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1-{2-[4-(furan-3-carbonyl)-1,4-diazepan-1-yl]-2-oxoethyl}-1,2-dihydropyrimidin-2-one
1-{5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carbonyl}azocane
(4aS,8aS)-2-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-decahydro-2,7-naphthyridin-4a-ol
1-(2-aminoethyl)-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
3-{[4-(2,6-diaminopyrimidin-4-yl)piperazin-1-yl]methyl}-7-methylquinolin-2-ol
3-chloro-N-(2-methoxyethyl)-4-({1-[(2-methylphenyl)methyl]piperidin-4-yl}oxy)benzamide
(3S,4S)-4-cyclopropyl-1-{[5-(1H-pyrazol-5-yl)furan-2-yl]sulfonyl}pyrrolidine-3-carboxylic acid
N5-(2-methoxyethyl)-N6-(2-methylprop-2-en-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
5-(hydroxymethyl)-2-methyl-4-{[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}pyridin-3-ol
9-benzoyl-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
(1R,5R)-6-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
1-[4-chloro-1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-4-methanesulfonylpiperazine
N-[2-(1H-imidazol-1-yl)propyl]-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
1-[(3-phenyl-1H-pyrazol-4-yl)methyl]-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
2-methoxy-N-[(5-{[(1s,4s)-4-aminocyclohexyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]acetamide
4-hydroxy-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-2-[(phenylsulfanyl)methyl]pyrimidine-5-carboxamide
(2S)-2-(methoxymethyl)-N-[3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]pyrrolidine-1-carboxamide
2-[(4aS,8aR)-1-butyl-2-oxo-decahydro-1,6-naphthyridine-6-carbonyl]benzonitrile
2-{[5-(4-cyclohexylphenyl)-1,2,4-triazin-3-yl](2-hydroxyethyl)amino}ethan-1-ol
N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
5-{2-[(3-methoxyphenyl)sulfanyl]acetyl}-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-(3-cyano-4-ethoxyphenyl)-4-[(3S,4R)-4-hydroxyoxolan-3-yl]-1,4-diazepane-1-carboxamide
[(3R,4R)-4-[(4-methylpiperazin-1-yl)methyl]-1-(3-propyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-yl]methanol
N-{4,6-dimethyl-[1,2]thiazolo[5,4-b]pyridin-3-yl}-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
(2R,6R)-11-methoxy-4-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-{[(2,3-difluoro-4-methoxyphenyl)methyl]amino}-N-(pyrazin-2-yl)acetamide
4-(4-methoxypyrimidin-2-yl)-N-(1-oxo-2,3-dihydro-1H-inden-5-yl)piperazine-1-carboxamide
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-methyl-1,3-oxazole-5-carboxamide
4-[3-(2,4-difluorophenyl)propanoyl]-1-(2-methylphenyl)piperazin-2-one
1-[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-1,2,4-triazol-5-yl]piperidine
5-{[1-ethyl-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-5-yl]methyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-cyclopropyl-3-(piperidine-1-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(ethanesulfonyl)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-6-one
N-(oxolan-2-ylmethyl)-4-[({[(propan-2-yl)carbamoyl]methyl}carbamoyl)amino]benzamide
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-1-[3-(2-fluorophenyl)pyrrolidin-1-yl]propan-1-one
4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-(1-methylcyclopropanecarbonyl)piperidine
(4aR,7aS)-1-(2-methoxyethyl)-4-(4-methylpent-3-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-{2-[cyclohexyl(methyl)amino]pyridine-3-carbonyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
7-(4-fluorophenyl)-2-[1-(2-methoxyethyl)piperidin-4-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-({3-methyl-3,9-diazaspiro[5.6]dodecan-9-yl}methyl)pyridin-2-amine
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-[(2-methoxyethyl)(methyl)amino]pyridine-3-carboxamide
2-[(1-{2,7-dimethylimidazo[1,2-a]pyridine-3-carbonyl}piperidin-4-yl)oxy]pyrimidine
2-ethyl-N,N-dimethyl-4-phenyl-2,9-diazaspiro[5.5]undecane-9-sulfonamide
[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl][(4-methanesulfonylphenyl)methyl]methylamine
N-methyl-1-[(2-methyl-1,3-thiazol-5-yl)methyl]-N-(2-phenylethyl)piperidin-3-amine
2-{6-[2-(dimethylamino)phenyl]pyridin-3-yl}acetic acid
N-butyl-2-(dimethylamino)-2-(4-fluorophenyl)-N-(pyridin-4-ylmethyl)acetamide
N-ethyl-4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxamide
8-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one