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4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-(3-phenylpropyl)benzamide
3-[4-(furan-2-carbonyl)-1,4-diazepane-1-carbonyl]-5-methyl-1H-indazole
6-{[4-(2-ethoxyphenyl)piperazin-1-yl]methyl}-2-oxo-N-[1-(thiophen-2-yl)ethyl]-1,2-dihydropyridine-3-carboxamide
N-ethyl-4-(4-{[2-(4-fluorophenyl)azetidin-1-yl]methyl}-1H-1,2,3-triazol-1-yl)piperidine-1-carboxamide
1-[(3-fluorophenyl)methyl]-4-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperazine
N-[2-(propan-2-yl)phenyl]-N'-[1-(pyrazin-2-yl)propan-2-yl]butanediamide
(1S,6R)-3-(3,5-difluoropyridine-2-carbonyl)-3,9-diazabicyclo[4.2.1]nonane
1-(benzylsulfamoyl)piperidine-2-carboxamide
8-(2,3-dihydro-1-benzofuran-5-carbonyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-ethyl-9-[(1-methyl-1H-imidazol-2-yl)methyl]-4-phenyl-2,9-diazaspiro[5.5]undecane
1,5-dimethyl-4-{[4-(piperidine-1-carbonyl)piperidin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
5-(2-phenylphenyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-(3,4-difluorophenoxymethyl)-N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-1,2-oxazole-3-carboxamide
3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-[(3-chlorophenyl)methyl]-N-propylpropanamide
4-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-methyl-6-(propan-2-yl)pyrimidine
1-cyclohexyl-N-[2-(3,4-dimethoxyphenyl)ethyl]-4-oxo-5-(pyrrolidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
5-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-(2-methoxyethyl)pyridin-2-amine
1-{6-[3-(3-ethylphenoxy)azetidin-1-yl]pyridin-2-yl}ethan-1-ol
N-[(5-methyl-2-{3-[3-(pyridin-3-yl)propanamido]phenyl}-1,3-oxazol-4-yl)methyl]-2-(methylsulfanyl)-1,3-thiazole-4-carboxamide
N-[(1-cyclopentylpiperidin-3-yl)methyl]-4,4,4-trifluoro-N-[2-(piperidin-1-yl)ethyl]butanamide
(2S,4R)-N-(2-methyl-1,3-benzothiazol-5-yl)-1-{[4-(methylsulfanyl)phenyl]methyl}-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carboxamide
N-[2-(5-benzyl-4-phenyl-1H-imidazol-1-yl)ethyl]-N-methylmethanesulfonamide
1-cyclopropanecarbonyl-3-[2-(2,4-difluorophenyl)ethyl]piperidine
4-[2-({1-[2-(dimethylamino)-6-ethylpyrimidin-4-yl]piperidin-4-yl}amino)ethyl]phenol
2-{[(4S,4aS,8aR)-4-hydroxy-4-phenyl-decahydroquinolin-1-yl]methyl}benzoic acid
1-[benzyl(methyl)amino]-3-(2-methoxy-5-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}phenoxy)propan-2-ol
7-(2-methoxyethyl)-2-[4-(methylamino)-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl]-2,7-diazaspiro[4.5]decan-6-one
2-[(5-methylpyrazin-2-yl)methyl]-9-[3-(1H-pyrazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
5-[3-(dimethylamino)pyrazin-2-yl]thiophene-2-carboxylic acid
N,4,6-trimethyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-2-oxo-2H-pyran-5-carboxamide
N-(3-carbamoyl-4-fluorophenyl)-8-methyl-9-oxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
2-(2H-1,2,3-benzotriazol-2-yl)-N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)acetamide
4-{2-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]phenyl}morpholine
1-benzyl-5-methanesulfonamido-2-methyl-N-[2-(thiophen-2-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
3-{1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidine-3-carbonyl}pyridine
({4-[1-(1-tert-butyl-1H-pyrrole-3-carbonyl)piperidin-2-yl]phenyl}methyl)dimethylamine
9-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
3-amino-N-({1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}methyl)propanamide
2-[4-(cyclohexylmethyl)-1-(2-phenylethyl)piperazin-2-yl]ethan-1-ol
3-(3-fluoro-4-phenylbenzoyl)-1-(1H-pyrazol-3-ylmethyl)piperidine
1-(2-chlorophenyl)-4-(2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}acetyl)piperazin-2-one
1-[3-({[2-methyl-1-(2-methylpropyl)-1H-indol-3-yl]methyl}amino)propyl]pyrrolidin-2-one
N-(2H-1,3-benzodioxol-5-yl)-4-[2-(methylsulfanyl)acetyl]morpholine-2-carboxamide
(1R,6S)-9-methyl-N-(1-phenyl-1H-pyrazol-5-yl)-3,9-diazabicyclo[4.2.1]nonane-3-carboxamide
N-ethyl-2,2-dimethyl-N-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)oxan-4-amine
4-(2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)piperazin-2-one
2-[4-(piperazin-1-yl)phenyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
8-(oxan-2-ylmethyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
N-[(3R,4S)-4-cyclopropyl-1-(oxane-4-carbonyl)pyrrolidin-3-yl]-2,5,6-trimethylpyrimidin-4-amine