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5-methoxy-4-(1-methyl-1H-pyrazol-5-yl)-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]pyrimidin-2-amine
N-[(2,3-difluorophenyl)methyl]-4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-[2-(dimethylamino)ethyl]-N-[(3-methylthiophen-2-yl)methyl]oxane-2-carboxamide
8-(2,3-dihydro-1H-inden-2-yl)-1-[2-(4-methoxyphenyl)ethyl]-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-cyclopropyl-N-ethyl-N-(pyridin-4-ylmethyl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
5-({[3-(5-fluoro-2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}sulfanyl)-1,3,4-thiadiazol-2-amine
3-(2-fluoro-4,5-dimethoxyphenyl)-[1,2,4]triazolo[4,3-a]pyridine
(3aS,6aR)-5-[(2-aminopyridin-3-yl)methyl]-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
(2S)-2-{3-[5-oxo-2-(thiophen-2-ylmethyl)pyrrolidin-2-yl]propanamido}-3-phenylpropanamide
2-[3-(4-phenoxybenzoyl)piperidine-1-carbonyl]pyridine
1-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-N-[1-(1-methyl-1H-imidazol-2-yl)butyl]piperidin-4-amine
1-(2-methoxyethyl)-4-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
6-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-2-methyl-1,3-benzoxazole
N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-1-(oxan-4-yl)piperidine-4-carboxamide
N-[(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
ethyl 4-{[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]carbamoyl}-3,5-dimethyl-1H-pyrrole-2-carboxylate
3-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-1-(3,4,5-trimethoxyphenyl)urea
N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-5-(oxolan-2-yl)thiophene-2-carboxamide
N-(3-phenylprop-2-yn-1-yl)-N-(prop-2-en-1-yl)thiophene-3-carboxamide
(2S)-2-{[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)carbamoyl]amino}-3-(4-hydroxyphenyl)propanamide
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]({[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl})methylamine
N3-[3-(4-hydroxyphenyl)propyl]-N1,N1-dimethylpiperidine-1,3-dicarboxamide
5-methyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
1-[2-(4-methoxyphenyl)ethyl]-3-(propan-2-yl)-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-{[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]propanamide
4-[3-(2,6-dimethylphenoxy)azetidin-1-yl]-6-methyl-5-(prop-2-en-1-yl)pyrimidin-2-amine
4-{2-[(cyclopropylmethyl)sulfanyl]acetyl}-1-[(3-fluorophenyl)methyl]piperazin-2-one
1-butyl-4-{2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperazine
N-cyclopentyl-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
N-(1-acetylpiperidin-3-yl)-7-chloro-3,5-dimethyl-1-benzofuran-2-carboxamide
1-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]pyrrolidin-3-amine
[(1-methylpiperidin-3-yl)methyl](2-phenylethyl){[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}amine
3-[3-(dimethylamino)propyl]-8-[(1-propyl-1H-imidazol-2-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[(2-methoxyphenyl)methyl]-6-(1-methylpiperidin-3-yl)-3,4-dihydropyrimidin-4-one
(5S)-5-{3-cyclopentyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}pyrrolidin-2-one
[(3S,5R)-5-[(dimethylamino)methyl]-1-{[3-(pyridin-2-ylmethoxy)phenyl]methyl}piperidin-3-yl]methanol
N,1-dimethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-{5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]-1H-pyrazol-3-yl}phenol
1-[(3S,4R)-1-[3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)propanoyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-(4-fluorophenyl)-N-(2-{4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)benzamide
3-(3-fluorophenyl)-N-methyl-N-(oxan-2-ylmethyl)-1H-pyrazole-4-carboxamide
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-2-methanesulfonylacetamide
6-fluoro-2-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)quinolin-4-ol
N-[(1-benzylpiperidin-4-yl)methyl]-N-methyl-2-oxo-1H,2H,5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-(4-methanesulfonylphenyl)-4-methoxypyrimidine
3-{2-[4-(benzyloxy)piperidin-1-yl]-2-oxoethyl}-4-(furan-3-ylmethyl)piperazin-2-one
methyl 5-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate