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N-(1-hydroxybutan-2-yl)-2-(pyridin-4-ylsulfanyl)-N-(thiophen-3-ylmethyl)acetamide
N-[cyclopropyl(pyridin-2-yl)methyl]-N,2,8-trimethylquinoline-3-carboxamide
3-cyclopropyl-N-(4-methyl-1,3-thiazol-2-yl)-1H-1,2,4-triazole-5-carboxamide
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-cyclopentylethan-1-one
N-[(3R,4R)-3-hydroxy-1-[2-(4-methylphenoxy)acetyl]piperidin-4-yl]pyrazine-2-carboxamide
3-(pyridin-3-yl)-1-{3-[1-(pyrimidin-2-yl)piperidin-4-yl]pyrrolidin-1-yl}propan-1-one
1-(2,3-dihydro-1H-inden-2-yl)-N-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-3-amine
2-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-2-oxoethyl}-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
N-({5-[(cyclohexylmethyl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}methyl)-1-[(1S,4R)-7,7-dimethyl-2-oxobicyclo[2.2.1]heptan-1-yl]methanesulfonamide
3-[2-benzyl-5-oxo-4-(3-phenylphenyl)piperazin-1-yl]-N-methylpropanamide
1-[4-(1-{[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-2-phenylethyl)piperidin-1-yl]-2-(pyrimidin-2-ylsulfanyl)ethan-1-one
2-{[(1-hydroxybutan-2-yl)(thiophen-3-ylmethyl)amino]methyl}benzoic acid
2-methyl-N-[4-(morpholin-4-yl)butan-2-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-hydroxy-1-[4-(2-methoxyphenoxy)piperidin-1-yl]ethan-1-one
(3aS,6aS)-2-(3-cyanopyridin-2-yl)-5-(dimethylcarbamoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-butyl-4-[2-(2,3-dihydro-1H-isoindol-2-yl)-2-oxo-1-phenylethyl]piperazine-2,3-dione
4-(3-methoxypropyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[2-(4-methoxyphenoxy)ethyl]-3-methyl-1,2-dihydroquinoxalin-2-one
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-[(2,3,4-trifluorophenyl)methyl]pyrrolidin-3-yl]methanol
2-[4-(4-cyclopentylpiperazine-1-carbonyl)-5-methyl-1H-pyrazol-1-yl]-4-(2-methoxyphenyl)pyrimidine
8-[(4-carboxyphenyl)carbamoyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-[(3R,4S)-3-amino-4-(3-methoxyphenyl)pyrrolidin-1-yl]-3-(2,3-dihydro-1H-isoindol-2-yl)propan-1-one
8-(2,5-dimethoxybenzenesulfonyl)-5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine
2-{1-[(5-methyl-1,2-oxazol-3-yl)methyl]-4-phenyl-1H-imidazol-5-yl}-1-(prop-2-en-1-yl)-1H-1,3-benzodiazole
1-(3-methylpyridin-4-yl)-4-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}-1,4-diazepane
4-methyl-5-[4-(pyrrolidine-1-sulfonyl)-1,4-diazepane-1-carbonyl]pyrimidin-2-amine
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}(2-methylpropyl)(pyridin-4-ylmethyl)amine
N-(2H-1,3-benzodioxol-5-yl)-1-{[4-chloro-2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperidin-3-amine
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(furan-2-ylmethyl)-N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}propanamide
2-{1-[3-(4H-1,2,4-triazol-4-yl)phenyl]-1H-pyrazol-3-yl}pyrazine
5-({[(3-{2-[4-(3-fluorobenzenesulfonyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)amino}methyl)pyrrolidin-2-one
methyl[(1-{[1-(5-methyl-1,3-benzoxazol-2-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]amine
2-benzyl-4-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1,3-thiazole
2-{1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-N-methylformamido}-2-(pyridin-3-yl)acetic acid
2-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-[(4,5-dimethyl-1H-imidazol-1-yl)methyl]-1H-1,2,4-triazol-3-yl]acetamide
2-[2-methyl-4-oxo-1-(3-phenylpropyl)-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
3-methanesulfonyl-N-[(3R,4S)-1-(6-methylpyridazin-3-yl)-4-propylpyrrolidin-3-yl]propanamide
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-2-methyl-3-[(pyridin-2-ylmethyl)amino]benzamide
2-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepane-1-carbonyl}benzonitrile
7-(4-chloro-1H-pyrazole-3-carbonyl)-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
6-(propan-2-yl)-N4-[3-(1H-1,2,3-triazol-1-yl)propyl]pyrimidine-2,4-diamine
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]acetamide
5-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-3,4-dihydropyrimidin-4-one
(3R,4R)-1-[2-(3-methoxyphenoxy)ethyl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
4-[4-(cyclopentylamino)piperidin-1-yl]-N-(1-phenylethyl)benzamide
5-({methyl[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amino}methyl)pyrimidin-2-amine
1-{2-[(2,4-dimethylphenyl)carbamoyl]acetyl}piperidine-3-carboxamide
5-[methyl(1,3-thiazol-2-ylmethyl)amino]-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
(4S)-3,3,4-trimethyl-1-{[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-ol
7-[1-(4-methoxyphenyl)piperidin-4-yl]-2-oxa-7-azaspiro[4.5]decane