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3-(3-methyl-1H-1,2,4-triazol-5-yl)-1-(3-phenylpropyl)piperidine
ethyl 2,4-dimethyl-5-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonane-9-carbonyl]-1H-pyrrole-3-carboxylate
N-[2-(dimethylsulfamoyl)ethyl]-1-(propan-2-yl)piperidine-3-carboxamide
(1R,2S)-1-({2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-2,3-dihydro-1H-inden-2-ol
5-ethyl-6-methyl-2-[4-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
N-[3-(4-fluorophenyl)propyl]-2-methyl-1H-imidazole-4-carboxamide
N,N,2-trimethyl-7-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
6-{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-3-yl}-2-methylpyrimidin-4-ol
1-methyl-6-(pyridin-4-yl)-N-(pyridin-4-ylmethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-{[6-(3-fluoro-4-methoxyphenyl)pyridazin-3-yl](methyl)amino}ethan-1-ol
N-({1-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]pyrrolidin-3-yl}methyl)methanesulfonamide
3-(2-methoxyphenyl)-N-[2-(propane-2-sulfonyl)ethyl]-1H-pyrazole-5-carboxamide
2-cyclopropyl-1-{4-[4-(2-hydroxypropan-2-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}ethan-1-one
N-[(4-methyl-1,3-thiazol-2-yl)methyl]-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetamide
3-methyl-8-(6-methyl-2-propylpyrimidin-4-yl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
5-[methyl(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)amino]-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
1-(2H-1,3-benzodioxol-5-ylmethyl)-6-methyl-4-oxo-2-propyl-N-[1-(thiophen-2-yl)propyl]-1,4-dihydropyridine-3-carboxamide
6-[(3R,4R)-3-{[ethyl(2-hydroxyethyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]pyridine-2-carbonitrile
N-cyclopropyl-N-({4-[3-(dimethylamino)propoxy]phenyl}methyl)cyclobutanecarboxamide
(1R,9aR)-N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-octahydro-1H-quinolizine-1-carboxamide
(3S,9aR)-8-[(2-fluoro-5-methylphenyl)methyl]-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-[3-(4-phenyl-4H-1,2,4-triazol-3-yl)propyl]morpholine
[(4aS,8aR)-6-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-1-(furan-3-ylmethyl)-decahydro-1,6-naphthyridin-4a-yl]methanol
2-(diethylamino)-N-[2-(dimethylamino)ethyl]-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)acetamide
(2S,4S)-4-amino-N-(propan-2-yl)-1-(2,3,4,9-tetrahydro-1H-carbazole-7-carbonyl)pyrrolidine-2-carboxamide
4-{2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1-benzofuran-5-yl}-1-[(4-methoxy-3-methylphenyl)methyl]piperidin-4-ol
5-{2-[(4aS,7aR)-4-(cyclopropylmethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-(propan-2-yl)-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
9-(cyclopropylmethyl)-4-[(4-ethoxyphenyl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
8-{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-oxa-8-azaspiro[4.6]undecan-9-one
2-[9-oxo-8-(2-phenylethyl)-2,8-diazaspiro[5.5]undecane-2-carbonyl]benzonitrile
2-(1-methylcyclopropanecarbonyl)-N-(2-phenoxyethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
2-(1-benzothiophen-3-yl)-6-(piperidine-1-carbonyl)pyrazine
4-[3-(2-fluorophenoxy)azetidine-1-carbonyl]-1-(propan-2-yl)piperidine
9-ethyl-4-{[3-(furan-2-yl)phenyl]methyl}-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
4-benzyl-1-cyclohexanecarbonyl-1,4-diazepan-5-one
N,5-dimethyl-N-(quinoxalin-2-ylmethyl)-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
3-[1-(thiophene-2-carbonyl)piperidin-3-yl]-N-[4-(trifluoromethyl)phenyl]propanamide
2-[(3S,4R)-3-cyclopropyl-4-(oxane-4-amido)pyrrolidin-1-yl]pyridine-3-carboxamide
6-(5-fluoro-2-methylphenyl)-N,N-dimethylpyridine-2-carboxamide
4-{4-[3-(2H-1,3-benzodioxol-5-yl)-2-methylpropyl]piperazin-1-yl}-6-methylpyrimidin-2-amine
3-{[(3S,4S)-3-(dimethylamino)-4-hydroxypyrrolidin-1-yl]methyl}benzoic acid
2-oxo-8-[3-(prop-2-en-1-yloxy)benzoyl]-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-cyclopropyl-2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-(4-fluorobenzenesulfonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
1-(4-{[4-(1-hydroxyethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-2-(1-methyl-1H-pyrrol-3-yl)ethan-1-one
2-{2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-2,3-dihydro-1H-isoindol-1-one
2-(2,2-dimethylpropanamido)-5-methyl-N-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]thiophene-3-carboxamide
2-[(4-methoxyphenyl)methyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
4-fluoro-N-[(1-{imidazo[1,2-a]pyrimidine-2-carbonyl}piperidin-3-yl)methyl]benzamide