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9-(4-chlorobenzoyl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-(2-methoxyphenoxymethyl)-N-(1-methyl-2-oxopyrrolidin-3-yl)-1H-pyrazole-3-carboxamide
1-methyl-4-[3-(piperidine-1-carbonyl)pyridin-2-yl]piperazine-2-carboxylic acid
1-(2,3-dimethoxybenzoyl)-4-(pyrimidin-2-yl)piperazine-2-carboxylic acid
2-{4-[(4-chlorophenyl)methyl]piperazine-1-carbonyl}-5-methoxy-4H-pyran-4-one
2-{8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-ethyl-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl}acetamide
[1-(2,6-dimethylpyridine-4-carbonyl)-3-(2-methoxyethyl)piperidin-3-yl]methanol
7-chloro-4-[(3,4-dimethoxyphenyl)methyl]-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-{1-[2-(4-methoxy-2,5-dimethylphenyl)-1H-imidazol-1-yl]ethyl}-2-methylpyridine
1-[1'-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
7-(cyclopropylmethyl)-2-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-2,7-diazaspiro[4.5]decane
2-[3-(hydroxymethyl)-3-propylpiperidine-1-carbonyl]-6-methyl-4H-pyran-4-one
{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}[(5-fluoro-1H-indol-2-yl)methyl]methylamine
({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)[(5-phenyl-1H-pyrazol-3-yl)methyl]amine
1-[3-(3-chlorophenyl)pyrrolidin-1-yl]-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propan-1-one
N-[3-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)-5-methylthiophen-2-yl]-2,2-dimethylpropanamide
N-[(5-chlorothiophen-2-yl)methyl]-6-(morpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
3-(1H-1,2,3-benzotriazol-1-yl)-1-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]propan-1-one
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
1-(3,5-dimethoxyphenyl)-2-{[6-(propan-2-yl)pyrimidin-4-yl]amino}ethan-1-ol
4,4-difluoro-1-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperidine
2-(4-{2-methyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}piperidin-1-yl)acetamide
(2S,4R)-4-amino-N,N-diethyl-1-(oxane-4-carbonyl)pyrrolidine-2-carboxamide
5-cyclopropanecarbonyl-1'-(5-ethyl-1,3-oxazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-[(2-fluorophenyl)methyl]benzamide
methyl 4-({2-[(3-fluorophenyl)methyl]morpholin-4-yl}methyl)benzoate
methyl 8-[2-(dimethylamino)benzoyl]-1-methoxy-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
N-[(3-chlorophenyl)methyl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(2S,4R)-4-amino-1-(azepane-1-sulfonyl)-N,N-diethylpyrrolidine-2-carboxamide
9-(1-ethyl-1H-pyrazole-3-carbonyl)-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-(1-hydroxybutan-2-yl)-N-(pyridin-2-ylmethyl)-2-(pyridin-3-yl)pyrimidine-5-carboxamide
[(3R,4R)-1-[4-(dimethylamino)benzoyl]-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
3-[4-(pyridazine-3-carbonyl)piperazin-1-yl]-1-azabicyclo[2.2.2]octane
5-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane-1-carbonyl]-N,4-dimethyl-1,3-thiazol-2-amine
1-methyl-N-[(4-methylpyridin-2-yl)methyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
1-(2-methylpropyl)-4-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
1-[(4-chloro-3-fluorophenyl)methyl]-4-[4-(piperidine-1-carbonyl)phenoxy]piperidine
4-[(4-fluorophenyl)methyl]-1-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-3-(propan-2-yl)-1,4-diazepan-5-one
8-(5-methyl-2-phenylfuran-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
1-methyl-4-[(4-methyl-1H-imidazol-2-yl)methyl]-2-phenylpiperazine
5-(2-chlorophenyl)-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]furan-2-carboxamide
1'-(2,4-dimethylpyrimidine-5-carbonyl)-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-[(5-propylfuran-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-[(1-ethyl-1H-imidazol-5-yl)methyl]-2-[4-(methylsulfanyl)phenyl]-1H-imidazole
4-{[5-(2,5-dimethylfuran-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}piperazin-2-one
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
2-{[3-(4-methyl-1H-pyrazol-1-yl)propyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
5-methyl-N-[(6-methylpyridin-2-yl)methyl]-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-2-{[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)amino}acetic acid
3-fluoro-4-methoxy-N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]benzamide