin-1-yl}benzamide
N-{[3-methyl-7-(1-methyl-1H-indole-2-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
1-[2-(5-amino-3-methyl-1H-pyrazol-1-yl)acetyl]-N-[3-(4-fluorophenyl)phenyl]piperidine-3-carboxamide
2-[2-(6-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid
2-({3-benzyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}methyl)phenol
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]piperidine
2-(1,2-oxazol-5-yl)-4-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}phenol
N-[(1R,3S)-3-{[2-(propan-2-yloxy)ethyl]carbamoyl}cyclopentyl]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
1-(3-phenylpiperidin-1-yl)-2-(pyridin-4-ylsulfanyl)ethan-1-one