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4-methanesulfonyl-2-({4-[3-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazol-1-yl}methyl)morpholine
2-[4-(4-chlorophenyl)-4-hydroxypiperidin-1-yl]-2-(4-fluorophenyl)acetic acid
4-{1-[2-(2-hydroxyethyl)phenyl]-1H-imidazol-2-yl}-N-methylbenzene-1-sulfonamide
1-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propan-1-one
1-[3-(benzyloxy)azetidin-1-yl]-4-(piperidin-1-yl)butan-1-one
N-({4-[(3-phenylpropyl)amino]quinazolin-2-yl}methyl)propane-2-sulfonamide
N,2-dimethyl-N-{[3-(methylsulfanyl)phenyl]methyl}-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}[2-(1H-imidazol-1-yl)ethyl]methylamine
N-[(2-ethoxyphenyl)methyl]-N-(prop-2-en-1-yl)-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
5-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonitrile
N-[(4-fluorophenyl)methyl]-1-methyl-5-[(pyridin-4-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
7-(3-chlorophenyl)-4-cyclopropanecarbonyl-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[2-(4-methoxyphenyl)ethyl]-6-methyl-N-(pyridin-2-ylmethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-methyl-1-[(3-methylpyridin-4-yl)methyl]-3-[4-(propylsulfamoyl)phenyl]urea
1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-[5-(furan-2-yl)-1,3,4-thiadiazol-2-yl]urea
4-(1-{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)thiomorpholine
1-cyclopropyl-4-[4-(2-methoxyphenyl)piperazine-1-carbonyl]pyrrolidin-2-one
N-(pyridin-4-ylmethyl)-4-[4-(thiophen-2-yl)butanoyl]morpholine-2-carboxamide
3-[1-({10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
5-fluoro-2-(1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}pyrrolidin-2-yl)-1H-1,3-benzodiazole
N-ethyl-5-methyl-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-{2-[(3-methylpyridin-2-yl)amino]ethyl}-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
N-methyl-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-cyclopropyl-4-methoxy-2-{[1-(4-phenylbutan-2-yl)piperidin-4-yl]oxy}benzamide
2-(cyclopropanesulfonyl)-7-{[2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}-1,2,3,4-tetrahydroisoquinoline
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]-4-phenoxybutan-1-one
N-(2-methoxyethyl)-2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}-N-(1,3-thiazol-2-ylmethyl)acetamide
N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
1-cyclobutyl-3-(6-methoxynaphthalene-2-carbonyl)piperidine
4-(2-methoxyethyl)-N-(3-phenyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
2-(4-{[4-(3-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]methyl}-3-methyl-1H-pyrazol-1-yl)ethan-1-ol
methyl({[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}){[3-(trifluoromethyl)phenyl]methyl}amine
N-(3-methoxyphenyl)-3-[(3S,4R)-1-(propan-2-yl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanamide
1-[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-7-yl]-3-(piperazin-1-yl)propan-1-one
N-[(2-chlorophenyl)methyl]-N-(2-methoxyethyl)-4,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
6-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]pyridin-3-ol
ethyl 2-{1-[2-(phenylformamido)acetyl]piperidin-2-yl}acetate
4-(3-cyclopropyl-5-{[(4-methyl-1,3-thiazol-2-yl)sulfanyl]methyl}-1H-1,2,4-triazol-1-yl)-3-methylpyridine
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
3-(3-chlorophenyl)-3-(3-hydroxyphenyl)-N-methyl-N-(oxan-4-yl)propanamide
N-[(2-chlorophenyl)methyl]-N-(propan-2-yl)quinoxaline-6-carboxamide
N-[2-(dimethylamino)-1-phenylethyl]-4-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
1-(4-chlorophenyl)-N-[2-(4-methyl-5-{[2-(morpholin-4-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]cyclobutane-1-carboxamide
ethyl 1-[5-(methoxymethyl)furan-2-carbonyl]-4-(2-phenylethyl)piperidine-4-carboxylate
1-(3,5-dimethylphenyl)-4-[(1R,2R)-2-phenylcyclopropanecarbonyl]piperazin-2-one
N-[(4-chlorophenyl)methyl]-2-cyclopropanecarbonyl-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
(3R,4R)-4-cyclobutyl-1-[3-(dimethylamino)pyrazin-2-yl]-3-methylpiperidin-4-ol
N-[3-(2,6-dimethoxyphenyl)phenyl]acetamide
[(2-cyclohexylpyrimidin-5-yl)methyl][1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]methylamine
2-[methyl({4-methyl-5-[1-(oxane-4-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amino]ethan-1-ol