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(1S,5R)-6-(4-ethenylbenzoyl)-3-methyl-3,6-diazabicyclo[3.2.2]nonane
(3S,4R)-1-(piperidine-1-sulfonyl)-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-4,4,4-trifluorobutanamide
3-[1-(cyclohex-3-ene-1-carbonyl)piperidin-4-yl]-N-[(4-fluorophenyl)methyl]propanamide
4-ethyl-5-{[2-(furan-3-yl)-1H-imidazol-1-yl]methyl}-2-methyl-1,3-thiazole
1-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
1-(3-benzoylpiperidin-1-yl)-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
1-[1-butyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]-2-methylpropan-1-ol
1-(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(pyridin-2-ylmethyl)-1,4-diazepane
5-{3-[2-(3,4-difluorophenyl)ethyl]piperidine-1-carbonyl}-N-(propan-2-yl)pyrimidin-2-amine
2-(1H-pyrazol-1-yl)-1-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)ethan-1-one
1-(4-{[4-(1-hydroxyethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-3-(2-methylphenyl)propan-1-one
5-[1-(2,3-dihydro-1H-inden-2-yl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]-1-methyl-1,2-dihydropyridin-2-one
1-(2-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}-4-fluorophenyl)ethan-1-one
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-1-benzoxepine-4-carboxamide
7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
6-(1-benzylpyrrolidin-3-yl)-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
5-{3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidine-1-carbonyl}-1H-indole
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-(6-oxo-1,6-dihydropyridazin-3-yl)propanamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-(morpholin-4-yl)pyrimidine-5-carboxamide
4-methyl-2-(1-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)-1H-1,3-benzodiazole
N-{[(2S,4S)-4-fluoro-1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]pyrrolidin-2-yl]methyl}cyclobutanecarboxamide
2-[(1-acetylpiperidin-4-yl)oxy]-5-methoxy-N-(oxolan-2-ylmethyl)benzamide
4-(4-methoxyphenyl)-1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-2-methylpiperazine
(2S,4S)-4-amino-N,N-diethyl-1-[(2-methyl-1-benzothiophen-3-yl)methyl]pyrrolidine-2-carboxamide
4,6-dimethyl-2-{1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-3-carbonitrile
3-{5-[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}phenol
1-[2-methoxy-1-(pyridin-2-yl)ethyl]-1-methyl-3-[2-(piperidin-1-ylmethyl)phenyl]urea
ethyl 4-{[3-(2-hydroxyethyl)-4-(2-phenylethyl)piperazin-1-yl]methyl}-1H-pyrazole-3-carboxylate
2-(1H-1,3-benzodiazol-2-yl)-N-[(2-methoxyphenyl)methyl]-N-propylacetamide
N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(piperidin-4-yl)piperidine
N-(1,3-dimethyl-1H-pyrazol-5-yl)-3-{[ethyl(oxolan-2-ylmethyl)amino]methyl}benzamide
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-(2-methylpyrimidin-4-yl)pyrrolidin-3-yl]acetamide
2-(3,5-dimethyl-1H-pyrazol-1-yl)-8-(4H-1,2,4-triazol-4-yl)quinoline
1-{5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1H-pyrazole-3-carbonyl}-2-methyl-1,4-diazepan-5-one
1-(3-chloro-2-fluorophenyl)-3-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}urea
2-(dimethylamino)-2-(2-fluorophenyl)-N-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]acetamide
N-[(1R,3R)-3-aminocyclopentyl]-3-sulfamoylthiophene-2-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
6-[1-(2,8-dimethylquinoline-4-carbonyl)piperidin-3-yl]-2-methylpyrimidin-4-ol
N-[(3R,5S)-5-(ethylcarbamoyl)-1-[2-(methylsulfanyl)acetyl]pyrrolidin-3-yl]-5-methyl-1,3-oxazole-4-carboxamide
1-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]-3-(methylsulfanyl)propan-1-one
2-({1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazol-4-yl}formamido)-N-(1,3-thiazol-2-yl)acetamide
2-[ethyl(methyl)amino]-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}acetamide
1-(1H-imidazol-4-ylmethyl)-N-[2-(4-methoxyphenyl)phenyl]pyrrolidine-2-carboxamide
(2S,4R)-1-[(2,5-dimethylphenyl)methyl]-N-(1,1-dioxo-1λ6-thiolan-3-yl)-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
methyl (2S,4R)-4-[2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)acetamido]-1-[(3-fluorophenyl)methyl]pyrrolidine-2-carboxylate
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-amino-1-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethan-1-one