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(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
N-cyclopentyl-N'-methyl-N'-(pyrimidin-4-ylmethyl)butanediamide
5-methyl-2-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine
4-(cyclopropylsulfamoyl)-N-[(1-propyl-1H-pyrazol-4-yl)methyl]benzamide
1-(3-{[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-2-methyl-2-(phenylamino)propan-1-one
(1H-imidazol-2-ylmethyl)(methyl)[1-(pyridin-2-yl)propan-2-yl]amine
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-5-phenoxyfuran-2-carboxamide
N-tert-butyl-2-[2-(1H-imidazol-4-yl)ethyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
dimethyl({5-[2-(pyridin-3-yl)ethyl]-1,2,4-oxadiazol-3-yl}methyl)amine
N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}-2-oxopentanamide
3-{[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]sulfamoyl}-N-(2-fluoroethyl)benzamide
5-methanesulfonyl-N-[(3-methoxyphenyl)methyl]-4-(piperidin-3-yl)pyrimidin-2-amine
N-{[5-(2,6-difluorophenyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(dimethylamino)-4-methylpyrimidine-5-carboxamide
[(1-ethyl-1H-pyrazol-4-yl)methyl][(2-methoxyphenyl)methyl](pyridin-3-ylmethyl)amine
[(5-tert-butyl-1H-pyrazol-3-yl)methyl](methyl)[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amine
2-[3-(2-methoxyethyl)-5-[2-(1H-1,2,4-triazol-1-yl)phenyl]-1H-1,2,4-triazol-1-yl]acetic acid
2-(4-methylpentyl)-4-[2-(morpholin-4-yl)benzoyl]morpholine
6-ethyl-2-methyl-4-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]quinoline
4-(oxane-2-amido)-N-phenylpiperidine-1-carboxamide
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-2-(2-oxopyrrolidin-1-yl)propanamide
5-[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]-N-methyl-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-(3,5-dimethylphenyl)-1-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]propan-1-one
4-(3-fluoro-4-methylbenzoyl)-1-(3-methoxyphenyl)piperazin-2-one
(3aR,6aR)-2-benzyl-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
(4aR,8aS)-1-[2-(3-fluorophenyl)ethyl]-6-(furan-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
2-(3-ethoxyphenyl)benzamide
1-methyl-5-[2-(morpholin-4-ylmethyl)phenyl]-1H-indazole
3-methyl-8-[(3-methylquinoxalin-2-yl)methyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}pyridin-3-ol
3-(2,4-difluorophenyl)-1-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]propan-1-one
ethyl 4-(3-phenylpropyl)-1-(pyridin-4-ylmethyl)piperidine-4-carboxylate
(2S,4S)-4-amino-N-ethyl-1-{[2-methoxy-5-(propan-2-yl)phenyl]methyl}pyrrolidine-2-carboxamide
N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
3-hydroxy-S-[2-(1,2-oxazole-3-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]butane-1-sulfonamido
N-ethyl-2,2-dimethyl-N-(1,3-thiazol-2-ylmethyl)oxan-4-amine
(2S)-N-(2H-1,3-benzodioxol-5-ylmethyl)-5-oxo-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
1-ethyl-2-[1-(pyridin-4-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1H-1,3-benzodiazole
4-(5-acetylpyridin-2-yl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
4-(4-{[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)-6-(1H-pyrazol-1-yl)pyrimidine
1-cyclopropanecarbonyl-4-{4-[3-(methoxymethyl)piperidine-1-carbonyl]phenoxy}piperidine
N-benzyl-1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-N-methylpiperidin-3-amine
6-{[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-[(1-acetylpiperidin-4-yl)oxy]-N-(2,2-dimethyloxan-4-yl)-3-methoxybenzamide
3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-(thiophene-3-carbonyl)piperidine
7-(2-cyclohexylethyl)-2-(5-methyl-1,3-oxazole-4-carbonyl)-2,7-diazaspiro[4.5]decane
3-[1-(cyclohex-3-ene-1-carbonyl)piperidin-4-yl]-1-(4-ethylpiperazin-1-yl)propan-1-one
2-(4-methoxyphenoxymethyl)-N-methyl-N-(quinolin-6-ylmethyl)-1,3-oxazole-4-carboxamide
2-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)-6-(piperidine-1-carbonyl)pyrazine
3-[(carbamoylmethyl)sulfamoyl]-N-[(5-ethylpyridin-2-yl)methyl]benzamide
3,5-dimethyl-N-{[5-(methylcarbamoyl)furan-2-yl]methyl}-1H-indole-2-carboxamide