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2-ethyl-N-{[6-(trifluoromethyl)pyridin-3-yl]methyl}-2H-1,2,3,4-tetrazol-5-amine
4-{3-[(5-methylpyridin-2-yl)amino]propyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-amino-4-ethyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1,3-thiazole-5-carboxamide
N-{2-[2-(9-ethyl-9H-carbazol-3-yl)-1H-imidazol-1-yl]ethyl}acetamide
3-{[5-(1H-pyrazol-5-yl)thiophen-2-yl]methyl}-3,9-diazaspiro[5.5]undecane
(2S)-2-amino-N-(2,3-dihydro-1H-inden-2-yl)-3-(1H-imidazol-4-yl)-N-methylpropanamide
ethyl 3-({3-[2-(methylsulfanyl)benzoyl]piperidine-1-carbonyl}amino)propanoate
2-[4-({[(8-methoxyquinolin-5-yl)methyl](methyl)amino}methyl)-3-methyl-1H-pyrazol-1-yl]ethan-1-ol
3-(pentan-2-yl)-8-(3-propyl-1H-pyrazole-5-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(2-{[(4-ethyl-1,3-thiazol-2-yl)methyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
4-(6-methoxypyridin-3-yl)-1-methyl-3-phenyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
7,7-dimethyl-2-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-yl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2,6-dimethyl-N-[2-(propylsulfanyl)ethyl]pyridine-4-carboxamide
N-cyclopropyl-N-{[6-(2,5-dimethoxyphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-5-methylthiophene-2-carboxamide
8-(3,6-dimethyl-1-benzofuran-2-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-(1,4-oxazepan-6-ylmethyl)-3-(trifluoromethyl)pyridin-2-amine
3-[3-(naphthalene-2-carbonyl)piperidine-1-carbonyl]pyridine
7-methoxy-5-(1H-pyrazol-4-yl)-1-benzofuran-2-carboxylic acid
1-(2-chloro-4-fluorobenzoyl)-3-(1-ethyl-1H-imidazol-2-yl)piperidine
N-(3-chlorophenyl)-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carboxamide
3-({1-[6-(4H-1,2,4-triazol-4-yl)pyridine-2-carbonyl]pyrrolidin-3-yl}methyl)benzamide
4-{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}piperazin-2-one
8-fluoro-2-{[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]methyl}quinoline
2-methyl-1-[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-1,4-diazepan-5-one
2-methoxy-5-[2-({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]phenol
1-[(3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}-2,5-dimethylphenyl)methyl]-2-methylpiperidine
3-[(4-fluorophenyl)methyl]-5-methyl-5-(1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
(3S,4R)-3-methoxy-1-(9H-purin-6-yl)piperidin-4-amine
1-[(3,5-dimethylphenyl)methyl]-4-[2-(1H-pyrazol-1-yl)acetyl]piperazin-2-one
1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
(2E)-1-{4-[4-(2-aminopropan-2-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-3-(pyridin-3-yl)prop-2-en-1-one
N-[2-({1H-pyrrolo[2,3-b]pyridin-6-yl}amino)ethyl]pyridine-4-carboxamide
5-ethyl-2,3-dimethyl-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)pyrazolo[1,5-a]pyrimidin-7-amine
5-(3-benzyl-1,2,4-oxadiazol-5-yl)-2-[4-(methoxymethyl)piperidin-1-yl]pyridine
3-(4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}benzenesulfonyl)propanoic acid
N-(3-methoxyphenyl)-3-[1-(thiolan-3-yl)piperidin-4-yl]propanamide
N-{imidazo[1,2-a]pyrazin-3-ylmethyl}-4-sulfamoylbenzamide
N-[(2,5-dimethoxyphenyl)methyl]-2-methyl-3-[(pyridin-3-ylmethyl)amino]benzamide
N-benzyl-N-methyl-1-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}piperidin-3-amine
(2R,3R)-1'-[2-(hydroxymethyl)pyridin-4-yl]-3-(pyrrolidin-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-methyl-4-(4-{[3-(pyridin-2-yl)azetidin-1-yl]methyl}phenyl)butan-2-ol
(3S,4R)-1-(4-methoxy-2-methylbenzoyl)-4-phenylpyrrolidine-3-carboxylic acid
1-[(1-{6-[(2-methoxyethyl)(methyl)amino]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
N-{4-[(4-phenyl-4H-1,2,4-triazol-3-yl)methyl]piperidine-1-carbonyl}benzamide
1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-(oxolan-2-ylmethyl)piperazine
N-cyclopropyl-4-methoxy-2-({1-[(5-methylthiophen-2-yl)methyl]piperidin-4-yl}oxy)benzamide
N-[2-(4-chlorophenyl)-2-(pyrrolidin-1-yl)ethyl]-3-ethyl-1H-pyrazole-4-carboxamide
1-(oxolan-3-ylmethyl)-N-[3-(1H-pyrazol-5-yl)phenyl]piperidine-4-carboxamide
1-cyclopentyl-4-[2-(4-phenylazepane-1-carbonyl)-1-benzofuran-5-yl]piperidin-4-ol
2-ethyl-8-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]-2,8-diazaspiro[5.5]undecan-3-one