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4-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-2-one
N-{2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}pyridine-4-carboxamide
2-(dimethylamino)-2-(2-methylphenyl)-1-{3-oxa-9-azaspiro[5.5]undecan-9-yl}ethan-1-one
3-(5-chloropyrazin-2-yl)quinoline
(2E)-N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]-3-(thiophen-2-yl)prop-2-enamide
5-(3-chlorothiophen-2-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-(2-oxopyrrolidin-1-yl)benzamide
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxy-N-[2-(3-methylpyridin-2-yl)ethyl]benzamide
methyl 6-[(2,4-difluorophenyl)methyl]-2-(ethylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-(5-methylpyrimidin-2-yl)-9-oxa-2-azaspiro[5.5]undecane
1-(2-cyclooctyl-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl)-N-(2-hydroxyethyl)piperidine-4-carboxamide
2-[4-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)piperidin-1-yl]acetamide
4-[3-({1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}oxy)benzoyl]morpholine
N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-(1H-pyrazol-4-yl)butanamide
2-[(3-methylquinoxalin-2-yl)methyl]-2-azaspiro[4.5]decan-3-one
1-(4-fluorophenyl)-3-[2-(methylsulfanyl)ethyl]-5-(1,3-thiazol-4-ylmethyl)-1H-1,2,4-triazole
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}oxane-4-carboxamide
2-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-4-yl)-1,2,3,4-tetrahydroisoquinoline
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-(2-methoxyethyl)-N-methylpiperidine-3-carboxamide
{1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(2-methoxyethyl)piperidin-3-yl}methanol
(2S,4S)-4-(cyclooctylamino)-1-{[4-(diethylamino)phenyl]methyl}-N-methylpyrrolidine-2-carboxamide
1-[(1-ethylpiperidin-4-yl)methyl]-4-(pyrrolidin-1-yl)piperidine
2-[1-(2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-1,3-oxazol-4-yl)-N-methylformamido]-N-methylpropanamide
4-[(4-cyclohexyl-3-oxopiperazin-1-yl)methyl]benzoic acid
N-({1-[6-amino-2-(morpholin-4-yl)pyrimidin-4-yl]piperidin-4-yl}methyl)acetamide
7-[3-(2-ethoxyethoxy)benzoyl]-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[2-(2,2-dimethyl-4-phenyloxan-4-yl)ethyl]-6-methyl-4-oxo-4H-pyran-2-carboxamide
2-methoxy-1-(4-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}piperidin-1-yl)ethan-1-one
1-(4-cyclopentyl-1,4-diazepan-1-yl)-4-(4-fluorophenyl)butane-1,4-dione
(3R,4R)-1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-methyl-3-(propan-2-yl)pyrrolidin-3-ol
2-[2-(dimethylamino)ethyl]-9-(oxolane-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(ethyl)(pyridin-4-ylmethyl)amine
N-[(2S)-1-hydroxybutan-2-yl]-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
1-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]-2-methoxyethan-1-one
1-cyclopropyl-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-6-oxopiperidine-3-carboxamide
[(5-cyclopropyl-1H-pyrazol-3-yl)methyl][(2,3-difluoro-6-methoxyphenyl)methyl]methylamine
4-{[(6-amino-2-methylpyrimidin-4-yl)amino]methyl}-1-phenylpyrrolidin-2-one
5-{[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
ethyl 5-(1H-indol-3-ylmethyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-(3,5-dimethyl-1H-pyrazol-4-yl)-5-(piperidine-1-carbonyl)pyridine
N-{2-[(5-acetylthiophen-3-yl)formamido]ethyl}pyridine-3-carboxamide
2-(4-fluorophenyl)-N-(2-{7-[(2-phenyl-1,3-thiazol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)acetamide
2-cyclopropyl-5-[4-(2-methoxyphenyl)-2-methylpiperazine-1-carbonyl]-3,4-dihydropyrimidin-4-one
1-{4-[4-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-3,5-dimethyl-1H-pyrrol-2-yl}ethan-1-one
N-{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-2-ethoxyacetamide
N-{[3-(difluoromethoxy)phenyl]methyl}-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
{[2-(cyclopentyloxy)phenyl]methyl}[(1-ethyl-1H-imidazol-2-yl)methyl]methylamine
3-{[3-methyl-4-(propan-2-yl)piperazin-1-yl]methyl}benzonitrile
N-cyclohexyl-3-{[4-(piperidin-3-yl)phenyl]formamido}propanamide