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1-[1,3-dioxo-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-methyl-N-(thiophen-2-ylmethyl)piperidine-4-carboxamide
2-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyridine-3-carboxamide
N,N-dimethyl-5-{[4-(pyrimidin-2-yloxy)piperidin-1-yl]methyl}pyridin-2-amine
2-{[4-(4-acetylphenyl)-5-(4-methyl-1H-imidazol-5-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
dimethyl(3-{2-[1-(5-methylpyridin-2-yl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)amine
(3R,4S)-1-(4-chloro-3-methylbenzoyl)-4-cyclopropylpyrrolidin-3-amine
(1S,6R)-9-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]acetyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
2-(2,3-dihydro-1H-indol-1-yl)-N-(4H-1,2,4-triazol-4-yl)acetamide
4-({2-[1-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
N-[(3S,5S)-1-[(2-aminopyridin-3-yl)methyl]-5-(ethylcarbamoyl)pyrrolidin-3-yl]pyridine-2-carboxamide
(1S,5R)-3-[2-(3-hydroxyphenyl)acetyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[(2-fluorophenyl)formamido]-N-[2-(morpholin-4-yl)ethyl]propanamide
1-{5-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]thiophen-2-yl}ethan-1-one
2-cyclopropyl-9-(1-methylpiperidin-4-yl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
2-[(4-benzylpiperazin-1-yl)methyl]-N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]-1,3-oxazole-4-carboxamide
4-ethyl-3-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{2-hydroxy-3-[4-methoxy-2-({[3-(1H-pyrazol-1-yl)propyl]amino}methyl)phenoxy]propyl}piperidin-4-ol
2-[2-(3-methoxypropyl)piperidine-1-carbonyl]benzonitrile
3-{2-[(4-methylphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]propanamide
N4-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-N4,N6,N6-trimethylpyrimidine-4,6-diamine
1-(diethylamino)-3-(2-methoxy-5-{[methyl(pyridin-3-ylmethyl)amino]methyl}phenoxy)propan-2-ol
1-{2-[1-(4-methyl-1,3-thiazol-2-yl)piperidin-4-yl]ethyl}pyrrolidin-2-one
4-methoxy-N-{2-[7-(3-methylbutyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}benzamide
6-{[(3R,4S)-4-cyclopropyl-1-(oxan-4-yl)pyrrolidin-3-yl]amino}-N,N-dimethylpyrazine-2-carboxamide
N-butyl-N-(furan-2-ylmethyl)-3-oxo-2,3-dihydro-1H-indene-1-carboxamide
1-(4-{[methyl(thian-4-yl)amino]methyl}phenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
5-{[(4-methoxynaphthalen-1-yl)oxy]methyl}-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1,2-oxazole-3-carboxamide
4-[1-(2-propyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]thiomorpholine
4-{1-benzyl-5-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}morpholine
(3aS,6aS)-1-oxo-2-(prop-2-en-1-yl)-5-(quinoxalin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(2,3-dihydro-1H-inden-1-yl)-N-methyl-N-[2-(pyridin-2-yl)ethyl]acetamide
ethyl 4-[(3-fluorophenyl)methyl]-1-(pyridin-3-ylmethyl)piperidine-4-carboxylate
N-(2-fluoroethyl)-4-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzamide
1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
1-(2,3-dihydro-1-benzofuran-5-carbonyl)-4-[(dimethylamino)methyl]azepan-4-ol
N-({5-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
N-[3-(4-methoxyphenyl)propyl]-6-(4-methylpiperazin-1-yl)pyridine-3-carboxamide
2-[4-fluoro-3-(hydroxymethyl)phenyl]-2-{1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}acetic acid
1-(1-methylpiperidin-4-yl)-3-(pyrrolidine-1-carbonyl)piperidine
2-{3-[3-(3-methoxypyridin-2-yl)phenyl]-1H-pyrazol-1-yl}-N-(pyrazin-2-yl)acetamide
3-chloro-N-cyclopentyl-4-{[1-(3,5-dimethylfuran-2-carbonyl)piperidin-4-yl]oxy}benzamide
3-[2-(methylamino)acetamido]-N-(naphthalen-1-yl)propanamide
{3-[2-(1-cycloheptanecarbonylpiperidin-3-yl)-1H-imidazol-1-yl]propyl}dimethylamine
4-[(2,3-difluoro-6-methoxyphenyl)methyl]-1-methylpiperazine-2-carboxylic acid
(2R,6S)-2,6-dimethyl-4-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}morpholine
3-methyl-1-{3-[(2-methylpiperidin-1-yl)methyl]phenyl}-3-(prop-2-en-1-yl)urea
4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
(3S,4R)-N,N-dimethyl-1-(2-phenylethyl)-4-propylpyrrolidin-3-amine
(3R,4S)-4-(propan-2-yl)-1-(pyridine-3-sulfonyl)pyrrolidin-3-amine
1-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]-2-(1,3-thiazol-4-yl)ethan-1-one