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1-{3-[1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenyl}-1H-pyrazole
1-[(2S)-1-hydroxy-3-phenylpropan-2-yl]-3-[3-(2-oxopyrrolidin-1-yl)phenyl]urea
(3R,5S)-1-benzyl-N-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(4-hydroxyphenyl)ethan-1-one
2-(piperidin-1-yl)-5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridine
2-[8-(3-hydroxypropyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]-6-methylpyridine-3-carbonitrile
2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(pyridin-3-yl)ethyl]acetamide
3-({4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}methyl)pyridin-2-amine
4-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-4-yl)thiomorpholine
N-[(3S,5S)-5-(diethylcarbamoyl)-1-[2-(methylsulfanyl)acetyl]pyrrolidin-3-yl]-1H-pyrazole-3-carboxamide
2-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}-2-(4-fluoro-3-methylphenyl)acetic acid
2-(2-methoxyethyl)-9-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
3-(2-methylphenyl)-3-phenyl-1-(thiomorpholin-4-yl)propan-1-one
N-(2-hydroxyethyl)-4-oxo-4-phenyl-N-[(2E)-3-phenylprop-2-en-1-yl]butanamide
8-(5-hydroxypyrazine-2-carbonyl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
dimethyl[(4-methyl-5-{1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]piperidin-3-yl}-4H-1,2,4-triazol-3-yl)methyl]amine
(3aR,5S,6S,7aS)-2-(7-methyl-2,3-dihydro-1,4-benzodioxine-6-carbonyl)-octahydro-1H-isoindole-5,6-diol
N-[(2-methylphenyl)(pyridin-4-yl)methyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
N-ethyl-3-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
N-(2-{3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}ethyl)pyridine-3-carboxamide
N-(2-methanesulfonylethyl)-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
2-[5-(1-methylpiperidine-3-carbonyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
5-methyl-3-(1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-1,2-oxazole
methyl[3-(methylsulfanyl)butyl]{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}amine
N-cyclopropyl-N-(1H-indol-5-ylmethyl)-4-(1H-pyrazol-3-yl)benzamide
N-[(3-fluoro-4-methylphenyl)methyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
2-[1-benzyl-4-(1H-indazole-3-carbonyl)piperazin-2-yl]ethan-1-ol
N-[2-(2-fluorophenyl)ethyl]-6-[4-(furan-2-carbonyl)piperazine-1-carbonyl]-5-methylthieno[2,3-d]pyrimidin-4-amine
(2S,4R)-N-ethyl-1-(furan-3-ylmethyl)-4-[2-(4-methyl-1H-pyrazol-1-yl)acetamido]pyrrolidine-2-carboxamide
[(4-methoxy-2,3-dimethylphenyl)methyl](methyl)[1-(pyridin-2-yl)ethyl]amine
1-{[2-methyl-5-(1,2-oxazol-5-yl)furan-3-yl]sulfonyl}azepan-4-amine
N-[(3R,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]naphthalene-2-carboxamide
N-(furan-2-ylmethyl)-2-[(2-methylpyrrolidin-1-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
10-methoxy-5-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
(3aR,5S,6S,7aS)-2-[(3-phenoxyphenyl)methyl]-octahydro-1H-isoindole-5,6-diol
({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(ethyl)(2-methylprop-2-en-1-yl)amine
1-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]-2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
1-[(2-methyl-1,3-thiazol-5-yl)methyl]-3-[4-(methylsulfanyl)benzoyl]piperidine
1-{2-[(4-chlorophenyl)methyl]-1,3-benzoxazole-5-carbonyl}piperidine-3-carboxamide
N-({3-[3-(dimethylamino)propoxy]-4-methoxyphenyl}methyl)-N-(pyridin-3-ylmethyl)cyclopropanecarboxamide
8-(3-phenoxybenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
4-[1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-2-[4-(propan-2-yl)phenyl]pyridine
1'-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
4-({[4-(dimethylsulfamoyl)phenyl]methyl}amino)pyrimidine-5-carboxylic acid
5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-(1-methoxypropan-2-yl)pyridin-2-amine
5-(3,4-difluorophenoxymethyl)-N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1,2-oxazole-3-carboxamide
2-[1-(thiophene-2-carbonyl)piperidin-4-yl]-2,8-diazaspiro[4.5]decane
[3-(2-methoxyethyl)-1-(1-methyl-1H-pyrazole-3-carbonyl)piperidin-3-yl]methanol
1-(3,5-dimethylphenyl)-4-(2-propyl-1,3-thiazole-4-carbonyl)piperazin-2-one
9-[2-(3-methyl-1H-1,2,4-triazol-5-yl)acetyl]-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one