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N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-(1-methylpiperidin-2-yl)acetamide
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}furan-3-carboxamide
2-(pyridin-3-yl)-1-[3-(pyrimidin-4-yl)piperidin-1-yl]ethan-1-one
2-{5-[(2S)-1-methanesulfonylpyrrolidin-2-yl]-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl}acetic acid
methyl (2S,4S)-1-methyl-4-[2-(4-methyl-2-oxo-1,2-dihydroquinolin-1-yl)acetamido]pyrrolidine-2-carboxylate
N-({1-[ethyl(methyl)amino]cyclohexyl}methyl)-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
[1-(5-methylpyrazine-2-carbonyl)-3-(2-phenylethyl)piperidin-3-yl]methanol
N-methyl-N-[2-({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]methanesulfonamide
6-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}-N,N-dimethylpyridine-3-carboxamide
4-[3-(3-methoxyphenoxy)propyl]-N,N-dimethylbenzamide
4-methyl-N-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
N-[(3,4-dimethoxyphenyl)methyl]-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(1R,5R)-6-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-(4-chlorophenyl)-5-[4-hydroxy-1-(2-methylpropyl)piperidin-4-yl]-1-benzofuran-2-carboxamide
N-[(3S,4R)-4-methoxyoxolan-3-yl]-5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carboxamide
(3aS,6aS)-2-methyl-5-{[5-(1,2-oxazol-5-yl)thiophen-2-yl]sulfonyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(1-{[(6-ethylpyrimidin-4-yl)(methyl)amino]methyl}cyclopentyl)methanol
methyl({[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl})[2-(pyridin-4-yl)ethyl]amine
4-[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-1,4-oxazepane
(2S,4S)-4-amino-N-ethyl-1-[3-(4-methylphenyl)benzoyl]pyrrolidine-2-carboxamide
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
2-ethyl-5-(1-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1H-imidazol-2-yl)-4-methyl-1H-imidazole
methyl 3-[4-({6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)-1H-pyrazol-1-yl]propanoate
N-cyclohexyl-N-[(3-methylphenyl)methyl]-1-(propan-2-yl)-1H-pyrazole-3-carboxamide
2-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
2-(3-methoxyphenyl)-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
dimethyl({4-methyl-5-[1-(1-methyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
N-[4-(dimethylamino)phenyl]-2-(3-methoxypropyl)piperidine-1-carboxamide
6-(3-chlorophenyl)-N-cyclohexyl-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
3-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]propanamide
(3aR,6aR)-2-(cyclobutylmethyl)-5-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[6-(6-{[2-(dimethylamino)ethyl]amino}-1H-pyrrolo[2,3-b]pyridin-4-yl)pyridin-3-yl]ethan-1-one
4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-1-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}piperidine
9-[2-(benzyloxy)acetyl]-2-(cyclopropylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(3-hydroxypropyl)-9-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-2,9-diazaspiro[5.5]undecan-3-one
ethyl 1-[(3-methoxyphenyl)methyl]-5-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-pyrazol-3-yl]phenyl}thiophene-2-carbonitrile
1-methanesulfonyl-4-{2-methylimidazo[1,2-a]pyridine-6-carbonyl}piperazine
2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]benzamide
2-(2H-1,2,3-benzotriazol-2-yl)-N-[(1-cyclopentylpiperidin-4-yl)methyl]-N-(oxolan-2-ylmethyl)acetamide
4-[(2-oxoazepan-3-yl)sulfamoyl]-N-(prop-2-en-1-yl)benzamide
2-ethyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}pyrimidine-5-carboxamide
N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-2-(4-oxo-3,4-dihydro-1,2,3-benzotriazin-3-yl)acetamide
1-ethyl-N-[(1-phenylcyclohexyl)methyl]-1H-pyrazole-5-carboxamide
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-5-methoxyfuran-2-carboxamide
1-(1-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)-3-methylbutan-1-ol
2-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]thiophene-3-sulfonamide
1-[4-(diphenylmethyl)piperazin-1-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-4-[3-(trifluoromethyl)phenyl]piperazine
6-oxo-1-(2-phenylethyl)-N-propyl-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide